GB9326332D0 - Indole derivatives - Google Patents

Indole derivatives

Info

Publication number: GB9326332D0
Authority: GB; United Kingdom
Prior art keywords: indole derivatives; indole; derivatives
Prior art date: 1993-12-23
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Pending

Application number

GB939326332A

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

KARO BIO

Original Assignee

KARO BIO

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-12-23

Filing date

1993-12-23

Publication date

1994-02-23

1993-12-23 Application filed by KARO BIO filed Critical KARO BIO

1993-12-23 Priority to GB939326332A priority Critical patent/GB9326332D0/en

1994-02-23 Publication of GB9326332D0 publication Critical patent/GB9326332D0/en

1994-12-23 Priority to CA002187296A priority patent/CA2187296A1/en

1994-12-23 Priority to PCT/EP1994/004250 priority patent/WO1995017383A1/en

1994-12-23 Priority to JP7517189A priority patent/JPH09510689A/en

1994-12-23 Priority to EP95904514A priority patent/EP0736008A1/en

1994-12-23 Priority to AU13169/95A priority patent/AU1316995A/en

Status Pending legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Hematology (AREA)
Diabetes (AREA)
Indole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

GB939326332A 1993-12-23 1993-12-23 Indole derivatives Pending GB9326332D0 (en)

Priority Applications (6)

Application Number	Priority Date	Filing Date	Title
GB939326332A GB9326332D0 (en)	1993-12-23	1993-12-23	Indole derivatives
CA002187296A CA2187296A1 (en)	1993-12-23	1994-12-23	Indole derivatives as anti-estrogens
PCT/EP1994/004250 WO1995017383A1 (en)	1993-12-23	1994-12-23	Indole derivatives as anti-estrogens
JP7517189A JPH09510689A (en)	1993-12-23	1994-12-23	Indole derivatives as antiestrogens
EP95904514A EP0736008A1 (en)	1993-12-23	1994-12-23	Indole derivatives as anti-estrogens
AU13169/95A AU1316995A (en)	1993-12-23	1994-12-23	Indole derivatives as anti-estrogens

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB939326332A GB9326332D0 (en)	1993-12-23	1993-12-23	Indole derivatives

Publications (1)

Publication Number	Publication Date
GB9326332D0 true GB9326332D0 (en)	1994-02-23

Family

ID=10747121

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
GB939326332A Pending GB9326332D0 (en)	1993-12-23	1993-12-23	Indole derivatives

Country Status (6)

Country	Link
EP (1)	EP0736008A1 (en)
JP (1)	JPH09510689A (en)
AU (1)	AU1316995A (en)
CA (1)	CA2187296A1 (en)
GB (1)	GB9326332D0 (en)
WO (1)	WO1995017383A1 (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4426625A1 (en) *	1994-07-27	1996-03-14	Schering Ag	2-phenylindoles, processes for their preparation, pharmaceutical preparations containing them and their use in the manufacture of medicaments
US5985910A (en) *	1996-04-19	1999-11-16	American Home Products Corporation	3- [4- (2- Phenyl-Indole-1-ylmethyl) Phenyl]- Acrylamides as estrogenic agents
US5880137A (en) *	1996-04-19	1999-03-09	American Home Products Corporation	2-phenyl-1- 4-(amino-1-yl-alk-1-ynyl)-benzyl!-1H-indol-5-ols as estrogenic agents
US5998402A (en)	1996-04-19	1999-12-07	American Home Products Corporation	2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
DK0802183T3 (en) *	1996-04-19	2002-02-04	American Home Prod	estrogen Compounds
TW397821B (en) *	1996-04-19	2000-07-11	American Home Produits Corp	3-[4-(2-phenyl-indole-1-ylmethyl)-phenyl]-acrylamides and 2-phenyl-1-[4-(amino-1-yl-alk-1-ynyl)-benzyl]-1H-indol-5-ol as well as pharmaceutical compositions of estrogenic agents thereof
US5780497A (en) *	1996-04-19	1998-07-14	American Home Products Corporation	2-phenyl-1- 4-(amino-1-yl-alk-1-ynyl)-benzyl!-1H-indol-5-ols as estrogenic agents
US6005102A (en)	1997-10-15	1999-12-21	American Home Products Corporation	Aryloxy-alkyl-dialkylamines
EE200000225A (en)	1997-10-15	2001-06-15	American Home Products Corporation	Aryloxyalkyl dialkylamines, methods for their preparation and pharmaceutical composition
US6326392B1 (en)	1997-11-06	2001-12-04	American Home Products Corporation	Anti-estrogen plus progestin containing oral contraceptives
US6069153A (en) *	1998-05-12	2000-05-30	American Home Products Corporation	Indenoindoles and benzocarbazoles as estrogenic agents
ID26890A (en) *	1998-05-15	2001-02-15	American Home Prod	2-FENIL-1- (4- (2-AMINOETOKSI) -BENZIL) -INDOL IN THE COMBINATION WITH ESTROGEN
US6479535B1 (en)	1998-05-15	2002-11-12	Wyeth	2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole and estrogen formulations
US6380185B1 (en)	1999-03-04	2002-04-30	American Home Products Corporation	N-substituted benzoyl indoles as estrogenic agents
US6159959A (en) *	1999-05-06	2000-12-12	American Home Products Corporation	Combined estrogen and antiestrogen therapy
TWI287018B (en) *	1999-09-13	2007-09-21	Wyeth Corp	Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1H-indol-5-ols
US6380166B1 (en)	1999-09-13	2002-04-30	American Home Products Corporation	Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1H-indol-5-ols
MX2010004195A (en)	2007-10-16	2010-06-02	Repros Therapeutics Inc	Trans-clomiphene for metabolic syndrome.
WO2013130832A1 (en)	2012-02-29	2013-09-06	Repros Therapeutics Inc.	Combination therapy for treating androgen deficiency
WO2017081171A1 (en)	2015-11-10	2017-05-18	Paracrine Therapeutics Ab	Treatment of er-negative breast cancer with an pdgf-cc inhibitor and an anti estrogen
CN105859606B (en) *	2016-04-06	2019-01-29	沈阳药科大学	Indole derivatives and its preparation method and application containing piperazinyl
CN105732465B (en) *	2016-04-06	2019-01-29	沈阳药科大学	Phenyl-indoles compound and its preparation method and application
EP4223293A1 (en) *	2020-09-30	2023-08-09	Tokyo Metropolitan Geriatric Hospital and Institute of Gerontology	Pharmaceutical composition for treatment of prostate cancer or breast cancer

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3821148A1 (en) *	1988-06-23	1989-12-28	Erwin Von Dr Angerer	AMINO ALKYLINDOLE, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEREOF
US5395842A (en) *	1988-10-31	1995-03-07	Endorecherche Inc.	Anti-estrogenic compounds and compositions

1993
- 1993-12-23 GB GB939326332A patent/GB9326332D0/en active Pending
1994
- 1994-12-23 JP JP7517189A patent/JPH09510689A/en active Pending
- 1994-12-23 AU AU13169/95A patent/AU1316995A/en not_active Abandoned
- 1994-12-23 CA CA002187296A patent/CA2187296A1/en not_active Abandoned
- 1994-12-23 EP EP95904514A patent/EP0736008A1/en not_active Withdrawn
- 1994-12-23 WO PCT/EP1994/004250 patent/WO1995017383A1/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
EP0736008A1 (en)	1996-10-09
WO1995017383A1 (en)	1995-06-29
AU1316995A (en)	1995-07-10
JPH09510689A (en)	1997-10-28
CA2187296A1 (en)	1995-06-29

Publication	Publication Date	Title
HU9402983D0 (en)	1995-02-28	Indol derivatives
GB2266091B (en)	1995-08-09	Indole derivatives
ZA942383B (en)	1995-10-09	New indole derivatives
ZA941483B (en)	1994-11-11	Indole derivatives
ZA932440B (en)	1994-10-05	Indole derivatives
ZA947210B (en)	1996-03-18	Indole derivatives
GB9326332D0 (en)	1994-02-23	Indole derivatives
PL313969A1 (en)	1996-08-05	Indole derivatives
EP0512350A3 (en)	1992-12-16	Indole derivatives
ZA942805B (en)	1995-10-23	Indole derivatives
GB9116732D0 (en)	1991-09-18	Indole derivatives
GB9204024D0 (en)	1992-04-08	Indole derivatives
GB9302577D0 (en)	1993-03-24	Indole derivatives
GB9319299D0 (en)	1993-11-03	Indole derivatives
GB9309148D0 (en)	1993-06-16	Indole derivatives
GB9310092D0 (en)	1993-06-30	Indole derivatives
GB9307080D0 (en)	1993-05-26	Indole derivatives
GB9206056D0 (en)	1992-05-06	Indole derivatives
GB9218595D0 (en)	1992-10-14	Indole derivatives
GB9206794D0 (en)	1992-05-13	Indole derivatives
GB9206809D0 (en)	1992-05-13	Indole derivatives
IL121326A0 (en)	1998-01-04	Indole derivatives
GB9206810D0 (en)	1992-05-13	Indole derivatives
GB9206787D0 (en)	1992-05-13	Indole derivatives
GB9215961D0 (en)	1992-09-09	Indole derivatives