GB1234058A - - Google Patents
Info
- Publication number
- GB1234058A GB1234058A GB1234058DA GB1234058A GB 1234058 A GB1234058 A GB 1234058A GB 1234058D A GB1234058D A GB 1234058DA GB 1234058 A GB1234058 A GB 1234058A
- Authority
- GB
- United Kingdom
- Prior art keywords
- group
- atom
- quaternary ammonium
- reaction
- general formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB4979868 | 1968-10-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
GB1234058A true GB1234058A (es) | 1971-06-03 |
Family
ID=10453571
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GB1234058D Expired GB1234058A (es) | 1968-10-21 | 1968-10-21 |
Country Status (4)
Country | Link |
---|---|
DE (1) | DE1804450A1 (es) |
FR (1) | FR1593614A (es) |
GB (1) | GB1234058A (es) |
NL (1) | NL6815409A (es) |
Cited By (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4182766A (en) * | 1977-09-19 | 1980-01-08 | Hoffmann-La Roche Inc. | Naphth[2,3-d]imidazoles |
WO1987005296A1 (en) * | 1986-03-07 | 1987-09-11 | Pfizer Inc. | 2-[(2-pyridyl)methylsulfinyl]thienoimidazoles and related compounds as antiulcer agents |
EP0254588A1 (en) * | 1986-07-25 | 1988-01-27 | Tokyo Tanabe Company Limited | Imidazo[4,5-b] pyridine compounds, process for preparing same and pharmaceutical compositions containing same |
US4738970A (en) * | 1984-12-18 | 1988-04-19 | Otsuka Pharmaceutical Co., Ltd. | Benzimidazolyl-thio-tetrahydroquinolines and anti-peptic ulcer compositions containing the same |
US4738974A (en) * | 1983-03-04 | 1988-04-19 | Aktiebolaget Hassle | Base addition salts of omeprazole |
US4758579A (en) * | 1984-06-16 | 1988-07-19 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Fluoroalkoxy substituted benzimidazoles useful as gastric acid secretion inhibitors |
US4791114A (en) * | 1986-01-20 | 1988-12-13 | 501 Laboratorios Del, Dr. Esteve | 2-Benzimidazolylalkylthio (or -sulfinyl or -sulfonyl) derivatives, their preparation and their application as medicinal products |
GB2161160B (en) * | 1984-07-06 | 1989-05-24 | Fisons Plc | Heterocyclic sulphinyl compounds |
US4873337A (en) * | 1985-07-31 | 1989-10-10 | The Upjohn Company | N-substituted derivatives of 2-(pyridylalkenesulfinyl) benzimidazoles as gastric antisecretory agents |
US5053417A (en) * | 1986-02-12 | 1991-10-01 | Tanabe Seiyaku Co., Ltd. | Imidazole derivatives and preparation thereof |
US5114955A (en) * | 1987-11-13 | 1992-05-19 | Hoechst Aketiengesellschaft | Substituted thienoimidazole derivatives |
US5389664A (en) * | 1992-07-08 | 1995-02-14 | Monsanto Company | Alleviating stomach ulcers in swine |
JP2679745B2 (ja) | 1989-06-29 | 1997-11-19 | 明治製菓株式会社 | アゾール誘導体及びそれらを有効成分とする抗潰瘍剤 |
US5703097A (en) * | 1994-02-28 | 1997-12-30 | Il-Yang Pharm. Co., Ltd. | 5-pyrrolyl-2-pyridylmethylsulfinyl benzimidazole derivatives |
US5859030A (en) * | 1994-06-10 | 1999-01-12 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Substituted arylalkylthioalkylthiopyridines for use in the control of helicobacter bacteria |
US6077541A (en) * | 1997-11-14 | 2000-06-20 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
US6174548B1 (en) | 1998-08-28 | 2001-01-16 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
US6733778B1 (en) | 1999-08-27 | 2004-05-11 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
EP3050565A1 (en) * | 2015-01-27 | 2016-08-03 | Ecole Polytechnique Fédérale de Lausanne (EPFL) | Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1259525B (de) * | 1961-11-21 | 1968-01-25 | Bauermann & Soehne G M B H W | Befestigungsvorrichtung fuer ein einstellbares Schutzdach an einer Sitz- bzw. Liegeschaukel |
SE418966B (sv) * | 1974-02-18 | 1981-07-06 | Haessle Ab | Analogiforfarande for framstellning av foreningar med magsyrasekretionsinhiberande verkan |
US4045564A (en) * | 1974-02-18 | 1977-08-30 | Ab Hassle | Benzimidazole derivatives useful as gastric acid secretion inhibitors |
SE416649B (sv) * | 1974-05-16 | 1981-01-26 | Haessle Ab | Forfarande for framstellning av foreningar som paverkar magsyrasekretionen |
SE7804231L (sv) * | 1978-04-14 | 1979-10-15 | Haessle Ab | Magsyrasekretionsmedel |
DE3216843C2 (de) * | 1982-05-05 | 1986-10-23 | Ludwig Heumann & Co GmbH, 8500 Nürnberg | 3-Thiomethyl-pyridin-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
CA1260474A (en) * | 1984-12-03 | 1989-09-26 | Raymond A. Stokbroekx | Benzoxazol- and benzothiazolamine derivatives |
SE8500996D0 (sv) * | 1985-03-01 | 1985-03-01 | Haessle Ab | Method of treatment |
DK399389A (da) * | 1988-08-18 | 1990-02-19 | Takeda Chemical Industries Ltd | Injicerbare oploesninger |
-
1968
- 1968-10-21 GB GB1234058D patent/GB1234058A/en not_active Expired
- 1968-10-22 DE DE19681804450 patent/DE1804450A1/de active Pending
- 1968-10-29 NL NL6815409A patent/NL6815409A/xx unknown
- 1968-11-05 FR FR172582A patent/FR1593614A/fr not_active Expired
Cited By (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4182766A (en) * | 1977-09-19 | 1980-01-08 | Hoffmann-La Roche Inc. | Naphth[2,3-d]imidazoles |
US4248880A (en) | 1977-09-19 | 1981-02-03 | Hoffmann-La Roche Inc. | Treatment of gastric ulcers with naphthimidazole derivatives |
US4738974A (en) * | 1983-03-04 | 1988-04-19 | Aktiebolaget Hassle | Base addition salts of omeprazole |
US4758579A (en) * | 1984-06-16 | 1988-07-19 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Fluoroalkoxy substituted benzimidazoles useful as gastric acid secretion inhibitors |
GB2161160B (en) * | 1984-07-06 | 1989-05-24 | Fisons Plc | Heterocyclic sulphinyl compounds |
US4738970A (en) * | 1984-12-18 | 1988-04-19 | Otsuka Pharmaceutical Co., Ltd. | Benzimidazolyl-thio-tetrahydroquinolines and anti-peptic ulcer compositions containing the same |
US4880815A (en) * | 1984-12-18 | 1989-11-14 | Otsuka Pharmaceutical Co., Ltd. | Imidazopyridyl-alkylthio-pyridines and anti-peptic ulcer compositions containing the same |
US4873337A (en) * | 1985-07-31 | 1989-10-10 | The Upjohn Company | N-substituted derivatives of 2-(pyridylalkenesulfinyl) benzimidazoles as gastric antisecretory agents |
US4791114A (en) * | 1986-01-20 | 1988-12-13 | 501 Laboratorios Del, Dr. Esteve | 2-Benzimidazolylalkylthio (or -sulfinyl or -sulfonyl) derivatives, their preparation and their application as medicinal products |
US5053417A (en) * | 1986-02-12 | 1991-10-01 | Tanabe Seiyaku Co., Ltd. | Imidazole derivatives and preparation thereof |
WO1987005296A1 (en) * | 1986-03-07 | 1987-09-11 | Pfizer Inc. | 2-[(2-pyridyl)methylsulfinyl]thienoimidazoles and related compounds as antiulcer agents |
EP0254588A1 (en) * | 1986-07-25 | 1988-01-27 | Tokyo Tanabe Company Limited | Imidazo[4,5-b] pyridine compounds, process for preparing same and pharmaceutical compositions containing same |
US5114955A (en) * | 1987-11-13 | 1992-05-19 | Hoechst Aketiengesellschaft | Substituted thienoimidazole derivatives |
JP2679745B2 (ja) | 1989-06-29 | 1997-11-19 | 明治製菓株式会社 | アゾール誘導体及びそれらを有効成分とする抗潰瘍剤 |
US5389664A (en) * | 1992-07-08 | 1995-02-14 | Monsanto Company | Alleviating stomach ulcers in swine |
US5703097A (en) * | 1994-02-28 | 1997-12-30 | Il-Yang Pharm. Co., Ltd. | 5-pyrrolyl-2-pyridylmethylsulfinyl benzimidazole derivatives |
US5859030A (en) * | 1994-06-10 | 1999-01-12 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Substituted arylalkylthioalkylthiopyridines for use in the control of helicobacter bacteria |
US6077541A (en) * | 1997-11-14 | 2000-06-20 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
US6780435B2 (en) | 1997-11-14 | 2004-08-24 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
US6174548B1 (en) | 1998-08-28 | 2001-01-16 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
US6855336B2 (en) | 1998-08-28 | 2005-02-15 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
US6733778B1 (en) | 1999-08-27 | 2004-05-11 | Andrx Pharmaceuticals, Inc. | Omeprazole formulation |
EP3050565A1 (en) * | 2015-01-27 | 2016-08-03 | Ecole Polytechnique Fédérale de Lausanne (EPFL) | Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis |
WO2016120259A1 (en) * | 2015-01-27 | 2016-08-04 | Ecole Polytechnique Federale De Lausanne (Epfl) | Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis |
US10137116B2 (en) | 2015-01-27 | 2018-11-27 | École Polytechnique Fédérale De Lausanne (Epfl) | Benzimidazole sulfide derivatives for the treatment or prevention of tuberculosis |
Also Published As
Publication number | Publication date |
---|---|
FR1593614A (es) | 1970-06-01 |
DE1804450A1 (de) | 1970-05-27 |
NL6815409A (es) | 1970-05-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PS | Patent sealed | ||
PLNP | Patent lapsed through nonpayment of renewal fees |