FR2763067B1 - Derives de 3-(1-azabicyclo[2.2.2] oct-3-ylalkyl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique - Google Patents

Derives de 3-(1-azabicyclo[2.2.2] oct-3-ylalkyl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique

Info

Publication number
FR2763067B1
FR2763067B1 FR9705537A FR9705537A FR2763067B1 FR 2763067 B1 FR2763067 B1 FR 2763067B1 FR 9705537 A FR9705537 A FR 9705537A FR 9705537 A FR9705537 A FR 9705537A FR 2763067 B1 FR2763067 B1 FR 2763067B1
Authority
FR
France
Prior art keywords
ylalkyl
oxadiazol
azabicyclo
therapeutics
oct
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
FR9705537A
Other languages
English (en)
Other versions
FR2763067A1 (fr
Inventor
Samir Jegham
Alistair Lochead
Alain Nedelec
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to FR9705537A priority Critical patent/FR2763067B1/fr
Priority to EP98924364A priority patent/EP0980370A1/fr
Priority to PCT/FR1998/000886 priority patent/WO1998050383A1/fr
Priority to AU76587/98A priority patent/AU7658798A/en
Priority to JP54777898A priority patent/JP2002504896A/ja
Priority to ZA983778A priority patent/ZA983778B/xx
Publication of FR2763067A1 publication Critical patent/FR2763067A1/fr
Application granted granted Critical
Publication of FR2763067B1 publication Critical patent/FR2763067B1/fr
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9705537A 1997-05-06 1997-05-06 Derives de 3-(1-azabicyclo[2.2.2] oct-3-ylalkyl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique Expired - Lifetime FR2763067B1 (fr)

Priority Applications (6)

Application Number Priority Date Filing Date Title
FR9705537A FR2763067B1 (fr) 1997-05-06 1997-05-06 Derives de 3-(1-azabicyclo[2.2.2] oct-3-ylalkyl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique
EP98924364A EP0980370A1 (fr) 1997-05-06 1998-05-04 Derives de 5-phenyl-1,3,4-oxadiazol-2(3h)-one et leur utilisation comme ligands 5-ht4
PCT/FR1998/000886 WO1998050383A1 (fr) 1997-05-06 1998-05-04 Derives de 5-phenyl-1,3,4-oxadiazol-2(3h)-one et leur utilisation comme ligands 5-ht4
AU76587/98A AU7658798A (en) 1997-05-06 1998-05-04 5-phenyl-1,3,4-oxadiazol-2(3h)-one derivatives and their use as 5-ht4 ligands
JP54777898A JP2002504896A (ja) 1997-05-06 1998-05-04 ５−フェニル−１，３，４−オキサジアゾール−２（３ｈ）−オン誘導体およびそれらの５−ｈｔ４リガンドとしての使用
ZA983778A ZA983778B (en) 1997-05-06 1998-05-05 Derivatives of 5-phenyl-1,3,4-oxadiazol-2(3H)-one their preparation and their application for therapeutic treatment

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9705537A FR2763067B1 (fr) 1997-05-06 1997-05-06 Derives de 3-(1-azabicyclo[2.2.2] oct-3-ylalkyl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
FR2763067A1 FR2763067A1 (fr) 1998-11-13
FR2763067B1 true FR2763067B1 (fr) 1999-06-04

Family

ID=9506607

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9705537A Expired - Lifetime FR2763067B1 (fr) 1997-05-06 1997-05-06 Derives de 3-(1-azabicyclo[2.2.2] oct-3-ylalkyl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique

Country Status (2)

Country Link
FR (1) FR2763067B1 (fr)
ZA (1) ZA983778B (fr)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8525844D0 (en) * 1985-10-19 1985-11-20 Beecham Group Plc Compounds
FR2719842B1 (fr) * 1994-05-10 1996-06-07 Synthelabo Sels quaternaires de dérivés de 1-azabicyclo [2.2.2] octane, leur préparation et leur application en thérapeutique.
AU6856094A (en) * 1994-06-01 1995-12-21 Yamanouchi Pharmaceutical Co., Ltd. Oxadiazole derivative and medicinal composition thereof

Also Published As

Publication number Publication date
FR2763067A1 (fr) 1998-11-13
ZA983778B (en) 1998-11-24

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