FI773738A - PROCEDURE FOR THE FRAMSTATION OF AV N- (BENTSTIAZOL-2-YL) -OXAMIDYRA DERIVATIVES - Google Patents

PROCEDURE FOR THE FRAMSTATION OF AV N- (BENTSTIAZOL-2-YL) -OXAMIDYRA DERIVATIVES

Info

Publication number
FI773738A
FI773738A FI773738A FI773738A FI773738A FI 773738 A FI773738 A FI 773738A FI 773738 A FI773738 A FI 773738A FI 773738 A FI773738 A FI 773738A FI 773738 A FI773738 A FI 773738A
Authority
FI
Finland
Prior art keywords
oxamidyra
bentstiazol
framstation
derivatives
procedure
Prior art date
Application number
FI773738A
Other languages
Finnish (fi)
Other versions
FI57594B (en
FI57594C (en
Inventor
Werner Winter
Max Thiel
Androniki Roesch
Otto-Henning Wilhelms
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Publication of FI773738A publication Critical patent/FI773738A/en
Publication of FI57594B publication Critical patent/FI57594B/en
Application granted granted Critical
Publication of FI57594C publication Critical patent/FI57594C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/66Nitrogen atoms not forming part of a nitro radical
FI773738A 1976-12-14 1977-12-12 PROCEDURE FOR THE FRAMSTATION OF ANTI-ALLERGIC VERKSAMMA N- (BENTSTIAZOL-2-YL) -OXAMIDSYRA DERIVATIVES FI57594C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19762656468 DE2656468A1 (en) 1976-12-14 1976-12-14 N- (BENZTHIAZOL-2-YL) -OXAMID ACID DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF
DE2656468 1976-12-14

Publications (3)

Publication Number Publication Date
FI773738A true FI773738A (en) 1978-06-15
FI57594B FI57594B (en) 1980-05-30
FI57594C FI57594C (en) 1980-09-10

Family

ID=5995427

Family Applications (1)

Application Number Title Priority Date Filing Date
FI773738A FI57594C (en) 1976-12-14 1977-12-12 PROCEDURE FOR THE FRAMSTATION OF ANTI-ALLERGIC VERKSAMMA N- (BENTSTIAZOL-2-YL) -OXAMIDSYRA DERIVATIVES

Country Status (17)

Country Link
JP (1) JPS5377058A (en)
AR (1) AR216496A1 (en)
AT (1) AT360523B (en)
AU (1) AU510730B2 (en)
BE (1) BE861794A (en)
CS (1) CS203179B2 (en)
DD (1) DD133329A5 (en)
DE (1) DE2656468A1 (en)
ES (1) ES465034A1 (en)
FI (1) FI57594C (en)
FR (1) FR2374317A1 (en)
GB (1) GB1538822A (en)
HU (1) HU175340B (en)
NL (1) NL7713580A (en)
SE (1) SE7714074L (en)
SU (1) SU680647A3 (en)
ZA (1) ZA777236B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2676775A (en) * 1949-10-24 1954-04-27 Gustav O Schulz Electric flatiron cord holder
DE3017976A1 (en) * 1980-05-10 1981-11-19 Dr. Karl Thomae Gmbh, 7950 Biberach SUBSTITUTED 2-AMINO-5-HALOGEN-BENZOTHIAZOLES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS
US4321372A (en) 1980-06-16 1982-03-23 Pfizer Inc. Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides
DE3027527A1 (en) 1980-07-19 1982-02-18 Basf Ag, 6700 Ludwigshafen NEW OXAMID ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THERAPEUTIC AGENTS CONTAINING THEM
GB2090826B (en) * 1981-01-09 1985-06-12 Usv Pharma Corp New heterocyclic compounds useful as anti-allergie agents
DE3135250A1 (en) * 1981-09-05 1983-03-17 Basf Ag, 6700 Ludwigshafen TRICYCLIC THIAZOLYLOXAMATES, METHOD FOR THE PRODUCTION THEREOF AND THERAPEUTIC AGENTS CONTAINING THEM
US4826860A (en) * 1987-03-16 1989-05-02 Warner-Lambert Company Substituted 2-aminobenzothiazoles and derivatives useful as cerebrovascular agents
FI91859C (en) * 1987-06-17 1994-08-25 Eisai Co Ltd Analogue method for the preparation of an active benzothiazole derivative as an antiallergic agent
SI1303272T1 (en) 2000-06-21 2008-06-30 Hoffmann La Roche Benzothiazole derivatives for the treatment of alzheimer's disease and parkinson's disease
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
NZ550763A (en) 2004-05-24 2010-07-30 Hoffmann La Roche 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide
CA2586931C (en) 2004-11-05 2013-08-06 Paul Spurr Process for preparation of isonicotinic acid derivatives
DE602006012815D1 (en) 2005-03-23 2010-04-22 Hoffmann La Roche ACETYLENYLPYRAZOLOPYRIMIDIN DERIVATIVES AS MGLUR2 ANTAGONSTES
AU2006298829B2 (en) 2005-09-27 2011-03-03 F. Hoffmann-La Roche Ag Oxadiazolyl pyrazolo-pyrimidines as mGluR2 antagonists

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4150140A (en) * 1976-12-23 1979-04-17 The Upjohn Company Benzothiazolyl oxanic acids, esters and salts

Also Published As

Publication number Publication date
FI57594B (en) 1980-05-30
DD133329A5 (en) 1978-12-27
ATA890777A (en) 1980-06-15
SU680647A3 (en) 1979-08-15
JPS5377058A (en) 1978-07-08
AR216496A1 (en) 1979-12-28
GB1538822A (en) 1979-01-24
FI57594C (en) 1980-09-10
AT360523B (en) 1981-01-12
FR2374317B1 (en) 1980-11-07
CS203179B2 (en) 1981-02-27
HU175340B (en) 1980-07-28
AU510730B2 (en) 1980-07-10
NL7713580A (en) 1978-06-16
ZA777236B (en) 1978-11-29
FR2374317A1 (en) 1978-07-13
ES465034A1 (en) 1978-09-01
SE7714074L (en) 1978-06-15
BE861794A (en) 1978-06-13
AU3137777A (en) 1979-06-14
DE2656468A1 (en) 1978-06-15

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Legal Events

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MM Patent lapsed

Owner name: BOEHRINGER MANNHEIM GMBH