GT201000099A - Productos quimioterapéuticos cristalinos - Google Patents

Productos quimioterapéuticos cristalinos

Info

Publication number
GT201000099A
GT201000099A GT201000099A GT201000099A GT201000099A GT 201000099 A GT201000099 A GT 201000099A GT 201000099 A GT201000099 A GT 201000099A GT 201000099 A GT201000099 A GT 201000099A GT 201000099 A GT201000099 A GT 201000099A
Authority
GT
Guatemala
Prior art keywords
crystal
chemotherapeutic products
chemotherapeutic
products
methylpenyl
Prior art date
Application number
GT201000099A
Other languages
English (en)
Inventor
Thomas B Borchardt
Alexander Chu-Kung
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT201000099A publication Critical patent/GT201000099A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

LA PRESENTE INVENCIÓN SE REFIERE A LA FORMA CRISTALINA 2 DE N-[4-(3-AMINO-1H-INDAZOL-4-IL) FENIL]-N´- (2-FLUORO -5-METILFENIL)UREA(ABT-869) QUE PERTENECE A UNA FAMILIA DE PROTEÍNA TIROSINA QUINASA (PTK) QUE CATALIZAN LA FOSFORILACIÓN DE RESIDUOS ESPECÍFICOS DE TIROSINA EN PROTEÍNAS POR LO QUE SON DE UTILIDAD EN TRASTORNOS O ENFERMEDADES PROLIFERATIVAS MALIGNAS RESULTANTES DE LA ACTIVACIÓN INAPROPIADA DEL SISTEMA INMUNE.
GT201000099A 2007-10-19 2010-04-16 Productos quimioterapéuticos cristalinos GT201000099A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US98126507P 2007-10-19 2007-10-19

Publications (1)

Publication Number Publication Date
GT201000099A true GT201000099A (es) 2012-03-26

Family

ID=40174735

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201000099A GT201000099A (es) 2007-10-19 2010-04-16 Productos quimioterapéuticos cristalinos

Country Status (19)

Country Link
US (1) US7772404B2 (es)
EP (1) EP2195299A1 (es)
JP (1) JP2011500708A (es)
KR (1) KR20100084665A (es)
CN (1) CN101827825B (es)
AU (1) AU2008312534A1 (es)
BR (1) BRPI0818337A2 (es)
CA (1) CA2699356A1 (es)
CO (1) CO6270221A2 (es)
CR (1) CR11444A (es)
DO (1) DOP2010000111A (es)
EC (1) ECSP10010175A (es)
GT (1) GT201000099A (es)
MX (1) MX2010004287A (es)
PA (1) PA8800401A1 (es)
RU (1) RU2010119920A (es)
UA (1) UA99490C2 (es)
WO (1) WO2009052231A1 (es)
ZA (1) ZA201002094B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013022801A1 (en) 2011-08-05 2013-02-14 Forsight Vision4, Inc. Small molecule delivery with implantable therapeutic device
CA2818612C (en) 2010-11-19 2020-12-29 Forsight Vision4, Inc. Therapeutic agent formulations for implanted devices
CA2905496A1 (en) 2013-03-14 2014-09-25 Forsight Vision4, Inc. Systems for sustained intraocular delivery of low solubility compounds from a port delivery system implant
WO2016022750A1 (en) 2014-08-08 2016-02-11 Forsight Vision4, Inc. Stable and soluble formulations of receptor tyrosine kinase inhibitors, and methods of preparation thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2346538T3 (es) * 2003-05-22 2010-10-18 Abbott Laboratories Inhibidores de quinasa de tipo indazol, benzisoxazol y benzisotiazol.
US7297709B2 (en) * 2003-05-22 2007-11-20 Abbott Laboratories Indazole, benzisoxazole, and benzisothiazole kinase inhibitors
US20100105031A1 (en) * 2005-08-01 2010-04-29 Esai R & D Management Co., Ltd. Method for prediction of the efficacy of vascularization inhibitor
EP1925676A4 (en) * 2005-08-02 2010-11-10 Eisai R&D Man Co Ltd TEST METHOD FOR THE EFFECT OF A VASCULARIZATION INHIBITOR
EP1962803A1 (en) * 2005-12-23 2008-09-03 Alcon, Inc. PHARMACEUTICAL FORMULATION FOR DELIVERY OF RECEPTOR TYROSINE KINASE INHIBITING (RTKi) COMPOUNDS TO THE EYE
AU2007316558A1 (en) * 2006-11-09 2008-05-15 Abbott Gmbh & Co. Kg Pharmaceutical dosage form for oral administration of tyrosine kinase inhibitor

Also Published As

Publication number Publication date
ZA201002094B (en) 2011-11-30
BRPI0818337A2 (pt) 2017-05-23
ECSP10010175A (es) 2010-06-29
CN101827825A (zh) 2010-09-08
WO2009052231A1 (en) 2009-04-23
US7772404B2 (en) 2010-08-10
CA2699356A1 (en) 2009-04-23
JP2011500708A (ja) 2011-01-06
CR11444A (es) 2010-10-05
CN101827825B (zh) 2012-11-21
UA99490C2 (en) 2012-08-27
CO6270221A2 (es) 2011-04-20
AU2008312534A1 (en) 2009-04-23
DOP2010000111A (es) 2010-07-15
PA8800401A1 (es) 2009-05-15
MX2010004287A (es) 2010-04-30
RU2010119920A (ru) 2011-11-27
EP2195299A1 (en) 2010-06-16
US20090124816A1 (en) 2009-05-14
KR20100084665A (ko) 2010-07-27

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