FR2789078B3 - Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant - Google Patents

Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant

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Publication number
FR2789078B3
FR2789078B3 FR9901201A FR9901201A FR2789078B3 FR 2789078 B3 FR2789078 B3 FR 2789078B3 FR 9901201 A FR9901201 A FR 9901201A FR 9901201 A FR9901201 A FR 9901201A FR 2789078 B3 FR2789078 B3 FR 2789078B3
Authority
FR
France
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
acid derivatives
pyrazolecarboxylic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
FR9901201A
Other languages
English (en)
Other versions
FR2789078A1 (fr
Inventor
Francis Barth
Frederic Larguier
Murielle Rinaldi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi SA filed Critical Sanofi SA
Priority to FR9901201A priority Critical patent/FR2789078B3/fr
Priority to FR9910166A priority patent/FR2789079B3/fr
Priority to EP00901661A priority patent/EP1150961B1/fr
Priority to PL350030A priority patent/PL198422B1/pl
Priority to JP2000597279A priority patent/JP3794925B2/ja
Priority to CA002358885A priority patent/CA2358885C/fr
Priority to MEP-2008-114A priority patent/ME00052B/fr
Priority to HU0201278A priority patent/HUP0201278A3/hu
Priority to DK00901661T priority patent/DK1150961T3/da
Priority to NZ512886A priority patent/NZ512886A/xx
Priority to IL14419800A priority patent/IL144198A0/xx
Priority to UA2001074905A priority patent/UA66900C2/uk
Priority to SI200030284T priority patent/SI1150961T1/xx
Priority to DE60006070T priority patent/DE60006070T2/de
Priority to AU22989/00A priority patent/AU754771B2/en
Priority to CNB008054681A priority patent/CN1146544C/zh
Priority to EEP200100399A priority patent/EE04343B1/xx
Priority to ES00901661T priority patent/ES2208267T3/es
Priority to RU2001121186/04A priority patent/RU2216542C2/ru
Priority to CZ20012697A priority patent/CZ297667B6/cs
Priority to ARP000100386A priority patent/AR020558A1/es
Priority to MEP-114/08A priority patent/MEP11408A/xx
Priority to IDW00200101603A priority patent/ID29534A/id
Priority to YUP-539/01A priority patent/RS50209B/sr
Priority to KR10-2001-7009572A priority patent/KR100425405B1/ko
Priority to SK1087-2001A priority patent/SK284203B6/sk
Priority to PE2000000066A priority patent/PE20001493A1/es
Priority to PT00901661T priority patent/PT1150961E/pt
Priority to TR2001/02054T priority patent/TR200102054T2/xx
Priority to BR0007895-6A priority patent/BR0007895A/pt
Priority to AT00901661T priority patent/ATE252562T1/de
Priority to US09/890,242 priority patent/US6432984B1/en
Priority to PCT/FR2000/000194 priority patent/WO2000046209A1/fr
Priority to TW089101649A priority patent/TW581764B/zh
Priority to CO00005429A priority patent/CO5160257A1/es
Publication of FR2789078A1 publication Critical patent/FR2789078A1/fr
Application granted granted Critical
Publication of FR2789078B3 publication Critical patent/FR2789078B3/fr
Priority to IL144198A priority patent/IL144198A/en
Priority to ZA200105739A priority patent/ZA200105739B/en
Priority to IS6002A priority patent/IS2448B/is
Priority to HR20010564A priority patent/HRP20010564B1/xx
Priority to BG105749A priority patent/BG65193B1/bg
Priority to NO20013736A priority patent/NO319824B1/no
Priority to HK02100712A priority patent/HK1039329A1/xx
Priority to US10/165,140 priority patent/US6645985B2/en
Priority to US10/455,220 priority patent/US20040039024A1/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/72—Hydrazones
    • C07C251/74—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C251/78—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
    • C07C251/80—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton the carbon skeleton containing rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9901201A 1999-02-01 1999-02-01 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant Expired - Lifetime FR2789078B3 (fr)

Priority Applications (44)

Application Number Priority Date Filing Date Title
FR9901201A FR2789078B3 (fr) 1999-02-01 1999-02-01 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant
FR9910166A FR2789079B3 (fr) 1999-02-01 1999-08-02 Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
EP00901661A EP1150961B1 (fr) 1999-02-01 2000-01-28 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant
PL350030A PL198422B1 (pl) 1999-02-01 2000-01-28 N-Piperydyno-5-(4-bromofenylo)-1-(2,4-dichlorofenylo)-4-etylopirazolo-3-karboksyamid, sposób jego wytwarzania, związki pośrednie, środek farmaceutyczny i zastosowanie
JP2000597279A JP3794925B2 (ja) 1999-02-01 2000-01-28 ピラゾールカルボン酸誘導体、その製造、それらを含む医薬組成物
CA002358885A CA2358885C (fr) 1999-02-01 2000-01-28 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant
MEP-2008-114A ME00052B (fr) 1999-02-01 2000-01-28 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant
HU0201278A HUP0201278A3 (en) 1999-02-01 2000-01-28 Pyrazolecarboamide derivative, its preparation, pharmaceutical compositions containing it and its intermediates
DK00901661T DK1150961T3 (da) 1999-02-01 2000-01-28 Pyrazolcarboxylsyrederivater, fremstilling af disse og farmaceutiske præparater indeholdende disse
NZ512886A NZ512886A (en) 1999-02-01 2000-01-28 N-Piperidino-5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole-3-carboxamide
IL14419800A IL144198A0 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
UA2001074905A UA66900C2 (uk) 1999-02-01 2000-01-28 Похідні піразолкарбонової кислоти, спосіб їх виготовлення, фармацевтична композиція, що їх містить
SI200030284T SI1150961T1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
DE60006070T DE60006070T2 (de) 1999-02-01 2000-01-28 Pyrazolcarbonsäurederivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen
AU22989/00A AU754771B2 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
CNB008054681A CN1146544C (zh) 1999-02-01 2000-01-28 吡唑甲酸类衍生物、其制备方法和含有它们的药物组合物
EEP200100399A EE04343B1 (et) 1999-02-01 2000-01-28 Pürasoolkarboksüülhappe derivaadid, nende valmistamine ja neid sisaldavad farmatseutilised kompositsioonid
ES00901661T ES2208267T3 (es) 1999-02-01 2000-01-28 Nevuo derivado de pirazol, sus sales y sus solvatos, procedimiento para su preparacion y composiciones farmaceuticas que los contienen.
RU2001121186/04A RU2216542C2 (ru) 1999-02-01 2000-01-28 Производные пиразолкарбоновой кислоты, их получение, содержащие их фармацевтические композиции
CZ20012697A CZ297667B6 (cs) 1999-02-01 2000-01-28 Derivát pyrazolkarboxylové kyseliny, zpusob jeho prípravy a farmaceutické prostredky, které ho obsahují
ARP000100386A AR020558A1 (es) 1999-02-01 2000-01-28 Un derivado de acido pirazolcarboxilico, su utilizacion, un procedimiento para su preparacion, composiciones farmaceuticas que lo contieneny compuestos utiles como intermediarios para prepararlo
MEP-114/08A MEP11408A (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing same
IDW00200101603A ID29534A (id) 1999-02-01 2000-01-28 Turunan-turunan asam pirazolkarboksilat, pembuatannya, komposisi-komposisi farmasi yang mengandungnya
YUP-539/01A RS50209B (sr) 1999-02-01 2000-01-28 Derivati pirazolokarboksilne kiseline, njihova priprema, farmaceutske kompozicije sa sadržajem istih
KR10-2001-7009572A KR100425405B1 (ko) 1999-02-01 2000-01-28 피라졸카르복실산 유도체, 그의 제조 방법, 및 그를함유하는 제약 조성물
SK1087-2001A SK284203B6 (sk) 1999-02-01 2000-01-28 Deriváty pyrazolkarboxylovej kyseliny, spôsob ich prípravy, farmaceutická kompozícia, ktorá ich obsahuje, a ich použitie
PE2000000066A PE20001493A1 (es) 1999-02-01 2000-01-28 Derivados de acido pirazolcarboxilico, un procedimiento para su preparacion y composiciones farmaceuticas que los contienen
PT00901661T PT1150961E (pt) 1999-02-01 2000-01-28 Derivados do acido pirazolecarboxilico processo para a sua preparacao e as composicoes farmaceuticas que os contem
TR2001/02054T TR200102054T2 (tr) 1999-02-01 2000-01-28 Pirazolkarboksilik asit türevleri, hazırlanmaları ve bunları içeren farmasötik kompozisyonlar.
BR0007895-6A BR0007895A (pt) 1999-02-01 2000-01-28 Derivados de ácido pirazolcarboxìlico, suapreparação e composições farmacêuticas que oscontêm
AT00901661T ATE252562T1 (de) 1999-02-01 2000-01-28 Pyrazolcarbonsäurederivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen
US09/890,242 US6432984B1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
PCT/FR2000/000194 WO2000046209A1 (fr) 1999-02-01 2000-01-28 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant
TW089101649A TW581764B (en) 1999-02-01 2000-01-31 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
CO00005429A CO5160257A1 (es) 1999-02-01 2000-01-31 La n-piperidino-5-(4-bromofenil)-1-(2,4-diclorofenil)-4-etilpirazol-3-carboxamida, sus sales, su preparacion y las composiciones farmaceuticas que la contienen
IL144198A IL144198A (en) 1999-02-01 2001-07-08 Derivatives of pyrazocarboxylic acid, their preparation, pharmaceutical compositions containing them
ZA200105739A ZA200105739B (en) 1999-02-01 2001-07-12 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them.
IS6002A IS2448B (is) 1999-02-01 2001-07-13 Pýrasólkarboxýlsýruafleiður, framleiðsla þeirra, lyfjasamsetningar sem innihalda þær
HR20010564A HRP20010564B1 (en) 1999-02-01 2001-07-26 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
BG105749A BG65193B1 (bg) 1999-02-01 2001-07-27 Производно на пиразолкарбоксилна киселина, неговото използване и фармацевтични състави, които го съдържат
NO20013736A NO319824B1 (no) 1999-02-01 2001-07-30 Pyrazolkarboksylsyrederivater, deres fremstilling og anvendelse og farmasoytiske preparater inneholdende de samme, samt mellomproduktforbindelser.
HK02100712A HK1039329A1 (en) 1999-02-01 2002-01-29 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
US10/165,140 US6645985B2 (en) 1999-02-01 2002-06-07 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them, and method of treating
US10/455,220 US20040039024A1 (en) 1999-02-01 2003-06-05 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9901201A FR2789078B3 (fr) 1999-02-01 1999-02-01 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant

Publications (2)

Publication Number Publication Date
FR2789078A1 FR2789078A1 (fr) 2000-08-04
FR2789078B3 true FR2789078B3 (fr) 2001-03-02

Family

ID=9541521

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9901201A Expired - Lifetime FR2789078B3 (fr) 1999-02-01 1999-02-01 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant

Country Status (2)

Country Link
FR (1) FR2789078B3 (fr)
ZA (1) ZA200105739B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1487436A4 (fr) 2002-03-08 2009-06-03 Signal Pharm Inc Polytherapie destinee a traiter, prevenir ou gerer des troubles proliferatifs et des cancers
CN100486973C (zh) 2002-07-29 2009-05-13 霍夫曼-拉罗奇有限公司 新苯并间二氧杂环戊烯类

Also Published As

Publication number Publication date
ZA200105739B (en) 2002-01-24
FR2789078A1 (fr) 2000-08-04

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