FI812270L - Antiinflammatoriska 4,5-diaryl-alfa-polyfluoralkyl-1h-imidazol-2-metanaminer - Google Patents

Antiinflammatoriska 4,5-diaryl-alfa-polyfluoralkyl-1h-imidazol-2-metanaminer

Info

Publication number
FI812270L
FI812270L FI812270A FI812270A FI812270L FI 812270 L FI812270 L FI 812270L FI 812270 A FI812270 A FI 812270A FI 812270 A FI812270 A FI 812270A FI 812270 L FI812270 L FI 812270L
Authority
FI
Finland
Prior art keywords
metanaminer
polyfluoralkyl
diaryl
imidazole
inflammatory
Prior art date
Application number
FI812270A
Other languages
English (en)
Inventor
Joel Gayton Whitney
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Publication of FI812270L publication Critical patent/FI812270L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI812270A 1980-07-21 1981-07-20 Antiinflammatoriska 4,5-diaryl-alfa-polyfluoralkyl-1h-imidazol-2-metanaminer FI812270L (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17087180A 1980-07-21 1980-07-21
US06/271,276 US4348404A (en) 1980-07-21 1981-06-15 Antiinflammatory 4,5-diaryl-α-polyfluoroalkyl-1H-imidazole-2-methanamines

Publications (1)

Publication Number Publication Date
FI812270L true FI812270L (fi) 1982-01-22

Family

ID=26866505

Family Applications (1)

Application Number Title Priority Date Filing Date
FI812270A FI812270L (fi) 1980-07-21 1981-07-20 Antiinflammatoriska 4,5-diaryl-alfa-polyfluoralkyl-1h-imidazol-2-metanaminer

Country Status (16)

Country Link
US (1) US4348404A (fi)
EP (1) EP0044486B1 (fi)
AU (1) AU7312581A (fi)
CA (1) CA1144552A (fi)
DE (1) DE3166949D1 (fi)
DK (1) DK323981A (fi)
ES (1) ES8301218A1 (fi)
FI (1) FI812270L (fi)
GR (1) GR76541B (fi)
HU (1) HU185938B (fi)
IL (1) IL63368A0 (fi)
NO (1) NO812484L (fi)
NZ (1) NZ197762A (fi)
PH (1) PH16513A (fi)
PT (1) PT73388B (fi)
YU (1) YU180181A (fi)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA826501B (en) * 1982-09-06 1984-04-25 Du Pont Anti-hypertensive imidazole derivative
US4478845A (en) * 1983-01-19 1984-10-23 E. I. Du Pont De Nemours And Company Antiinflammatory and/or analgesic imidazoimidazoles
US4632930A (en) * 1984-11-30 1986-12-30 E. I. Du Pont De Nemours And Company Antihypertensive alkyl-arylimidazole, thiazole and oxazole derivatives
NZ238688A (en) * 1990-06-28 1992-05-26 Smithkline Beecham Corp Substituted histidines: pharmaceutical compositions, preparation and uses thereof
US6426360B1 (en) * 1994-07-28 2002-07-30 G D Searle & Co. 4,5-substituted imidazolyl compounds for the treatment of inflammation
US5620999A (en) * 1994-07-28 1997-04-15 Weier; Richard M. Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation
US5700826A (en) * 1995-06-07 1997-12-23 Ontogen Corporation 1,2,4,5-tetra substituted imidazoles as modulators of multi-drug resistance
CA2295021A1 (en) * 1997-06-30 1999-01-28 Ortho-Mcneil Pharmaceutical, Inc. 2-substituted imidazoles useful in the treatment of inflammatory diseases
US5840721A (en) * 1997-07-09 1998-11-24 Ontogen Corporation Imidazole derivatives as MDR modulators
HUP0102058A3 (en) 1998-05-22 2002-05-28 Smithkline Beecham Corp Novel 2-alkyl substituted imidazole compounds, process for their preparation, pharmaceutical compositions containing them and their use
TWI292316B (en) * 1999-10-11 2008-01-11 Sod Conseils Rech Applic Pharmaceutical composition of thiazole derivatives intended to inhibit mao and/or lipidic peroxidation and/or to act as modulators of sodium channels and the use thereof
TR200201364T2 (tr) * 1999-11-22 2002-10-21 Smithkline Beecham P. L. C. Yeni bileşikler.
HUP0204144A3 (en) * 1999-12-17 2003-07-28 Procter & Gamble N-(1-phenylethyl)-5-phenyl-imidazole-2-amine compounds, their compositions and uses
US6596739B2 (en) 2000-03-29 2003-07-22 The Procter & Gamble Company N-(1-phenylethyl)-5-phenyl-imidazole-2-amine compounds, their compositions and uses
GB0112348D0 (en) * 2001-05-19 2001-07-11 Smithkline Beecham Plc Compounds
US20040192689A1 (en) * 2001-09-05 2004-09-30 Dean David Kenneth Heterocycle-carboxamide derivatives as raf kinase inhibitors
DE60304778T2 (de) 2002-08-30 2006-09-21 Ishida Co., Ltd. Display-Streifen

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2532547A (en) * 1950-12-05 Z-aminoalkyl-glyoxaline derivatives
US3197480A (en) * 1962-12-12 1965-07-27 Du Pont 2 and 2, 4-(alpha hydroxypolyperhalocycloalkyl)-thiophenes, pyrroles, and furans; 2 and 2, 4-[(alpha hydroxyalpha, alpha dipolyperhalo hydrocarbon) methyl]-thiophenes, pyrroles and furans and process for making them
US3707475A (en) * 1970-11-16 1972-12-26 Pfizer Antiinflammatory imidazoles
US3929807A (en) * 1971-05-10 1975-12-30 Ciba Geigy Corp 2-Substituted-4(5)-(aryl)-5(4)-(2,3 or -4-pyridyl)-imidazoles
BE793407A (fr) 1971-12-28 1973-06-28 Hoechst Ag Imidazolyl - (2) -carbinols ayant une activite hypolipidemique et leur procede de preparation
US4190666A (en) * 1975-08-11 1980-02-26 E. I. Du Pont De Nemours And Company Anti-inflammatory 4,5-diarly-2-(substituted-thio)imidazoles and their corresponding sulfoxides and sulfones
US4159338A (en) * 1977-02-09 1979-06-26 E. I. Du Pont De Nemours And Company Antiinflammatory-4,5-dicyclic-2-(substituted thio)-imidazoles and their corresponding sulfoxides and sulfones
DE2960506D1 (en) * 1978-04-24 1981-10-29 Dumex Ltd As Arylimidazoles, their synthesis and pharmaceutical or veterinary preparations containing them
US4199592A (en) * 1978-08-29 1980-04-22 E. I. Du Pont De Nemours And Company Antiinflammatory 4,5-diaryl-2-nitroimidazoles

Also Published As

Publication number Publication date
NO812484L (no) 1982-01-22
EP0044486A1 (en) 1982-01-27
PT73388A (en) 1981-08-01
CA1144552A (en) 1983-04-12
DE3166949D1 (de) 1984-12-06
YU180181A (en) 1984-02-29
AU7312581A (en) 1982-01-28
PH16513A (en) 1983-11-08
ES504121A0 (es) 1982-12-01
EP0044486B1 (en) 1984-10-31
PT73388B (en) 1983-09-14
GR76541B (fi) 1984-08-10
US4348404A (en) 1982-09-07
HU185938B (en) 1985-04-28
NZ197762A (en) 1984-09-28
DK323981A (da) 1982-01-22
ES8301218A1 (es) 1982-12-01
IL63368A0 (en) 1981-10-30

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Legal Events

Date Code Title Description
FD Application lapsed

Owner name: E.I. DU PONT DE NEMOURS AND COMPANY