GT200800226A - Derivados de acido benzoazepin-oxi-acetico como agonistas de receptores activados por proliferador de peroxisoma delta usados para incrementar la lipoproteina de alta densidad-colesterol, reducir la lipoproteina de baja densidad-colesterol y reducir - Google Patents

Derivados de acido benzoazepin-oxi-acetico como agonistas de receptores activados por proliferador de peroxisoma delta usados para incrementar la lipoproteina de alta densidad-colesterol, reducir la lipoproteina de baja densidad-colesterol y reducir

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Publication number
GT200800226A
GT200800226A GT200800226A GT200800226A GT200800226A GT 200800226 A GT200800226 A GT 200800226A GT 200800226 A GT200800226 A GT 200800226A GT 200800226 A GT200800226 A GT 200800226A GT 200800226 A GT200800226 A GT 200800226A
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GT
Guatemala
Prior art keywords
colesterol
lipoprotein
redesteru
peroxisoma
benzoazepin
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GT200800226A
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English (en)
Inventor
Gee-Hong Kuo
Yan Zhang
Lan Shen
Songfeng Lu
Keith T Demarest
Patricia Pelton
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38610435&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT200800226(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
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Publication of GT200800226A publication Critical patent/GT200800226A/es

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    • C07D233/06—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms
    • C07D233/08—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms with alkyl radicals, containing more than four carbon atoms, directly attached to ring carbon atoms
    • C07D233/12—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms with alkyl radicals, containing more than four carbon atoms, directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
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    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
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  • Other In-Based Heterocyclic Compounds (AREA)
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

LA INVENCIÓN ESTÁ DIRIGIDA A COMPUESTOS DE LA FÓRMULA (I) ÚTILES COMO AGONISTAS DE PPAR; TAMBIÉN SE DESCRIBEN COMPOSICIONES FARMACÉUTICAS Y MÉTODOS PARA TRATAR UNA O MÁS CONDICIONES INCLUYENDO, PERO SIN LIMITARSE A, DIABETES, NEFROPATÍA, NEUROPATÍA, RETINOPATÍA, SÍNDROME DE OVARIO POLICÍSTICO, HIPERTENSIÓN, ISQUEMIA, ACCIDENTE VASCULAR CEREBRAL, TRASTORNO INTESTINAL METABÓLICO X, HIPER-LDL-COLESTEROLEMIA, DISLIPIDEMIA (INCLUYENDO HIPERTRIGLICERIDEMIA, HIPERCOLESTEROLEMIA, HIPERLIPIDEMIA MIXTA, E HIPO-HDL-COLESTEROLEMIA), ATEROSCLEROSIS, OBESIDAD Y TRASTORNOS RELACIONADOS CON EL METABOLISMO DE LÍPIDOS Y COMPLICACIONES DE HOMEOSTASIS DE ENERGÍA DE LOS MISMOS, USANDO COMPUESTOS DE LA INVENCIÓN. T2008
GT200800226A 2006-04-18 2008-10-21 Derivados de acido benzoazepin-oxi-acetico como agonistas de receptores activados por proliferador de peroxisoma delta usados para incrementar la lipoproteina de alta densidad-colesterol, reducir la lipoproteina de baja densidad-colesterol y reducir GT200800226A (es)

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US79300106P 2006-04-18 2006-04-18

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GT200800226A true GT200800226A (es) 2009-03-13

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US (2) US7678786B2 (es)
EP (1) EP2010289B1 (es)
JP (1) JP5232771B2 (es)
KR (1) KR101472370B1 (es)
CN (1) CN101479008B (es)
AR (1) AR060489A1 (es)
AT (1) ATE535282T1 (es)
AU (1) AU2007237928B2 (es)
BR (1) BRPI0711695A2 (es)
CA (1) CA2649700C (es)
CO (1) CO6160296A2 (es)
CR (1) CR10447A (es)
EA (1) EA016583B1 (es)
EC (1) ECSP088841A (es)
ES (1) ES2375754T3 (es)
GT (1) GT200800226A (es)
HK (1) HK1124797A1 (es)
HN (1) HN2008001559A (es)
IL (1) IL194850A (es)
JO (1) JO3444B1 (es)
MX (1) MX2008013534A (es)
MY (1) MY144637A (es)
NO (1) NO344334B1 (es)
NZ (1) NZ571998A (es)
PE (1) PE20080188A1 (es)
TW (1) TWI404712B (es)
UA (1) UA96150C2 (es)
UY (1) UY30288A1 (es)
WO (1) WO2007121432A2 (es)
ZA (1) ZA200809790B (es)

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