FR2436780A1 - Nouveau procede de preparation de nitroimidazoles - Google Patents

Nouveau procede de preparation de nitroimidazoles

Info

Publication number
FR2436780A1
FR2436780A1 FR7833416A FR7833416A FR2436780A1 FR 2436780 A1 FR2436780 A1 FR 2436780A1 FR 7833416 A FR7833416 A FR 7833416A FR 7833416 A FR7833416 A FR 7833416A FR 2436780 A1 FR2436780 A1 FR 2436780A1
Authority
FR
France
Prior art keywords
opt
cpd
nitro
halo
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7833416A
Other languages
English (en)
Other versions
FR2436780B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Farchemia SpA
Original Assignee
Farchemia SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farchemia SpA filed Critical Farchemia SpA
Publication of FR2436780A1 publication Critical patent/FR2436780A1/fr
Application granted granted Critical
Publication of FR2436780B1 publication Critical patent/FR2436780B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/91—Nitro radicals
    • C07D233/92—Nitro radicals attached in position 4 or 5

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

L'INVENTION SE RAPPORTE A LA CHIMIE ORGANIQUE. ELLE CONCERNE UN PROCEDE DE PREPARATION DE NITROIMIDAZOLES DE LA FORMULE: (CF DESSIN DANS BOPI) OU R ET R REPRESENTENT DIVERS SUBSTITUANTS, PAR REACTION D'UN 1-AMINO-SUBSTITUE-2-NITROETHYLENE AVEC UNE N-HALOGENOAMIDINE SUBSTITUEE. UTILISATION PAR L'INDUSTRIE PHARMACEUTIQUE POUR LA PREPARATION D'AGENTS ANTI-MICROBIENS CONNUS EN EUX-MEMES.
FR7833416A 1978-09-19 1978-11-27 Nouveau procede de preparation de nitroimidazoles Granted FR2436780A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT27866/78A IT1098864B (it) 1978-09-19 1978-09-19 Processo per la preparazione di nitroimidazoli

Publications (2)

Publication Number Publication Date
FR2436780A1 true FR2436780A1 (fr) 1980-04-18
FR2436780B1 FR2436780B1 (fr) 1982-04-09

Family

ID=11222488

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7833416A Granted FR2436780A1 (fr) 1978-09-19 1978-11-27 Nouveau procede de preparation de nitroimidazoles

Country Status (2)

Country Link
FR (1) FR2436780A1 (fr)
IT (1) IT1098864B (fr)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0049913A2 (fr) * 1980-09-17 1982-04-21 Gist-Brocades N.V. Dérivés d'imidazole éthénylique, procédé pour leur préparation et compositions pharmaceutiques les contenant; intermédiaires, utiles pour leur préparation et un procédé pour leur préparation
EP0057365A2 (fr) * 1981-01-30 1982-08-11 BASF Aktiengesellschaft Azoles vinyliques, procédé pour leur préparation et leur application comme fongicide
FR2504134A1 (fr) * 1981-04-21 1982-10-22 Bononi Loris Nouveaux derives du nitroimidazole, un procede pour leur preparation et compositions therapeutiques trichomonoacides en contenant
EP0103100A1 (fr) * 1982-08-20 1984-03-21 Euroresearch S.R.L. Dérivés de méthyl-1-nitro-5-imidazoline et compositions thérapeutiques les contenant
EP0111657A2 (fr) * 1982-10-27 1984-06-27 Pietro Tommaso Tessitore 2-(1-alkyl-5-nitro)-imidazolyl-1-(2-hydroxy-5-alkyl)-phényl-carbinols, procédé de leur préparation et leurs compositions pharmaceutiques
FR2625997A1 (fr) * 1988-01-15 1989-07-21 Rhone Poulenc Sante Procede de preparation du dimethyl-1,2 nitro-5 imidazole
EP0325512A1 (fr) * 1988-01-15 1989-07-26 Rhone-Poulenc Sante Procédé de préparation d'alkyl-1 nitro-5 imidazoles

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1119636A (en) * 1966-04-12 1968-07-10 Hoffmann La Roche A novel imidazole derivative and a novel intermediate therefor

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1119636A (en) * 1966-04-12 1968-07-10 Hoffmann La Roche A novel imidazole derivative and a novel intermediate therefor

Cited By (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0049913A2 (fr) * 1980-09-17 1982-04-21 Gist-Brocades N.V. Dérivés d'imidazole éthénylique, procédé pour leur préparation et compositions pharmaceutiques les contenant; intermédiaires, utiles pour leur préparation et un procédé pour leur préparation
EP0049913A3 (en) * 1980-09-17 1982-10-06 Gist - Brocades N.V. New ethenylimidazole derivatives, processes for their preparation and pharmaceutical compositions containing them; intermediates, useful in their preparation and a process for the preparation thereof
EP0057365A2 (fr) * 1981-01-30 1982-08-11 BASF Aktiengesellschaft Azoles vinyliques, procédé pour leur préparation et leur application comme fongicide
EP0057365A3 (en) * 1981-01-30 1982-09-01 Basf Aktiengesellschaft Vinyl azoles, process for their preparation and their application as fungicides
EP0063401A3 (en) * 1981-04-21 1983-09-21 Loris Jacopo Bononi Nitroimidazoles having trichomonacidal activity, a process for their preparation and related pharmaceutical compositions
EP0063401A2 (fr) * 1981-04-21 1982-10-27 Loris Jacopo Bononi Nitroimidazoles avec une activité trichomonicide, procédé pour leur préparation et leurs compositions pharmaceutiques
FR2504134A1 (fr) * 1981-04-21 1982-10-22 Bononi Loris Nouveaux derives du nitroimidazole, un procede pour leur preparation et compositions therapeutiques trichomonoacides en contenant
US4463012A (en) * 1981-04-21 1984-07-31 Bononi Loris J Nitroimidazoles having trichomonacidal activity and pharmaceutical compositions thereof
EP0103100A1 (fr) * 1982-08-20 1984-03-21 Euroresearch S.R.L. Dérivés de méthyl-1-nitro-5-imidazoline et compositions thérapeutiques les contenant
US4476138A (en) * 1982-08-20 1984-10-09 Farmatis S.R.L. 1-Methyl-5-nitro-(2-substituted)-2H-imidazole derivatives, and use as bactericidal and protozoacidal agents
EP0111657A2 (fr) * 1982-10-27 1984-06-27 Pietro Tommaso Tessitore 2-(1-alkyl-5-nitro)-imidazolyl-1-(2-hydroxy-5-alkyl)-phényl-carbinols, procédé de leur préparation et leurs compositions pharmaceutiques
EP0111657A3 (fr) * 1982-10-27 1984-07-25 Pietro Tommaso Tessitore 2-(1-alkyl-5-nitro)-imidazolyl-1-(2-hydroxy-5-alkyl)-phényl-carbinols, procédé de leur préparation et leurs compositions pharmaceutiques
US4478846A (en) * 1982-10-27 1984-10-23 Tessitore Pietro T 2-(1-Alkyl-5-nitro)-imidazolyl-1-(2-hydroxy-5-alkyl)-phenyl carbinols and pharmaceutical compositions containing them
FR2625997A1 (fr) * 1988-01-15 1989-07-21 Rhone Poulenc Sante Procede de preparation du dimethyl-1,2 nitro-5 imidazole
EP0325512A1 (fr) * 1988-01-15 1989-07-26 Rhone-Poulenc Sante Procédé de préparation d'alkyl-1 nitro-5 imidazoles

Also Published As

Publication number Publication date
IT7827866A0 (it) 1978-09-19
FR2436780B1 (fr) 1982-04-09
IT1098864B (it) 1985-09-18

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