ES8801921A1 - Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados - Google Patents

Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados

Info

Publication number
ES8801921A1
ES8801921A1 ES557728A ES557728A ES8801921A1 ES 8801921 A1 ES8801921 A1 ES 8801921A1 ES 557728 A ES557728 A ES 557728A ES 557728 A ES557728 A ES 557728A ES 8801921 A1 ES8801921 A1 ES 8801921A1
Authority
ES
Spain
Prior art keywords
preparation
medicaments
quinolone
bridged
well
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES557728A
Other languages
English (en)
Other versions
ES557728A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of ES8801921A1 publication Critical patent/ES8801921A1/es
Publication of ES557728A0 publication Critical patent/ES557728A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)

Abstract

LOS ACIDOS 4-QUINOLON-3-CARBOXILICOS 1,8-PUENTEADOS Y SUS DERIVADOS (I), DONDE NO EXCLUSIVAMENTE, Y ES UN CARBOXILO O NITRILO, X1 HIDROGENO O NITRO, X5 HALOGENO, R1010 Y R11 FORMAN CON SU N UN HETEROCICLO DE 5 O 6 MIEMBROS; R1, R2 Y R3 ALQUILO C1-2 Y R Y R4, R5 Y R6 ALQUILO C1-6; SE OBTIENE POR REACCIONDE DERIVADOS DEL ACIDO 11-(1-PIPEROZINIL) QUINOLONCARBOXILICO (II) (NF1) CON ACEPTORES DE MICHAEL (III), DONDE B ES CN Y OTROS. FARMACEUTICAMENTE APLICABLES EN EL TRATAMIENTO DE INFECCIONES EN MEDICINA Y VETERINARIA.
ES557728A 1985-06-22 1987-09-15 Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados Expired ES8801921A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19853522405 DE3522405A1 (de) 1985-06-22 1985-06-22 1,8-verbrueckte 4-chinolon-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende arzneimittel und ihre verwendung zur herstellung von arzneimitteln

Publications (2)

Publication Number Publication Date
ES8801921A1 true ES8801921A1 (es) 1988-03-01
ES557728A0 ES557728A0 (es) 1988-03-01

Family

ID=6273929

Family Applications (3)

Application Number Title Priority Date Filing Date
ES556369A Expired ES8802301A1 (es) 1985-06-22 1986-06-20 Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8- puenteados.
ES557728A Expired ES8801921A1 (es) 1985-06-22 1987-09-15 Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados
ES557727A Expired ES8802050A1 (es) 1985-06-22 1987-09-15 Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES556369A Expired ES8802301A1 (es) 1985-06-22 1986-06-20 Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8- puenteados.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES557727A Expired ES8802050A1 (es) 1985-06-22 1987-09-15 Procedimiento para la obtencion de acidos 4-quinolon-3-carboxilicos 1,8-puenteados

Country Status (17)

Country Link
US (1) US4847375A (es)
EP (1) EP0206076A3 (es)
JP (1) JPS62490A (es)
KR (1) KR870000337A (es)
CN (1) CN86104256A (es)
AU (1) AU564013B2 (es)
DE (1) DE3522405A1 (es)
DK (1) DK291886A (es)
ES (3) ES8802301A1 (es)
FI (1) FI862640A (es)
GR (1) GR861602B (es)
HU (1) HU195662B (es)
IL (1) IL79163A0 (es)
NO (1) NO862198L (es)
NZ (1) NZ216598A (es)
PT (1) PT82802B (es)
ZA (1) ZA864604B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3623757A1 (de) * 1986-07-15 1988-01-21 Bayer Ag Neue 1,8-verbrueckte 4-chinoloncarbonsaeuren und diese enthaltende arzneimittel
JPH0228178A (ja) * 1988-04-23 1990-01-30 Toyama Chem Co Ltd 新規なピリドンカルボン酸誘導体およびその塩並びにそれらの製造法
US5286723A (en) * 1988-08-31 1994-02-15 Daiichi Seiyaku Co., Ltd. Spiro compound
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
JPH10127313A (ja) * 1996-10-31 1998-05-19 Ykk Corp 自動停止装置付スライドファスナー用スライダー
US6673793B2 (en) 2000-07-12 2004-01-06 Pharmacia & Upjohn Co. Oxazinoquinolones useful for the treatment of viral infections
JP3927922B2 (ja) 2003-05-21 2007-06-13 Ｙｋｋ株式会社 スライドファスナー用スプリング体及び同スプリング体が装着されたスライダー
PL2383271T3 (pl) * 2006-03-13 2013-12-31 Kyorin Seiyaku Kk Aminochinolony jako inhibitory GSK-3
MX2010002667A (es) * 2007-09-11 2010-04-01 Activx Biosciences Inc Cianoaminoquinolonas y tetrazoloaminoquinolonas como inhibidores de gsk-3.
BRPI0816814B1 (pt) 2007-09-12 2021-08-31 Kyorin Pharmaceutical Co. Ltd Composto, composição farmacêutica e uso de um composto
AU2010221990B2 (en) * 2009-03-11 2015-06-04 Kyorin Pharmaceutical Co., Ltd. 7-cycloalkylaminoquinolones as GSK-3 inhibitors

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5746986A (en) * 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
JPS57149286A (en) * 1981-03-13 1982-09-14 Dai Ichi Seiyaku Co Ltd 8-aminopyrido(1,2,3-de)(1,4)banzoxazine derivative
DE3122911C2 (de) * 1981-06-10 1983-04-28 Benckiser-Knapsack Gmbh, 6802 Ladenburg Verfahren zum Deinken von bedrucktem Altpapier
PH22140A (en) * 1982-06-29 1988-06-01 Daiichi Seiyaku Co Tricyclic compounds
US4443447A (en) * 1982-10-25 1984-04-17 Riker Laboratories, Inc. Phenyl-substituted tricyclic antibacterial agents
JPS59137482A (ja) * 1983-01-26 1984-08-07 Otsuka Pharmaceut Co Ltd ピロロ〔３，２，１，−ｉｊ〕キノリン−５−カルボン酸誘導体
US4473568A (en) * 1983-03-01 1984-09-25 Warner Lambert Company Antibacterial thiazolidine or thiomorpholine substituted quinolines
US4571396A (en) * 1984-04-16 1986-02-18 Warner-Lambert Company Antibacterial agents
EP0160284B1 (en) * 1984-04-26 1990-10-24 Abbott Laboratories Quino-benoxazine antibacterial compounds
US4771054A (en) * 1985-01-23 1988-09-13 Warner-Lambert Company Antibacterial agents
DE3522406A1 (de) * 1985-06-22 1987-01-02 Bayer Ag Verfahren zur herstellung von 1,8-verbrueckten 4-chinolon-3-carbonsaeuren
DE3600891A1 (de) * 1986-01-15 1987-07-16 Bayer Ag 1,8-verbrueckte 4-chinolon-3-carbonsaeuren und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
GR861602B (en) 1986-10-20
CN86104256A (zh) 1987-03-18
FI862640A0 (fi) 1986-06-19
NO862198L (no) 1986-12-23
AU5920786A (en) 1987-02-05
JPS62490A (ja) 1987-01-06
DE3522405A1 (de) 1987-01-02
DK291886A (da) 1986-12-23
HUT44256A (en) 1988-02-29
PT82802A (en) 1986-07-01
AU564013B2 (en) 1987-07-30
NO862198D0 (no) 1986-06-03
IL79163A0 (en) 1986-09-30
PT82802B (en) 1988-05-23
ES8802301A1 (es) 1988-05-01
EP0206076A3 (de) 1988-07-27
HU195662B (en) 1988-06-28
US4847375A (en) 1989-07-11
KR870000337A (ko) 1987-02-17
DK291886D0 (da) 1986-06-20
ES556369A0 (es) 1988-05-01
EP0206076A2 (de) 1986-12-30
NZ216598A (en) 1989-07-27
FI862640A (fi) 1986-12-23
ES557728A0 (es) 1988-03-01
ES8802050A1 (es) 1988-03-16
ZA864604B (en) 1987-02-25
ES557727A0 (es) 1988-03-16

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