FI935658A - Nya selektiva aromatasinhiberande 4(5)-imidazoler - Google Patents
Nya selektiva aromatasinhiberande 4(5)-imidazoler Download PDFInfo
- Publication number
- FI935658A FI935658A FI935658A FI935658A FI935658A FI 935658 A FI935658 A FI 935658A FI 935658 A FI935658 A FI 935658A FI 935658 A FI935658 A FI 935658A FI 935658 A FI935658 A FI 935658A
- Authority
- FI
- Finland
- Prior art keywords
- hiberande
- aromatasin
- imidazoler
- nya
- selective
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB919113142A GB9113142D0 (en) | 1991-06-18 | 1991-06-18 | New selective aromatase inhibiting 4(5)-imidazoles |
GB919125924A GB9125924D0 (en) | 1991-06-18 | 1991-12-05 | Stereoisomers of an imidazole derivative |
PCT/FI1992/000184 WO1992022537A1 (en) | 1991-06-18 | 1992-06-12 | New selective aromatase inhibiting 4(5)-imidazoles |
Publications (2)
Publication Number | Publication Date |
---|---|
FI935658A true FI935658A (fi) | 1993-12-16 |
FI935658A0 FI935658A0 (fi) | 1993-12-16 |
Family
ID=26299089
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI935658A FI935658A0 (fi) | 1991-06-18 | 1993-12-16 | Nya selektiva aromatasinhiberande 4(5)-imidazoler |
Country Status (25)
Country | Link |
---|---|
US (1) | US5559141A (fi) |
EP (1) | EP0589975A1 (fi) |
JP (1) | JPH06508119A (fi) |
KR (1) | KR940701386A (fi) |
CN (1) | CN1068819A (fi) |
AU (1) | AU665002B2 (fi) |
BG (1) | BG98306A (fi) |
CA (1) | CA2111469A1 (fi) |
CZ (1) | CZ280293A3 (fi) |
FI (1) | FI935658A0 (fi) |
GB (1) | GB9125924D0 (fi) |
HR (1) | HRP920170A2 (fi) |
HU (1) | HUT67325A (fi) |
IE (1) | IE921963A1 (fi) |
IL (2) | IL102216A (fi) |
LT (1) | LT3164B (fi) |
LV (1) | LV10093B (fi) |
MX (1) | MX9203000A (fi) |
NO (1) | NO934688L (fi) |
NZ (1) | NZ243139A (fi) |
PT (1) | PT100604A (fi) |
SI (1) | SI9200113A (fi) |
SK (1) | SK144393A3 (fi) |
TW (1) | TW206217B (fi) |
WO (1) | WO1992022537A1 (fi) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2273704B (en) * | 1992-12-16 | 1997-01-22 | Orion Yhtymae Oy | Triazolyl diaryl selective aromatase inhibiting compounds |
SE9302333D0 (sv) * | 1993-07-06 | 1993-07-06 | Ab Astra | New compounds |
US6080870A (en) * | 1996-04-03 | 2000-06-27 | Merck & Co., Inc. | Biaryl substituted imidazole compounds useful as farnesyl-protein transferase inhibitors |
US6063930A (en) * | 1996-04-03 | 2000-05-16 | Merck & Co., Inc. | Substituted imidazole compounds useful as farnesyl-protein transferase inhibitors |
AU716123B2 (en) * | 1996-04-03 | 2000-02-17 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
US6297239B1 (en) * | 1997-10-08 | 2001-10-02 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
KR20030031132A (ko) | 2000-07-28 | 2003-04-18 | 스미또모 세이야꾸 가부시키가이샤 | 피롤 유도체 |
JP4667384B2 (ja) * | 2003-10-07 | 2011-04-13 | レノビス, インコーポレイテッド | イオンチャネルリガンドとしてのアミド誘導体および薬学的組成物、ならびにこれらを使用する方法 |
BRPI0606365A2 (pt) * | 2005-02-28 | 2017-06-27 | Renovis Inc | composto ou um sal, solvato ou pró-droga farmaceuticamente aceitável do mesmo e estereoisômeros e tautômeros do mesmo, composição farmacêutica, métodos para prevenir, tratar, melhorar ou controlar uma doença ou condição e para preparar um composto, uso de um composto ou um sal, solvato ou composição farmaceuticamente aceitável do mesmo, método de tratamento de um mamífero, e, combinação |
US7576099B2 (en) | 2005-02-28 | 2009-08-18 | Renovis, Inc. | Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
US7902247B2 (en) * | 2008-01-09 | 2011-03-08 | Allergan, Inc. | Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4605661A (en) * | 1984-06-18 | 1986-08-12 | Eli Lilly And Company | Aromastase inhibiting α,α-diarylimidazole-4(5)-propionitriles, α,α-diarylimidazole-4(5)-propionamides, and 4(5)-(2,2-diarylethyl)imidazoles |
GB2210875B (en) * | 1987-10-09 | 1991-05-29 | Farmos Oy | Aromatase inhibiting 4(5)-imidazoles |
GB2248058B (en) * | 1990-09-21 | 1994-09-14 | Orion Yhtymae Oy | Aromatase inhibiting 4(5)-imidazoles |
US5439928A (en) * | 1989-03-30 | 1995-08-08 | Orion-Yhtyma Oy | Aromatase inhibiting 4(5)-imidazoles |
AU627559B2 (en) * | 1989-03-30 | 1992-08-27 | Farmos-Yhtyma Oy | Novel aromatase inhibiting 4(5)-imidazoles |
-
1991
- 1991-12-05 GB GB919125924A patent/GB9125924D0/en active Pending
-
1992
- 1992-06-12 KR KR1019930703934A patent/KR940701386A/ko not_active Application Discontinuation
- 1992-06-12 AU AU19783/92A patent/AU665002B2/en not_active Ceased
- 1992-06-12 CA CA002111469A patent/CA2111469A1/en not_active Abandoned
- 1992-06-12 CZ CS932802A patent/CZ280293A3/cs unknown
- 1992-06-12 WO PCT/FI1992/000184 patent/WO1992022537A1/en not_active Application Discontinuation
- 1992-06-12 US US08/167,873 patent/US5559141A/en not_active Expired - Fee Related
- 1992-06-12 SK SK1443-93A patent/SK144393A3/sk unknown
- 1992-06-12 EP EP92912309A patent/EP0589975A1/en not_active Withdrawn
- 1992-06-12 JP JP4511061A patent/JPH06508119A/ja active Pending
- 1992-06-15 LV LVP-92-29A patent/LV10093B/en unknown
- 1992-06-15 NZ NZ243139A patent/NZ243139A/en unknown
- 1992-06-16 IL IL10221692A patent/IL102216A/en not_active IP Right Cessation
- 1992-06-17 HR HR920170A patent/HRP920170A2/hr not_active Application Discontinuation
- 1992-06-17 TW TW081104752A patent/TW206217B/zh active
- 1992-06-17 PT PT100604A patent/PT100604A/pt not_active Application Discontinuation
- 1992-06-18 CN CN92105664A patent/CN1068819A/zh active Pending
- 1992-06-18 SI SI19929200113A patent/SI9200113A/sl unknown
- 1992-06-18 MX MX9203000A patent/MX9203000A/es unknown
- 1992-07-01 IE IE196392A patent/IE921963A1/en not_active Application Discontinuation
- 1992-08-28 LT LTIP175A patent/LT3164B/lt not_active IP Right Cessation
-
1993
- 1993-12-16 FI FI935658A patent/FI935658A0/fi not_active Application Discontinuation
- 1993-12-17 HU HU9303653A patent/HUT67325A/hu active IP Right Revival
- 1993-12-17 BG BG98306A patent/BG98306A/bg unknown
- 1993-12-17 NO NO934688A patent/NO934688L/no unknown
-
1995
- 1995-09-27 IL IL11543995A patent/IL115439A0/xx unknown
Also Published As
Publication number | Publication date |
---|---|
SI9200113A (en) | 1992-12-31 |
IE921963A1 (en) | 1992-12-30 |
IL115439A0 (en) | 1995-12-31 |
WO1992022537A1 (en) | 1992-12-23 |
LT3164B (en) | 1995-02-27 |
HU9303653D0 (en) | 1994-04-28 |
BG98306A (bg) | 1994-08-30 |
MX9203000A (es) | 1993-02-01 |
HUT67325A (en) | 1995-03-28 |
JPH06508119A (ja) | 1994-09-14 |
NO934688D0 (no) | 1993-12-17 |
GB9125924D0 (en) | 1992-02-05 |
AU1978392A (en) | 1993-01-12 |
AU665002B2 (en) | 1995-12-14 |
CZ280293A3 (en) | 1994-05-18 |
LV10093B (en) | 1995-02-20 |
HRP920170A2 (en) | 1994-08-31 |
FI935658A0 (fi) | 1993-12-16 |
US5559141A (en) | 1996-09-24 |
NZ243139A (en) | 1994-08-26 |
NO934688L (no) | 1993-12-17 |
CA2111469A1 (en) | 1992-12-23 |
LV10093A (lv) | 1994-05-10 |
PT100604A (pt) | 1993-10-29 |
CN1068819A (zh) | 1993-02-10 |
EP0589975A1 (en) | 1994-04-06 |
IL102216A0 (en) | 1993-01-14 |
LTIP175A (lt) | 1994-08-25 |
SK144393A3 (en) | 1994-11-09 |
TW206217B (fi) | 1993-05-21 |
KR940701386A (ko) | 1994-05-28 |
IL102216A (en) | 1996-06-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |