ES2070772B1 - DERIVATIVES OF ACILAMINOINDOL - Google Patents

DERIVATIVES OF ACILAMINOINDOL

Info

Publication number
ES2070772B1
ES2070772B1 ES9301772A ES9301772A ES2070772B1 ES 2070772 B1 ES2070772 B1 ES 2070772B1 ES 9301772 A ES9301772 A ES 9301772A ES 9301772 A ES9301772 A ES 9301772A ES 2070772 B1 ES2070772 B1 ES 2070772B1
Authority
ES
Spain
Prior art keywords
compounds
disorders
yigrah
treatment
useful
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
ES9301772A
Other languages
Spanish (es)
Other versions
ES2070772A1 (en
Inventor
John E Macor
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Priority to ES9301772A priority Critical patent/ES2070772B1/en
Publication of ES2070772A1 publication Critical patent/ES2070772A1/en
Application granted granted Critical
Publication of ES2070772B1 publication Critical patent/ES2070772B1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

COMPUESTOS DE LA FORMULA *FIG* EN LA QUE N, M, Y Y W, R1, R2 Y R6 SE DEFINEN DETALLADAMENTE EN LA MEMORIA. ESTOS COMPUESTOS SON UTILES EN EL TRATAMIENTO DE MIGRAÑAS Y OTROS TRASTORNOS. ESTOS COMPUESTOS SON PSICOTERAPEUTICOS UTILES Y SON AGONISTAS DE SEROTONINA (5-HT1) POTENTES Y SE PUEDEN EMPLEAR EN EL TRATAMIENTO DE DEPRESION, ANSIEDAD, TRASTORNOS DEL APETITO, OBESIDAD, ABUSO DE DROGAS, CEFALEA AGRUPADA, MIGRAÑA, DOLOR, Y HEMICRANEA PAROXISTICA CRONICA Y CEFALEA ASOCIADA CON TRASTORNOS VASCULARES, Y OTROS TRASTORNOS QUE PROCEDEN DE NEUROTRANSMISION SEROTONERGICA DEFICIENTE. LOS COMPUESTOS SE PUEDEN EMPLEAR TAMBIEN COMO ANTIHIPERTENSORES Y VASODILATADORES QUE ACTUAN CENTRALMENTE.COMPOUNDS OF THE FORMULA * FIG * IN WHICH N, M, Y AND W, R1, R2 AND R6 ARE DEFINED IN DETAIL IN MEMORY. THESE COMPOUNDS ARE USEFUL IN THE TREATMENT OF MIGRAINS AND OTHER DISORDERS. THESE COMPOUNDS ARE USEFUL PSYCHOTHERAPEUTICS AND ARE POWERFUL SEROTONINE (5-HT1) AGONISTS AND MAY BE USED IN THE TREATMENT OF DEPRESSION, ANXIETY, APPETITE DISORDERS, OBESITY, DRUG ABUSE, YICRA, YIGRAH, YIGRAH, YIGRAH, MIGRAINE HEADACHE ASSOCIATED WITH VASCULAR DISORDERS, AND OTHER DISORDERS THAT PROCEED FROM DEFICIENT SEROTONERGIC NEUROTRANSMISSION. THE COMPOUNDS MAY ALSO BE USED AS ANTI-HYPERTENSIONERS AND VASODILATORS THAT ACT CENTRALLY.

ES9301772A 1993-08-09 1993-08-09 DERIVATIVES OF ACILAMINOINDOL Expired - Fee Related ES2070772B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ES9301772A ES2070772B1 (en) 1993-08-09 1993-08-09 DERIVATIVES OF ACILAMINOINDOL

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES9301772A ES2070772B1 (en) 1993-08-09 1993-08-09 DERIVATIVES OF ACILAMINOINDOL

Publications (2)

Publication Number Publication Date
ES2070772A1 ES2070772A1 (en) 1995-06-01
ES2070772B1 true ES2070772B1 (en) 1996-02-16

Family

ID=8282816

Family Applications (1)

Application Number Title Priority Date Filing Date
ES9301772A Expired - Fee Related ES2070772B1 (en) 1993-08-09 1993-08-09 DERIVATIVES OF ACILAMINOINDOL

Country Status (1)

Country Link
ES (1) ES2070772B1 (en)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ197998A (en) * 1980-08-12 1985-08-16 Glaxo Group Ltd 5-amino(methyl)-1h-indol-3-ylalkaneamines
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
RU2095360C1 (en) * 1990-10-15 1997-11-10 Пфайзер Инк. Indole derivatives, their optical isomers and pharmaceutically acceptable salts
DE69307875T2 (en) * 1992-04-10 1997-05-22 Pfizer ACYLAMINOINDOL DERIVATIVES AS 5-HT1 AGONISTS

Also Published As

Publication number Publication date
ES2070772A1 (en) 1995-06-01

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20050810