FI916036A0 - Menetelmä valmistaa farmaseuttisesti käyttökelpoista spirofuraanijohdosta - Google Patents

Menetelmä valmistaa farmaseuttisesti käyttökelpoista spirofuraanijohdosta

Info

Publication number
FI916036A0
FI916036A0 FI916036A FI916036A FI916036A0 FI 916036 A0 FI916036 A0 FI 916036A0 FI 916036 A FI916036 A FI 916036A FI 916036 A FI916036 A FI 916036A FI 916036 A0 FI916036 A0 FI 916036A0
Authority
FI
Finland
Prior art keywords
spirofuran
derivative
prepared
pharmaceutically acceptable
pharmaceutically
Prior art date
Application number
FI916036A
Other languages
English (en)
Swedish (sv)
Other versions
FI96114C (fi
FI96114B (fi
Inventor
Wu Edwin Schen-Chou
Ronald Conrad Griffith
Original Assignee
Fisons Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fisons Corp filed Critical Fisons Corp
Publication of FI916036A0 publication Critical patent/FI916036A0/fi
Application granted granted Critical
Publication of FI96114B publication Critical patent/FI96114B/fi
Publication of FI96114C publication Critical patent/FI96114C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI916036A 1989-06-21 1991-12-20 Menetelmä valmistaa farmaseuttisesti käyttökelpoista spirofuraanijohdosta FI96114C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US36932489 1989-06-21
US07/369,324 US5075317A (en) 1989-06-21 1989-06-21 Spirofurane derivatives
US9003351 1990-06-20
PCT/US1990/003351 WO1990015804A1 (en) 1989-06-21 1990-06-20 Novel spirofurane derivatives

Publications (3)

Publication Number Publication Date
FI916036A0 true FI916036A0 (fi) 1991-12-20
FI96114B FI96114B (fi) 1996-01-31
FI96114C FI96114C (fi) 1996-05-10

Family

ID=23454995

Family Applications (1)

Application Number Title Priority Date Filing Date
FI916036A FI96114C (fi) 1989-06-21 1991-12-20 Menetelmä valmistaa farmaseuttisesti käyttökelpoista spirofuraanijohdosta

Country Status (9)

Country Link
US (1) US5075317A (fi)
EP (1) EP0490901A1 (fi)
JP (1) JPH04506210A (fi)
CA (1) CA2062809A1 (fi)
FI (1) FI96114C (fi)
GR (1) GR1000887B (fi)
IE (1) IE902242A1 (fi)
PT (1) PT94440A (fi)
WO (1) WO1990015804A1 (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE914238A1 (en) * 1990-12-19 1992-07-01 Fisons Corp Novel spirofurane derivatives
RU2057132C1 (ru) * 1991-05-15 1996-03-27 Яманоути Фармасьютикал Ко., Лтд. Моногидрат (-)-(s)-2,8-диметил-3-метилен-1-окса-8-азаспиро[4,5]-декана l-тартрата и способ его получения
IL107881A0 (en) * 1992-12-05 1994-04-12 Fisons Corp Furanone derivatives and pharmaceutical compositions containing them
EP0681571B1 (en) * 1993-01-28 1998-07-29 Merck & Co. Inc. Spiro-substituted azacycles as tachykinin receptor antagonists
DE69318854T2 (de) * 1993-03-04 1998-10-08 Pfizer Spiroazacyclischderivate als substanz p antagonisten
DE102006050503A1 (de) * 2006-10-26 2008-04-30 GM Global Technology Operations, Inc., Detroit Schaltkupplung für Schalt-/Synchronisiereinrichtung, insbesondere für Schaltgetriebe eines Kraftfahrzeugs
US9034891B2 (en) 2009-01-26 2015-05-19 Israel Institute For Biological Research Bicyclic heterocyclic spiro compounds
BRPI1007350B8 (pt) * 2009-01-26 2021-05-25 Israel Institute For Biological Res compostos espiro heterocíclicos bicíclicos

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0189370A3 (de) * 1985-01-16 1988-01-27 Sandoz Ag Spiro-dioxolane, -dithiolane und -oxothiolane
NZ219646A (en) * 1986-03-27 1990-10-26 Merck Sharp & Dohme Oxadiazole derivatives of azacyclics for treating cns disorders
US4798841A (en) * 1987-03-31 1989-01-17 Warner-Lambert Company Tetrahydropyridine oxime cholinergic agents and method of treatment
EP0311313B1 (en) * 1987-10-05 1995-05-10 Yamanouchi Pharmaceutical Co. Ltd. Heterocyclic spiro compounds and their preparation
JPH0238175A (ja) * 1988-07-29 1990-02-07 Aisin Seiki Co Ltd ブレーキ圧制御装置

Also Published As

Publication number Publication date
GR900100476A (en) 1991-11-15
PT94440A (pt) 1991-02-08
GR1000887B (el) 1993-03-16
IE902242L (en) 1990-12-21
US5075317A (en) 1991-12-24
IE902242A1 (en) 1991-01-16
EP0490901A1 (en) 1992-06-24
FI96114C (fi) 1996-05-10
EP0490901A4 (en) 1992-04-13
CA2062809A1 (en) 1990-12-22
FI96114B (fi) 1996-01-31
WO1990015804A1 (en) 1990-12-27
JPH04506210A (ja) 1992-10-29

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Legal Events

Date Code Title Description
BB Publication of examined application
GB Transfer or assigment of application

Owner name: ASTRA AB

MM Patent lapsed