FR2829136B1 - Derives lipidiques d'aminoglycosides - Google Patents
Derives lipidiques d'aminoglycosidesInfo
- Publication number
- FR2829136B1 FR2829136B1 FR0111199A FR0111199A FR2829136B1 FR 2829136 B1 FR2829136 B1 FR 2829136B1 FR 0111199 A FR0111199 A FR 0111199A FR 0111199 A FR0111199 A FR 0111199A FR 2829136 B1 FR2829136 B1 FR 2829136B1
- Authority
- FR
- France
- Prior art keywords
- aminoglycosides
- lipid derivatives
- lipid
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0055—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of at least three carbon atoms which may or may not be branched, e.g. cholane or cholestane derivatives, optionally cyclised, e.g. 17-beta-phenyl or 17-beta-furyl derivatives
Priority Applications (9)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0111199A FR2829136B1 (fr) | 2001-08-29 | 2001-08-29 | Derives lipidiques d'aminoglycosides |
US10/228,959 US7772003B2 (en) | 2001-08-29 | 2002-08-28 | Lipid derivatives of aminoglycosides |
AT02796324T ATE430758T1 (de) | 2001-08-29 | 2002-08-29 | Lipid-aminoglykosid konjugate zur transfektion |
DE60232258T DE60232258D1 (de) | 2001-08-29 | 2002-08-29 | Lipid-aminoglykosid konjugate zur transfektion |
EP02796324A EP1430074B1 (fr) | 2001-08-29 | 2002-08-29 | Derives lipidiques d'aminoglycosides-pour la transfection |
AU2002334051A AU2002334051B2 (en) | 2001-08-29 | 2002-08-29 | Aminoglycoside lipid derivatives for transfection |
PCT/FR2002/002959 WO2003018603A1 (fr) | 2001-08-29 | 2002-08-29 | Derives lipidiques d'aminoglycosides_pour la transfection |
CA2458626A CA2458626C (fr) | 2001-08-29 | 2002-08-29 | Derives lipidiques d'aminoglycosides pour la transfection |
JP2003523262A JP4629333B2 (ja) | 2001-08-29 | 2002-08-29 | アミノグリコシドの脂質誘導体 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0111199A FR2829136B1 (fr) | 2001-08-29 | 2001-08-29 | Derives lipidiques d'aminoglycosides |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2829136A1 FR2829136A1 (fr) | 2003-03-07 |
FR2829136B1 true FR2829136B1 (fr) | 2006-11-17 |
Family
ID=8866791
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0111199A Expired - Lifetime FR2829136B1 (fr) | 2001-08-29 | 2001-08-29 | Derives lipidiques d'aminoglycosides |
Country Status (2)
Country | Link |
---|---|
US (1) | US7772003B2 (fr) |
FR (1) | FR2829136B1 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20080226605A1 (en) * | 2005-05-19 | 2008-09-18 | Dev Priya Arya | Methods and Compositions Facilitating Entry of Compounds Into Cells |
JP5407862B2 (ja) | 2006-10-04 | 2014-02-05 | サントル・ナシオナル・ドゥ・ラ・ルシェルシュ・シアンティフィーク(セーエヌエールエス) | siRNAおよび脂質性4,5−二置換2−デオキシストレプタミン環アミノグリコシド誘導体を含む組成物ならびにその用途 |
CA2729852A1 (fr) * | 2008-07-09 | 2010-01-14 | University Of Manitoba | Aminoglycosides ameliores au plan de l'hydrophobicite |
EP2542265A2 (fr) * | 2010-03-05 | 2013-01-09 | The University of Manitoba | Conjugués aminoglycoside-lipide guanidinylés |
Family Cites Families (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3293128A (en) * | 1961-11-24 | 1966-12-20 | Lilly Co Eli | Anthelmintic hygromycin b derivatives and process of using same |
BE758942A (fr) * | 1969-11-15 | 1971-04-16 | Abbou Richard | Medicament pour le traitement d'affections infectieuses et/ou inflammatoires |
US4400375A (en) * | 1981-11-23 | 1983-08-23 | Eli Lilly And Company | Tobramycin-double stranded RNA complex suitable for inducing interferon |
DE3486053T3 (de) | 1983-10-20 | 2004-01-08 | The Research Foundation Of State University Of New York | Regulierung von Gen-Expression durch Translationshemmung unter Verwendung von m-RNS hinderndem Komplementär-RNS. |
US6696420B1 (en) | 1984-11-20 | 2004-02-24 | Institut Pasteur | Adenoviral vector with a deletion in the E1A coding region expressing a hetorologous protein |
FR2573436B1 (fr) | 1984-11-20 | 1989-02-17 | Pasteur Institut | Adn recombinant comportant une sequence nucleotidique codant pour un polypeptide determine sous le controle d'un promoteur d'adenovirus, vecteurs contenant cet adn recombinant, cellules eucaryotes transformees par cet adn recombinant, produits d'excretion de ces cellules transformees et leurs applications, notamment a la constitution de vaccins |
FR2602790B1 (fr) | 1986-08-13 | 1990-06-01 | Transgene Sa | Expression d'un antigene specifique de tumeur par un virus vecteur recombinant et utilisation de celui-ci pour le traitement preventif ou curatif de la tumeur correspondante |
US5744133A (en) | 1986-08-13 | 1998-04-28 | Transgene S.A. | Expression of a tumor-specific antigen by a recombinant vector virus and use thereof in preventitive or curative treatment of the corresponding tumor |
WO1989005852A1 (fr) | 1987-12-15 | 1989-06-29 | Macphillamy Cummins & Gibson | Ribozymes |
US5543389A (en) * | 1990-11-01 | 1996-08-06 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education On Behalf Of The Oregon Health Sciences University, A Non Profit Organization | Covalent polar lipid-peptide conjugates for use in salves |
US6743623B2 (en) | 1991-09-27 | 2004-06-01 | Centre National De La Recherche Scientifique | Viral recombinant vectors for expression in muscle cells |
FR2681786A1 (fr) | 1991-09-27 | 1993-04-02 | Centre Nat Rech Scient | Vecteurs recombinants d'origine virale, leur procede d'obtention et leur utilisation pour l'expression de polypeptides dans des cellules musculaires. |
FR2688514A1 (fr) | 1992-03-16 | 1993-09-17 | Centre Nat Rech Scient | Adenovirus recombinants defectifs exprimant des cytokines et medicaments antitumoraux les contenant. |
FR2704234B1 (fr) | 1993-04-22 | 1995-07-21 | Centre Nat Rech Scient | Virus recombinants, preparation et utilisation en therapie genique. |
FR2704556B1 (fr) | 1993-04-30 | 1995-07-13 | Rhone Poulenc Rorer Sa | Virus recombinants et leur utilisation en thérapie génique. |
US6015686A (en) * | 1993-09-15 | 2000-01-18 | Chiron Viagene, Inc. | Eukaryotic layered vector initiation systems |
WO1996024334A1 (fr) * | 1995-02-10 | 1996-08-15 | Nexstar Pharmaceuticals, Inc. | Produits de synthese lipidique destines a la diffusion cytoplasmique d'agents |
FR2730637B1 (fr) | 1995-02-17 | 1997-03-28 | Rhone Poulenc Rorer Sa | Composition pharmaceutique contenant des acides nucleiques, et ses utilisations |
FR2739292B1 (fr) | 1995-09-28 | 1997-10-31 | Rhone Poulenc Rorer Sa | Composition pharmaceutique utile pour la transfection d'acides nucleiques et ses utilisations |
FR2741066B1 (fr) * | 1995-11-14 | 1997-12-12 | Rhone Poulenc Rorer Sa | Nouveaux agents de transfection et leurs applications pharmaceutiques |
DK0888379T3 (da) | 1996-03-01 | 2001-01-29 | Centre Nat Rech Scient | Forbindelser tilhørende amidinium-familien, farmaceutiske præparater indeholdende disse forbindelser og anvendelsen deraf |
US6071533A (en) * | 1996-11-12 | 2000-06-06 | The Regents Of The University Of California | Preparation of stable formulations of lipid-nucleic acid complexes for efficient in vivo delivery |
FR2764304B1 (fr) * | 1997-06-06 | 1999-07-16 | Rhone Poulenc Rorer Sa | Nouvelle classe d'agents transfectants cationiques des acides nucleiques |
JP2001515913A (ja) * | 1997-09-08 | 2001-09-25 | バレンティス・インコーポレーテッド | 疎水性グリコシルアミン誘導体の組成物及び使用方法 |
IL127773A0 (en) * | 1998-12-28 | 1999-10-28 | Yeda Res & Dev | Saccharide conjugates and pharmaceutical compositions comprising them |
AU2600100A (en) * | 1999-01-05 | 2000-07-24 | Valentis, Inc. | Methods and compositions for delivering nucleic acids |
GB9930533D0 (en) * | 1999-12-23 | 2000-02-16 | Mitsubishi Tokyo Pharm Inc | Nucleic acid delivery |
-
2001
- 2001-08-29 FR FR0111199A patent/FR2829136B1/fr not_active Expired - Lifetime
-
2002
- 2002-08-28 US US10/228,959 patent/US7772003B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
US7772003B2 (en) | 2010-08-10 |
US20030054556A1 (en) | 2003-03-20 |
FR2829136A1 (fr) | 2003-03-07 |
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Legal Events
Date | Code | Title | Description |
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PLFP | Fee payment |
Year of fee payment: 16 |
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PLFP | Fee payment |
Year of fee payment: 17 |
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PLFP | Fee payment |
Year of fee payment: 18 |
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PLFP | Fee payment |
Year of fee payment: 19 |
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PLFP | Fee payment |
Year of fee payment: 20 |