FI941212A - Fuusioituneet trisykliset, typpeä sisältävät heterosykliset yhdisteet - Google Patents

Fuusioituneet trisykliset, typpeä sisältävät heterosykliset yhdisteet Download PDF

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Publication number
FI941212A
FI941212A FI941212A FI941212A FI941212A FI 941212 A FI941212 A FI 941212A FI 941212 A FI941212 A FI 941212A FI 941212 A FI941212 A FI 941212A FI 941212 A FI941212 A FI 941212A
Authority
FI
Finland
Prior art keywords
pct
containing heterocyclic
heterocyclic compounds
fused tricyclic
compounds
Prior art date
Application number
FI941212A
Other languages
English (en)
Swedish (sv)
Other versions
FI941212A0 (fi
Inventor
John A Lowe Iii
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI941212A0 publication Critical patent/FI941212A0/fi
Publication of FI941212A publication Critical patent/FI941212A/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
FI941212A 1991-09-26 1994-03-15 Fuusioituneet trisykliset, typpeä sisältävät heterosykliset yhdisteet FI941212A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76648891A 1991-09-26 1991-09-26
PCT/US1992/006819 WO1993006099A1 (en) 1991-09-16 1992-08-20 Fused tricyclic nitrogen containing heterocycles as substance p receptor antagonists

Publications (2)

Publication Number Publication Date
FI941212A0 FI941212A0 (fi) 1994-03-15
FI941212A true FI941212A (fi) 1994-03-15

Family

ID=25076576

Family Applications (1)

Application Number Title Priority Date Filing Date
FI941212A FI941212A (fi) 1991-09-26 1994-03-15 Fuusioituneet trisykliset, typpeä sisältävät heterosykliset yhdisteet

Country Status (19)

Country Link
US (1) US5527808A (fi)
EP (1) EP0607164B1 (fi)
JP (1) JP2535134B2 (fi)
CN (1) CN1071168A (fi)
AT (1) ATE216996T1 (fi)
AU (1) AU2481292A (fi)
BR (1) BR9206500A (fi)
CA (1) CA2118704C (fi)
CZ (1) CZ59394A3 (fi)
DE (1) DE69232588T2 (fi)
DK (1) DK0607164T3 (fi)
ES (1) ES2174836T3 (fi)
FI (1) FI941212A (fi)
HU (1) HU9400728D0 (fi)
MX (1) MX9205242A (fi)
NO (1) NO940927L (fi)
PT (1) PT100901A (fi)
WO (1) WO1993006099A1 (fi)
ZA (1) ZA927370B (fi)

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FR2700472B1 (fr) 1993-01-19 1995-02-17 Rhone Poulenc Rorer Sa Association synergisante ayant un effet antagoniste des récepteurs NK1 et NK2.
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
EP0653208A3 (en) * 1993-11-17 1995-10-11 Pfizer Substance P antagonists for the treatment or prevention of sunburn.
EP0659409A3 (en) * 1993-11-23 1995-08-09 Pfizer Substance P antagonists for the inhibition of angiogenesis.
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IL116249A (en) * 1994-12-12 2003-07-06 Pfizer Nk-1 receptor antagonists for the treatment of neuronal damage and stroke
FR2728265A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p dans une composition pharmaceutique
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2728169A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
TW458774B (en) 1995-10-20 2001-10-11 Pfizer Antiemetic pharmaceutical compositions
FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
CA2324116A1 (en) * 1999-10-25 2001-04-25 Susan Beth Sobolov-Jaynes Nk-1 receptor antagonists and eletriptan for the treatment of migraine
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US20110218176A1 (en) 2006-11-01 2011-09-08 Barbara Brooke Jennings-Spring Compounds, methods, and treatments for abnormal signaling pathways for prenatal and postnatal development
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US8389553B2 (en) 2007-06-27 2013-03-05 Merck Sharp & Dohme Corp. 4-carboxybenzylamino derivatives as histone deacetylase inhibitors
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JP5739415B2 (ja) 2009-05-12 2015-06-24 ブリストル−マイヤーズ スクウィブ カンパニー （Ｓ）−７−（［１，２，４］トリアゾロ［１，５−ａ］ピリジン−６−イル）−４−（３，４−ジクロロフェニル）−１，２，３，４−テトラヒドロイソキノリンの結晶形態およびその使用
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Family Cites Families (4)

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US3534053A (en) * 1967-05-24 1970-10-13 American Home Prod Quinuclidine derivatives
US3506673A (en) * 1968-03-29 1970-04-14 Aldrich Chem Co Inc 2-(4'halo)-benzhydryl-3-quinuclidinols
WO1990005525A1 (en) * 1988-11-23 1990-05-31 Pfizer Inc. Quinuclidine derivatives as substance p antagonists
DE69106365T2 (de) * 1990-07-23 1995-05-04 Pfizer Chinuclidinderivate.

Also Published As

Publication number Publication date
PT100901A (pt) 1994-02-28
JPH06507179A (ja) 1994-08-11
BR9206500A (pt) 1995-10-03
NO940927D0 (no) 1994-03-15
CZ59394A3 (en) 1994-11-16
US5527808A (en) 1996-06-18
HU9400728D0 (en) 1994-06-28
NO940927L (no) 1994-03-15
DK0607164T3 (da) 2002-06-17
WO1993006099A1 (en) 1993-04-01
DE69232588D1 (de) 2002-06-06
CA2118704C (en) 1997-01-21
EP0607164B1 (en) 2002-05-02
CN1071168A (zh) 1993-04-21
DE69232588T2 (de) 2002-08-22
ATE216996T1 (de) 2002-05-15
EP0607164A1 (en) 1994-07-27
ES2174836T3 (es) 2002-11-16
AU2481292A (en) 1993-04-27
FI941212A0 (fi) 1994-03-15
MX9205242A (es) 1993-03-01
JP2535134B2 (ja) 1996-09-18
ZA927370B (en) 1994-03-25
CA2118704A1 (en) 1993-04-01

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