ES530153A0 - Un procedimiento para la preparacion de compuestos de beta-lactama - Google Patents

Un procedimiento para la preparacion de compuestos de beta-lactama

Info

Publication number
ES530153A0
ES530153A0 ES530153A ES530153A ES530153A0 ES 530153 A0 ES530153 A0 ES 530153A0 ES 530153 A ES530153 A ES 530153A ES 530153 A ES530153 A ES 530153A ES 530153 A0 ES530153 A0 ES 530153A0
Authority
ES
Spain
Prior art keywords
lactama
beta
compounds
procedure
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES530153A
Other languages
English (en)
Other versions
ES8605810A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838305704A external-priority patent/GB8305704D0/en
Priority claimed from GB838330516A external-priority patent/GB8330516D0/en
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of ES530153A0 publication Critical patent/ES530153A0/es
Publication of ES8605810A1 publication Critical patent/ES8605810A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/04Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/10Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568Four-membered rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES530153A 1983-03-02 1984-02-29 Un procedimiento para la preparacion de compuestos de beta-lactama Expired ES8605810A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB838305704A GB8305704D0 (en) 1983-03-02 1983-03-02 Beta-lactam compounds
GB838330516A GB8330516D0 (en) 1983-11-16 1983-11-16 Compounds

Publications (2)

Publication Number Publication Date
ES530153A0 true ES530153A0 (es) 1986-04-01
ES8605810A1 ES8605810A1 (es) 1986-04-01

Family

ID=26285399

Family Applications (3)

Application Number Title Priority Date Filing Date
ES530153A Expired ES8605810A1 (es) 1983-03-02 1984-02-29 Un procedimiento para la preparacion de compuestos de beta-lactama
ES537351A Granted ES537351A0 (es) 1983-03-02 1984-11-02 Un procedimiento para la preparacion de compuestos de -lactama
ES537350A Granted ES537350A0 (es) 1983-03-02 1984-11-02 Un procedimiento para la preparacion de compuestos de -lactama

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES537351A Granted ES537351A0 (es) 1983-03-02 1984-11-02 Un procedimiento para la preparacion de compuestos de -lactama
ES537350A Granted ES537350A0 (es) 1983-03-02 1984-11-02 Un procedimiento para la preparacion de compuestos de -lactama

Country Status (5)

Country Link
EP (1) EP0120613A1 (es)
AU (1) AU568119B2 (es)
ES (3) ES8605810A1 (es)
GR (1) GR79528B (es)
NZ (1) NZ207315A (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI82471C (fi) * 1984-01-26 1991-03-11 Beecham Group Plc Foerfarande foer framstaellning av farmakologiskt aktiva 6-metylenpenemderivater.
GB8518416D0 (en) * 1985-07-22 1985-08-29 Beecham Group Plc Compounds
GB8518422D0 (en) * 1985-07-22 1985-08-29 Beecham Group Plc Compounds
DE3618813A1 (de) * 1986-06-04 1987-12-10 Hoechst Ag Pharmazeutische zubereitung zur behandlung bakterieller infektionen
GB8711391D0 (en) * 1987-05-14 1987-06-17 Beecham Group Plc Process
CA2105746A1 (en) * 1992-09-09 1994-03-10 Akira Yoshida Process for preparing carbapenem and penem compounds and new compounds involved in that process
US6472383B1 (en) 1994-04-25 2002-10-29 Smithkline Beecham P.L.C. Pharmaceutical formulations
CN1094353C (zh) * 1994-04-25 2002-11-20 史密斯克莱·比奇曼公司 含有β-内酰胺酶抑制性青霉烯与β-内酰胺抗生素复合的药物制剂及其在治疗细菌感染中的应用
US5629306A (en) * 1994-12-09 1997-05-13 Research Corporation Technologies, Inc. 7-alkylidene cephalosporanic acid derivatives and methods of using the same
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
AR039774A1 (es) 2002-05-01 2005-03-02 Wyeth Corp 6-alquiliden-penems biciclicos como inhibidores de beta-lactamasas
AR039475A1 (es) 2002-05-01 2005-02-23 Wyeth Corp 6-alquiliden-penems triciclicos como inhibidores de beta-lactamasa
EP2167081B1 (en) 2007-05-21 2013-06-26 Hans Rudolf Pfaendler Bactericidal anti-mrsa active pharmaceutical composition containing carbapenems

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3176517D1 (en) * 1980-04-24 1987-12-17 Beecham Group Plc Beta-lactam compounds, their preparation and use
CA1180005A (en) * 1980-10-24 1984-12-27 Solange Adam-Molina .beta.-LACTAMS

Also Published As

Publication number Publication date
ES8603404A1 (es) 1985-12-16
ES537351A0 (es) 1985-12-16
GR79528B (es) 1984-10-30
AU2518984A (en) 1984-09-06
NZ207315A (en) 1987-07-31
AU568119B2 (en) 1987-12-17
EP0120613A1 (en) 1984-10-03
ES8605810A1 (es) 1986-04-01
ES8507146A1 (es) 1985-08-16
ES537350A0 (es) 1985-08-16

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