GB9301003D0 - Substituted pyrazoles,isoxazo-les and isothiazoles as neurotensin antagonists - Google Patents

Substituted pyrazoles,isoxazo-les and isothiazoles as neurotensin antagonists

Info

Publication number
GB9301003D0
GB9301003D0 GB939301003A GB9301003A GB9301003D0 GB 9301003 D0 GB9301003 D0 GB 9301003D0 GB 939301003 A GB939301003 A GB 939301003A GB 9301003 A GB9301003 A GB 9301003A GB 9301003 D0 GB9301003 D0 GB 9301003D0
Authority
GB
United Kingdom
Prior art keywords
isoxazo
isothiazoles
les
substituted pyrazoles
neurotensin antagonists
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
GB939301003A
Other versions
GB2263638A (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of GB9301003D0 publication Critical patent/GB9301003D0/en
Publication of GB2263638A publication Critical patent/GB2263638A/en
Withdrawn legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
GB9301003A 1992-01-28 1993-01-20 Substituted pyrazoles, isoxazoles and isothiazoles as neurotensin antagonists Withdrawn GB2263638A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US82712692A 1992-01-28 1992-01-28

Publications (2)

Publication Number Publication Date
GB9301003D0 true GB9301003D0 (en) 1993-03-10
GB2263638A GB2263638A (en) 1993-08-04

Family

ID=25248370

Family Applications (1)

Application Number Title Priority Date Filing Date
GB9301003A Withdrawn GB2263638A (en) 1992-01-28 1993-01-20 Substituted pyrazoles, isoxazoles and isothiazoles as neurotensin antagonists

Country Status (1)

Country Link
GB (1) GB2263638A (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5491172A (en) * 1993-05-14 1996-02-13 Warner-Lambert Company N-acyl sulfamic acid esters (or thioesters), N-acyl sulfonamides, and N-sulfonyl carbamic acid esters (or thioesters) as hypercholesterolemic agents
IL109431A (en) * 1993-05-14 2001-01-11 Warner Lambert Co Pharmaceutical compositions containing n-acyl sulfamic acid esters (or thioesters), n-acyl sulfonamides, and n-sulfonyl carbamic acid esters (or thioesters), for regulating plasma cholesterol concentration, and certain such novel compounds
FR2723317B1 (en) * 1994-08-04 1996-10-31 Sanofi Sa USE OF NEUROTENSIN ANTAGONISTS FOR THE PREPARATION OF DIURETIC DRUGS
SE9502219D0 (en) * 1995-06-19 1995-06-19 Astra Ab Novel medical use
US6297198B1 (en) 1996-05-14 2001-10-02 Syngenta Participations Ag Isoxazole derivatives and their use as herbicides
CA3121202A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9005354D0 (en) * 1990-03-09 1990-05-02 Glaxo Group Ltd Chemical compounds
JPH05505822A (en) * 1990-03-30 1993-08-26 メルク・エンド・カムパニー・インコーポレーテツド Pyrazoles, isoxazoles and isothiazole substituted products

Also Published As

Publication number Publication date
GB2263638A (en) 1993-08-04

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Legal Events

Date Code Title Description
WAP Application withdrawn, taken to be withdrawn or refused ** after publication under section 16(1)