ES548472A0 - Un procedimiento para la preparacion de una macrolida - Google Patents

Un procedimiento para la preparacion de una macrolida

Info

Publication number
ES548472A0
ES548472A0 ES548472A ES548472A ES548472A0 ES 548472 A0 ES548472 A0 ES 548472A0 ES 548472 A ES548472 A ES 548472A ES 548472 A ES548472 A ES 548472A ES 548472 A0 ES548472 A0 ES 548472A0
Authority
ES
Spain
Prior art keywords
macrolide
procedure
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES548472A
Other languages
English (en)
Other versions
ES8607336A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES8607336A1 publication Critical patent/ES8607336A1/es
Publication of ES548472A0 publication Critical patent/ES548472A0/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Fodder In General (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ES548472A 1982-09-13 1985-10-31 Un procedimiento para la preparacion de una macrolida Expired ES8607336A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41724782A 1982-09-13 1982-09-13

Publications (2)

Publication Number Publication Date
ES8607336A1 ES8607336A1 (es) 1986-06-01
ES548472A0 true ES548472A0 (es) 1986-06-01

Family

ID=23653182

Family Applications (2)

Application Number Title Priority Date Filing Date
ES525544A Expired ES8604596A1 (es) 1982-09-13 1983-09-12 Un procedimiento para la preparacion de una macrolida
ES548472A Expired ES8607336A1 (es) 1982-09-13 1985-10-31 Un procedimiento para la preparacion de una macrolida

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES525544A Expired ES8604596A1 (es) 1982-09-13 1983-09-12 Un procedimiento para la preparacion de una macrolida

Country Status (34)

Country Link
EP (1) EP0103465B1 (es)
JP (1) JPS5973598A (es)
KR (1) KR850000961B1 (es)
AR (1) AR241595A1 (es)
AT (1) AT381707B (es)
AU (1) AU561147B2 (es)
BG (1) BG42675A3 (es)
CA (1) CA1243310A (es)
CS (1) CS259862B2 (es)
CY (1) CY1417A (es)
DD (1) DD210284A5 (es)
DE (1) DE3366097D1 (es)
DK (1) DK153555C (es)
EG (1) EG16287A (es)
ES (2) ES8604596A1 (es)
FI (1) FI73222C (es)
GB (1) GB2127017B (es)
GR (1) GR79067B (es)
HK (1) HK21888A (es)
HU (1) HU194271B (es)
IE (1) IE55916B1 (es)
IL (1) IL69666A (es)
LU (1) LU90240I2 (es)
MY (1) MY8700756A (es)
NL (1) NL950001I2 (es)
NZ (1) NZ205501A (es)
PH (1) PH23242A (es)
PL (2) PL142304B1 (es)
PT (1) PT77335B (es)
RO (1) RO89235A (es)
SG (1) SG99287G (es)
SU (1) SU1375135A3 (es)
UA (1) UA6045A1 (es)
ZA (1) ZA836741B (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59181294A (ja) * 1983-03-30 1984-10-15 Satoshi Omura 抗生物質ptl−448とその誘導体およびそれらの製造方法
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
EP0262903A3 (en) * 1986-09-29 1988-11-02 Eli Lilly And Company New acyl derivatives of 20-modified tylosin and desmycosin compounds
US4820694A (en) * 1986-09-29 1989-04-11 Eli Lilly And Company Modifications of 3-O-demethylmycinose in macrocin and lactenocin
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW226373B (es) * 1992-07-15 1994-07-11 Pfizer
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
WO1996009312A1 (en) * 1994-09-22 1996-03-28 Pfizer Inc. Antibiotic macrolides
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
US6605599B1 (en) 1997-07-08 2003-08-12 Bristol-Myers Squibb Company Epothilone derivatives
SI0948967T1 (en) * 1998-03-02 2005-06-30 Eli Lilly And Company Treatment of viral disease in swine
EP2019112A1 (en) 2007-07-26 2009-01-28 Intervet International BV Macrolide solid-state forms
CA2657483C (en) 2006-07-28 2012-10-09 Intervet International B.V. Macrolide synthesis process
RU2497803C2 (ru) * 2007-12-07 2013-11-10 ЭЙСАЙ Ар ЭНД Ди МЕНЕДЖМЕНТ КО., ЛТД Промежуточные продукты в синтезе аналогов зеараленоновых макролидов
PE20160207A1 (es) * 2013-05-23 2016-05-22 Kitasato Inst Derivados de tilosina y metodo para su preparacion
CN103880903B (zh) * 2014-03-21 2016-06-15 烟台万润药业有限公司 一种泰乐菌素类大环内酯及其衍生物的制备方法
CN117510561B (zh) * 2023-11-30 2024-04-02 中国农业科学院饲料研究所 一种泰乐菌素衍生物及其制备方法与应用
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE32839B1 (en) * 1967-12-04 1973-12-28 Lilly Co Eli Urea-antibiotic adducts and process for preparing the same
US4279896A (en) * 1980-06-23 1981-07-21 Schering Corporation Novel 20-imino macrolide antibacterial agents
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質

Also Published As

Publication number Publication date
GB2127017A (en) 1984-04-04
ATA320683A (de) 1986-04-15
PL243718A1 (en) 1985-04-09
SG99287G (en) 1988-09-23
DK153555C (da) 1988-12-05
FI833229A (fi) 1984-03-14
GB2127017B (en) 1986-01-15
PL250619A1 (en) 1985-07-30
PT77335A (en) 1983-10-01
PL142304B1 (en) 1987-10-31
DK413783D0 (da) 1983-09-12
HUT35272A (en) 1985-06-28
EG16287A (en) 1987-04-30
HU194271B (en) 1988-01-28
PH23242A (en) 1989-06-06
UA6045A1 (uk) 1994-12-29
NL950001I2 (nl) 1997-05-01
ZA836741B (en) 1984-04-25
PL142251B1 (en) 1987-10-31
GR79067B (es) 1984-10-02
JPS5973598A (ja) 1984-04-25
JPH021840B2 (es) 1990-01-12
AU561147B2 (en) 1987-04-30
DE3366097D1 (en) 1986-10-16
FI73222B (fi) 1987-05-29
NZ205501A (en) 1985-09-13
ES8607336A1 (es) 1986-06-01
AU1871083A (en) 1984-03-22
IL69666A (en) 1987-10-20
ES8604596A1 (es) 1986-02-01
IE832131L (en) 1984-03-13
CY1417A (en) 1988-04-22
FI833229A0 (fi) 1983-09-09
ES525544A0 (es) 1986-02-01
MY8700756A (en) 1987-12-31
DK153555B (da) 1988-07-25
EP0103465A1 (en) 1984-03-21
IE55916B1 (en) 1991-02-27
GB8324044D0 (en) 1983-10-12
LU90240I2 (fr) 1998-07-06
IL69666A0 (en) 1983-12-30
KR840005734A (ko) 1984-11-15
CS665383A2 (en) 1988-04-15
PT77335B (en) 1986-05-19
AT381707B (de) 1986-11-25
NL950001I1 (nl) 1995-02-16
AR241595A1 (es) 1992-09-30
DD210284A5 (de) 1984-06-06
CS259862B2 (en) 1988-11-15
KR850000961B1 (ko) 1985-07-02
SU1375135A3 (ru) 1988-02-15
BG42675A3 (en) 1988-01-15
HK21888A (en) 1988-03-31
DK413783A (da) 1984-03-14
EP0103465B1 (en) 1986-09-10
FI73222C (fi) 1987-09-10
RO89235A (ro) 1986-03-15
CA1243310A (en) 1988-10-18

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20051219