GR1007629B - Φαρμακευτικο σκευασμα ελεγχομενης αποδεσμευσης ενος μη εργολινικου αγωνιστη της ντοπαμινης - Google Patents

Φαρμακευτικο σκευασμα ελεγχομενης αποδεσμευσης ενος μη εργολινικου αγωνιστη της ντοπαμινης

Info

Publication number
GR1007629B
GR1007629B GR20110100407A GR20110100407A GR1007629B GR 1007629 B GR1007629 B GR 1007629B GR 20110100407 A GR20110100407 A GR 20110100407A GR 20110100407 A GR20110100407 A GR 20110100407A GR 1007629 B GR1007629 B GR 1007629B
Authority
GR
Greece
Prior art keywords
release pharmaceutical
controlled
pharmaceutical formulation
dopamine agonist
ergoline
Prior art date
Application number
GR20110100407A
Other languages
English (en)
Inventor
Ευθυμιος Χρηστου Κουτρης
Ευαγγελος Ανδρεα Καραβας
Βικυ Χρηστου Σαμαρα
Δημητριος Νικολαου Μπικιαρης
Αναστασια Λεωνιδα Καλασκανη
Γεωργιος Θεμιστοκλη Γκοτζαμανης
Original Assignee
Φαρματεν Αβεε,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Φαρματεν Αβεε, filed Critical Φαρματεν Αβεε,
Priority to GR20110100407A priority Critical patent/GR1007629B/el
Publication of GR1007629B publication Critical patent/GR1007629B/el
Priority to PCT/EP2012/002831 priority patent/WO2013007360A1/en
Priority to EP12751249.9A priority patent/EP2731592A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/4045Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Η παρούσα εφεύρεση αφορά μια στερεά φαρμακευτική σύνθεση ελεγχόμενης αποδέσμευσης για από του στόματος χορήγηση που περιέχει μια θεραπευτικώς αποτελεσματική ποσότητα ενός μη εργολινικού αγωνιστή της ντοπαμίνης ή ένα φαρμακευτικά αποδεκτό άλας, παράγωγο ή πολύμορφο αυτής, η οποία σύνθεση χαρακτηρίζεται από το ότι περιέχει μια αποτελεσματική ποσότητα τουλάχιστον ενός εκδόχου που επιλέγεται από έναν μη διογκούμενο παράγοντα, έναν παράγοντα που δημιουργεί γέλη, και μια αμφιφιλική ουσία. Επίσης παρέχεται μέθοδος για την παρασκευή της εν λόγω σύνθεσης.
GR20110100407A 2011-07-13 2011-07-13 Φαρμακευτικο σκευασμα ελεγχομενης αποδεσμευσης ενος μη εργολινικου αγωνιστη της ντοπαμινης GR1007629B (el)

Priority Applications (3)

Application Number Priority Date Filing Date Title
GR20110100407A GR1007629B (el) 2011-07-13 2011-07-13 Φαρμακευτικο σκευασμα ελεγχομενης αποδεσμευσης ενος μη εργολινικου αγωνιστη της ντοπαμινης
PCT/EP2012/002831 WO2013007360A1 (en) 2011-07-13 2012-07-05 Controlled release pharmaceutical composition of non-ergoline dopamine agonist
EP12751249.9A EP2731592A1 (en) 2011-07-13 2012-07-05 Controlled release pharmaceutical composition of non-ergoline dopamine agonist

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GR20110100407A GR1007629B (el) 2011-07-13 2011-07-13 Φαρμακευτικο σκευασμα ελεγχομενης αποδεσμευσης ενος μη εργολινικου αγωνιστη της ντοπαμινης

Publications (1)

Publication Number Publication Date
GR1007629B true GR1007629B (el) 2012-06-29

Family

ID=45930912

Family Applications (1)

Application Number Title Priority Date Filing Date
GR20110100407A GR1007629B (el) 2011-07-13 2011-07-13 Φαρμακευτικο σκευασμα ελεγχομενης αποδεσμευσης ενος μη εργολινικου αγωνιστη της ντοπαμινης

Country Status (3)

Country Link
EP (1) EP2731592A1 (el)
GR (1) GR1007629B (el)
WO (1) WO2013007360A1 (el)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070059365A1 (en) * 2003-08-22 2007-03-15 Pollock Peta E Novel formulation of ropinirole
WO2009023761A2 (en) * 2007-08-14 2009-02-19 Dr. Reddy's Laboratories Ltd. Pharmaceutical compositions comprising ropinirole
WO2010012482A1 (en) * 2008-08-01 2010-02-04 Krka, Tovarna Zdravil, D.D., Novo Mesto Ropinirole composition

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR030557A1 (es) 2000-04-14 2003-08-27 Jagotec Ag Una tableta en multicapa de liberacion controlada y metodo de tratamiento

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070059365A1 (en) * 2003-08-22 2007-03-15 Pollock Peta E Novel formulation of ropinirole
WO2009023761A2 (en) * 2007-08-14 2009-02-19 Dr. Reddy's Laboratories Ltd. Pharmaceutical compositions comprising ropinirole
WO2010012482A1 (en) * 2008-08-01 2010-02-04 Krka, Tovarna Zdravil, D.D., Novo Mesto Ropinirole composition

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
R. B. NILESH ET AL: "Formulation and Evaluation of Transdermal patches of Ropinirole HCl", RESEARCH JOURNAL OF PHARMACEUTICAL, BIOLOGICAL AND CHEMICAL SCIENCES, vol. 2, no. 1, 1 March 2011 (2011-03-01), pages 138 - 148, XP055025644 *
SRAVANTHI ANAMPALLY ET AL: "Development of ropinirole (free base) transdermal patch using blends of hydroxypropyl methylcellulose/ Eudragits and its in vitro/ in vivo characterization", ASIAN JOURNAL OF PHARMACEUTICAL RESEARCH AND HEALTH CARE, vol. 3, no. 4, 1 July 2011 (2011-07-01), pages 89 - 98, XP055025634 *

Also Published As

Publication number Publication date
WO2013007360A1 (en) 2013-01-17
EP2731592A1 (en) 2014-05-21

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PG Patent granted

Effective date: 20120713

ML Lapse due to non-payment of fees

Effective date: 20170207