FI961599A - 1N-alkyl-N-arylpyrimidinamines and their derivatives - Google Patents

1N-alkyl-N-arylpyrimidinamines and their derivatives Download PDF

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Publication number
FI961599A
FI961599A FI961599A FI961599A FI961599A FI 961599 A FI961599 A FI 961599A FI 961599 A FI961599 A FI 961599A FI 961599 A FI961599 A FI 961599A FI 961599 A FI961599 A FI 961599A
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Finland
Prior art keywords
arylpyrimidinamines
derivatives
alkyl
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FI961599A
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Finnish (fi)
Swedish (sv)
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FI961599A0 (en
Inventor
Paul Edward Aldrich
Argyrios Georgios Arvanitis
Robert Scott Cheeseman
Robert John Chorvat
Thomas Eugene Christos
Paul Joseph Gilligan
Dimitri Emil Grigoriadis
Carl Nicholas Hodge
Paul John Krenitsky
Everett Latham Scholfield
Sang William Tam
Zelda Rakowitz Wasserman
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Du Pont Merck Pharma
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Publication of FI961599A0 publication Critical patent/FI961599A0/en
Publication of FI961599A publication Critical patent/FI961599A/en

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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FI961599A 1993-10-12 1996-04-11 1N-alkyl-N-arylpyrimidinamines and their derivatives FI961599A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US13420993A 1993-10-12 1993-10-12
US29727494A 1994-08-26 1994-08-26
PCT/US1994/011050 WO1995010506A1 (en) 1993-10-12 1994-10-06 1n-alkyl-n-arylpyrimidinamines and derivatives thereof

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FI961599A0 FI961599A0 (en) 1996-04-11
FI961599A true FI961599A (en) 1996-06-07

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JP (1) JP3398152B2 (en)
CN (1) CN1142817A (en)
FI (1) FI961599A (en)
RU (1) RU2153494C2 (en)
TW (1) TW286316B (en)
WO (1) WO1995010506A1 (en)

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CA2188427C (en) * 1994-04-29 2000-06-27 Robert A. Volkmann Neurotransmitter release enhancers
TW530047B (en) * 1994-06-08 2003-05-01 Pfizer Corticotropin releasing factor antagonists
JP2891544B2 (en) 1994-06-16 1999-05-17 ファイザー・インコーポレーテッド Pyrazolo and pyrrolopyridines
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