FR2073338A1 - 6-(methyleneamino)-penicillanic acid derivs - Google Patents

6-(methyleneamino)-penicillanic acid derivs

Info

Publication number
FR2073338A1
FR2073338A1 FR7040428A FR7040428A FR2073338A1 FR 2073338 A1 FR2073338 A1 FR 2073338A1 FR 7040428 A FR7040428 A FR 7040428A FR 7040428 A FR7040428 A FR 7040428A FR 2073338 A1 FR2073338 A1 FR 2073338A1
Authority
FR
France
Prior art keywords
alkyl
heterocyclic
penicillanic acid
residue
methyleneamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7040428A
Other languages
French (fr)
Other versions
FR2073338B1 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SARATH
Original Assignee
SARATH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB33211/70A external-priority patent/GB1293590A/en
Application filed by SARATH filed Critical SARATH
Publication of FR2073338A1 publication Critical patent/FR2073338A1/en
Application granted granted Critical
Publication of FR2073338B1 publication Critical patent/FR2073338B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/02—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Penicillanic acid derivs. of formula (I) : (where R1 and R2 = an aliphatic hydrocarbon residue, a mono- or bi-cyclic aryl residue, aralkyl, cycloalkyl, cycloalkylalkyl, a heterocyclic or heterocyclic substd. alkyl gp., or R1R2N = a heterocyclic residue and R4 = H, alkyl, aryl, aralkyl, cycloalkylalkyl, haloalkyl, O-alkyl, alkanoyl, aroyl, CN, CO2 alkyl or acyloxymethyl) and salts of (I), are antibacterials of low toxicity. (I) are prepd. by condensing (a) 6-aminopenicillanic acid (II) with a reactive amide or thioamide deriv. : R1R2NCH=R5, or (b) a reactive deriv. of (III) with an amine R1R2NH.
FR7040428A 1969-11-11 1970-11-10 6-(methyleneamino)-penicillanic acid derivs Granted FR2073338A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB5520969 1969-11-11
GB33211/70A GB1293590A (en) 1969-11-11 1969-11-11 New penicillanic acid derivatives

Publications (2)

Publication Number Publication Date
FR2073338A1 true FR2073338A1 (en) 1971-10-01
FR2073338B1 FR2073338B1 (en) 1974-02-15

Family

ID=26261769

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7040428A Granted FR2073338A1 (en) 1969-11-11 1970-11-10 6-(methyleneamino)-penicillanic acid derivs

Country Status (22)

Country Link
JP (1) JPS518955B1 (en)
AT (1) AT301026B (en)
BE (1) BE758782A (en)
BG (1) BG18619A3 (en)
CH (2) CH559752A5 (en)
CS (1) CS166020B2 (en)
DE (1) DE2055531C3 (en)
DK (1) DK135127B (en)
ES (1) ES385437A1 (en)
FI (1) FI54601C (en)
FR (1) FR2073338A1 (en)
HU (1) HU162440B (en)
IE (1) IE34620B1 (en)
IL (1) IL35490A (en)
IT (1) IT1044209B (en)
LU (1) LU62031A1 (en)
NL (1) NL168227C (en)
NO (1) NO137826C (en)
PL (1) PL90581B1 (en)
RO (2) RO56878A (en)
SE (1) SE397355B (en)
SU (1) SU406362A3 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2296638A1 (en) * 1975-01-06 1976-07-30 Inst Organicheskogo Sinteza Ak PROCESS FOR PREPARING 6-B-AMIDINOPENICILLANIC ACID DERIVATIVES

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL79157B1 (en) * 1970-12-22 1975-06-30
GB1364672A (en) * 1971-06-09 1974-08-29 Beecham Group Ltd Penicillins
GB1427139A (en) * 1972-03-13 1976-03-10 Astra Laekemedel Ab Penicillins
GB1417099A (en) * 1973-02-02 1975-12-10 Leo Pharm Prod Ltd Method for the production of derivatives of 6-aminopenicillanic acid
GB1579931A (en) * 1976-04-15 1980-11-26 Leo Pharm Prod Ltd Bis-penicillanoyl-oxy-alkanes
TWI375678B (en) 2005-06-09 2012-11-01 Yakult Honsha Kk A method of preparation of a tricyclic ketone

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3135755A (en) * 1961-11-20 1964-06-02 Hoffmann La Roche Pyrimidine formamidines of primary amines
US3322781A (en) * 1963-10-18 1967-05-30 Bristol Myers Co 6-(substituted-hydroxyamidino)-penicillanic acids
CH480792A (en) * 1967-01-26 1969-11-15 Ciba Geigy Pesticides

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
NEANT *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2296638A1 (en) * 1975-01-06 1976-07-30 Inst Organicheskogo Sinteza Ak PROCESS FOR PREPARING 6-B-AMIDINOPENICILLANIC ACID DERIVATIVES

Also Published As

Publication number Publication date
JPS518955B1 (en) 1976-03-22
SE397355B (en) 1977-10-31
SU406362A3 (en) 1973-11-05
FI54601B (en) 1978-09-29
DK135127C (en) 1977-08-15
IE34620B1 (en) 1975-06-25
NL168227B (en) 1981-10-16
DK135127B (en) 1977-03-07
FI54601C (en) 1979-01-10
BE758782A (en) 1971-05-10
NO137826B (en) 1978-01-23
IL35490A0 (en) 1970-12-24
DE2055531C3 (en) 1982-02-25
DE2055531B2 (en) 1980-01-10
IT1044209B (en) 1980-03-20
CH559752A5 (en) 1975-03-14
IE34620L (en) 1971-05-11
RO56878A (en) 1975-02-15
NL7016435A (en) 1971-05-13
NL168227C (en) 1982-03-16
IL35490A (en) 1974-11-29
ES385437A1 (en) 1973-11-01
AT301026B (en) 1972-08-25
HU162440B (en) 1973-02-28
FR2073338B1 (en) 1974-02-15
NO137826C (en) 1982-02-16
RO60563A (en) 1977-01-15
LU62031A1 (en) 1971-05-10
DE2055531A1 (en) 1971-05-27
PL90581B1 (en) 1977-01-31
CS166020B2 (en) 1976-01-29
CH559753A5 (en) 1975-03-14
BG18619A3 (en) 1975-02-25

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Legal Events

Date Code Title Description
TP Transmission of property
CC Supplementary protection certificate (spc) laid open to the public (law of 25 june 1990)

Free format text: 92C0027, 920225

CB Supplementary protection certificate (spc) granted (law of 25 june 1990)

Free format text: 92C0027, 701110

CP Supplementary protection certificate (spc) filed