ES378467A1 - Novel aminopiperidines, processes for their preparation, and compositions incorporating them - Google Patents
Novel aminopiperidines, processes for their preparation, and compositions incorporating themInfo
- Publication number
- ES378467A1 ES378467A1 ES378467A ES378467A ES378467A1 ES 378467 A1 ES378467 A1 ES 378467A1 ES 378467 A ES378467 A ES 378467A ES 378467 A ES378467 A ES 378467A ES 378467 A1 ES378467 A1 ES 378467A1
- Authority
- ES
- Spain
- Prior art keywords
- radical
- preparation
- aminopiperidines
- novel
- processes
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/02—Preparation by ring-closure or hydrogenation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Procedure for the preparation of aminopiperidine derivatives, of formula: **(See formula)** wherein each of R1, R2 and R3 are hydrogen or lower alkoxy, which can be independently exchanged, and the substituted benzamide radical is attached to positions 2, 3 or 4 of the piperidine nucleus, and R'1 and R' 2 are hydrogen or an amino radical and at least one of R'1 and R'2 represents an amino radical, characterized in that it comprises hydrogenating the compound of formula: **(See formula)** wherein R1, R2, R3 and the position of the substituted benzamide radical are defined as above and R''1 and R''2 represent hydrogen or a nitro radical and at least one of R''1 and r'' 2 means the nitro radical. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5165169A JPS4939679B1 (en) | 1969-06-30 | 1969-06-30 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES378467A1 true ES378467A1 (en) | 1972-06-16 |
Family
ID=12892751
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES369746A Expired ES369746A1 (en) | 1969-06-30 | 1969-07-22 | Novel aminopiperidines, processes for their preparation, and compositions incorporating them |
ES378467A Expired ES378467A1 (en) | 1969-06-30 | 1970-04-11 | Novel aminopiperidines, processes for their preparation, and compositions incorporating them |
ES378466A Expired ES378466A1 (en) | 1969-06-30 | 1970-04-11 | Novel aminopiperidines, processes for their preparation, and compositions incorporating them |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES369746A Expired ES369746A1 (en) | 1969-06-30 | 1969-07-22 | Novel aminopiperidines, processes for their preparation, and compositions incorporating them |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES378466A Expired ES378466A1 (en) | 1969-06-30 | 1970-04-11 | Novel aminopiperidines, processes for their preparation, and compositions incorporating them |
Country Status (8)
Country | Link |
---|---|
JP (1) | JPS4939679B1 (en) |
BE (1) | BE736840A (en) |
BR (2) | BR7020067D0 (en) |
CA (1) | CA931574A (en) |
DE (2) | DE1938512C3 (en) |
ES (3) | ES369746A1 (en) |
FR (1) | FR2048024B1 (en) |
GB (2) | GB1276813A (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2534255B1 (en) * | 1982-10-11 | 1985-07-12 | Delalande Sa | NOVEL 4-AROYLAMINO PIPERIDINE DERIVATIVES, PREPARATION METHOD THEREOF AND THERAPEUTIC APPLICATION THEREOF |
GB8419103D0 (en) * | 1984-07-26 | 1984-08-30 | Beecham Wuelfing Gmbh & Co Kg | Compounds |
AUPP818099A0 (en) * | 1999-01-14 | 1999-02-11 | Fujisawa Pharmaceutical Co., Ltd. | New n-containing heterocyclic compounds |
GB0325956D0 (en) * | 2003-11-06 | 2003-12-10 | Addex Pharmaceuticals Sa | Novel compounds |
EP1778229A4 (en) * | 2004-08-10 | 2009-06-17 | Incyte Corp | Amido compounds and their use as pharmaceuticals |
EP3375778A1 (en) * | 2017-03-14 | 2018-09-19 | Artax Biopharma Inc. | Aryl-piperidine derivatives |
-
1969
- 1969-06-30 JP JP5165169A patent/JPS4939679B1/ja active Pending
- 1969-07-21 CA CA057606A patent/CA931574A/en not_active Expired
- 1969-07-22 ES ES369746A patent/ES369746A1/en not_active Expired
- 1969-07-29 DE DE19691938512 patent/DE1938512C3/en not_active Expired
- 1969-07-29 DE DE19691967324 patent/DE1967324C2/en not_active Expired
- 1969-07-31 BE BE736840D patent/BE736840A/xx not_active IP Right Cessation
- 1969-10-14 FR FR6935135A patent/FR2048024B1/fr not_active Expired
-
1970
- 1970-01-30 GB GB4350071A patent/GB1276813A/en not_active Expired
- 1970-01-30 GB GB452270A patent/GB1276812A/en not_active Expired
- 1970-04-11 ES ES378467A patent/ES378467A1/en not_active Expired
- 1970-04-11 ES ES378466A patent/ES378466A1/en not_active Expired
- 1970-06-26 BR BR22006770A patent/BR7020067D0/en unknown
- 1970-06-29 BR BR21133970A patent/BR7011339D0/en unknown
Also Published As
Publication number | Publication date |
---|---|
BE736840A (en) | 1969-12-31 |
DE1967324C2 (en) | 1982-04-22 |
GB1276812A (en) | 1972-06-07 |
DE1938512C3 (en) | 1982-05-06 |
GB1276813A (en) | 1972-06-07 |
DE1938512A1 (en) | 1971-01-14 |
BR7011339D0 (en) | 1973-02-13 |
FR2048024B1 (en) | 1973-04-27 |
BR7020067D0 (en) | 1973-03-07 |
JPS4939679B1 (en) | 1974-10-28 |
FR2048024A1 (en) | 1971-03-19 |
ES369746A1 (en) | 1971-04-01 |
CA931574A (en) | 1973-08-07 |
ES378466A1 (en) | 1972-06-16 |
DE1938512B2 (en) | 1981-07-16 |
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