EP1789055A4 - Thiazolopyridine kinase inhibitors - Google Patents
Thiazolopyridine kinase inhibitorsInfo
- Publication number
- EP1789055A4 EP1789055A4 EP05810363A EP05810363A EP1789055A4 EP 1789055 A4 EP1789055 A4 EP 1789055A4 EP 05810363 A EP05810363 A EP 05810363A EP 05810363 A EP05810363 A EP 05810363A EP 1789055 A4 EP1789055 A4 EP 1789055A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- thiazolopyridine
- kinase inhibitors
- kinase
- inhibitors
- thiazolopyridine kinase
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D497/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D497/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D497/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US60999204P | 2004-09-15 | 2004-09-15 | |
PCT/US2005/032837 WO2006031929A2 (en) | 2004-09-15 | 2005-09-15 | Thiazolopyridine kinase inhibitors |
Publications (2)
Publication Number | Publication Date |
---|---|
EP1789055A2 EP1789055A2 (en) | 2007-05-30 |
EP1789055A4 true EP1789055A4 (en) | 2009-11-11 |
Family
ID=36060693
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP05810363A Withdrawn EP1789055A4 (en) | 2004-09-15 | 2005-09-15 | Thiazolopyridine kinase inhibitors |
Country Status (6)
Country | Link |
---|---|
US (1) | US7659284B2 (en) |
EP (1) | EP1789055A4 (en) |
JP (1) | JP2008513463A (en) |
CN (1) | CN101056639A (en) |
AU (1) | AU2005284796A1 (en) |
WO (1) | WO2006031929A2 (en) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20070619A1 (en) * | 2005-09-27 | 2007-07-02 | Wyeth Corp | I HAVE (2,3-b) PYRIDIN-5-CARBONITRILES AS PROTEIN KINASE INHIBITORS |
AU2007207607B2 (en) * | 2006-01-17 | 2012-04-19 | Stiefel Laboratories, Inc. | Treatment of inflammatory disorders with triazole compounds |
EP2117544A4 (en) * | 2006-12-19 | 2010-03-03 | Univ Texas | Biomarker identifying the reactivation of stat3 after src inhibition |
US20100034816A1 (en) * | 2006-12-22 | 2010-02-11 | Novelix Therapeutics Gmbh | Treatment of Diabetes by at Least One Epidermal Growth Factor Receptor Specific Antibody or a Derivative Thereof |
WO2008094602A2 (en) * | 2007-01-30 | 2008-08-07 | Biogen Idec Ma Inc. | 1-h-pyrazolo (3,4b) pyrimidine derivatives and their use as modulators of mitotic kinases |
JO3793B1 (en) | 2015-12-10 | 2021-01-31 | Janssen Pharmaceutica Nv | Inhibitors of bruton’s tyrosine kinase and methods of their use |
JO3794B1 (en) | 2015-12-10 | 2021-01-31 | Janssen Pharmaceutica Nv | Polycyclic compounds as inhibitors of bruton's tyrosine kinase |
WO2018103058A1 (en) * | 2016-12-09 | 2018-06-14 | Janssen Pharmaceutica Nv | Inhibitors of bruton's tyrosine kinase and methods of their use |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0284567B1 (en) | 1987-03-27 | 1995-03-01 | Ciba-Geigy Ag | Cationic azo dyes |
DD285982A5 (en) | 1989-11-08 | 1991-01-10 | Wilhelm-Pieck-Universitaet Rostock,Sektion Chemie,Dd | METHOD FOR THE PRODUCTION OF SUBSTITUTED THIAZOLO [4,5-B] -PYRIDINES |
AU3766897A (en) | 1996-07-13 | 1998-02-09 | Glaxo Group Limited | Fused heterocyclic compounds as protein tyrosine kinase inhibitors |
US6232320B1 (en) | 1998-06-04 | 2001-05-15 | Abbott Laboratories | Cell adhesion-inhibiting antiinflammatory compounds |
US6452014B1 (en) | 2000-12-22 | 2002-09-17 | Geron Corporation | Telomerase inhibitors and methods of their use |
CN100343238C (en) | 2001-11-03 | 2007-10-17 | 阿斯特拉曾尼卡有限公司 | Quinazoline derivatives as antitumor agents |
US20040127395A1 (en) | 2002-09-06 | 2004-07-01 | Desai Pragnya J. | Use of histamine H4 receptor modulators for the treatment of allergy and asthma |
RU2005106274A (en) | 2002-09-06 | 2005-11-10 | Янссен Фармацевтика, Н.В. (Be) | HETEROCYCLIC COMPOUNDS |
EP1567506A4 (en) | 2002-11-20 | 2007-06-20 | Array Biopharma Inc | Cyanoguanidines and cyanoamidines as erbb2 and egfr inhibitors |
-
2005
- 2005-09-15 US US11/226,961 patent/US7659284B2/en not_active Expired - Fee Related
- 2005-09-15 AU AU2005284796A patent/AU2005284796A1/en not_active Abandoned
- 2005-09-15 WO PCT/US2005/032837 patent/WO2006031929A2/en active Application Filing
- 2005-09-15 CN CNA2005800389019A patent/CN101056639A/en active Pending
- 2005-09-15 EP EP05810363A patent/EP1789055A4/en not_active Withdrawn
- 2005-09-15 JP JP2007532441A patent/JP2008513463A/en not_active Withdrawn
Non-Patent Citations (3)
Title |
---|
DIANE H. BOSCHELLI: "4-Anilino-3-quinolinecarbonitriles: an emerging class of kinase inhibitors", CURRENT TOPICS IN MEDICINAL CHEMISTRY, BENTHAM SCIENCE PUBLISHERS, HILVERSUM, NL, vol. 2, no. 9, 1 September 2002 (2002-09-01), pages 1051 - 1063, XP009026991, ISSN: 1568-0266 * |
DIANE H. BOSCHELLI: "Identification of 7-phenylaminothieno[3,2-b]pyridine-6-carbonitriles as a new class of Src kinase inhibitors", JOURNAL OF MEDICINAL CHEMISTRY, vol. 47, no. 27, 12 July 2004 (2004-07-12), pages 6666 - 6668, XP002546910 * |
SIGMOND G. JOHNSON ET AL: "A concise synthesis of 7-chloro-2-methylsulfanyl- thiazolo[4,5-b]pyridine-6-carbonitrile, a versatile intermediate for substituted 6-cyanothiazolopyridines", TETRAHEDRON LETTERS, ELSEVIER, AMSTERDAM, vol. 47, no. 28, 12 July 2006 (2006-07-12), pages 4853 - 4856, XP025004418, ISSN: 0040-4039, [retrieved on 20060712] * |
Also Published As
Publication number | Publication date |
---|---|
JP2008513463A (en) | 2008-05-01 |
CN101056639A (en) | 2007-10-17 |
WO2006031929A2 (en) | 2006-03-23 |
US20060058341A1 (en) | 2006-03-16 |
WO2006031929A3 (en) | 2006-06-01 |
EP1789055A2 (en) | 2007-05-30 |
US7659284B2 (en) | 2010-02-09 |
AU2005284796A1 (en) | 2006-03-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
17P | Request for examination filed |
Effective date: 20070307 |
|
AK | Designated contracting states |
Kind code of ref document: A2 Designated state(s): AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR |
|
DAX | Request for extension of the european patent (deleted) | ||
RIC1 | Information provided on ipc code assigned before grant |
Ipc: A61K 31/445 20060101ALI20090930BHEP Ipc: A61K 31/5377 20060101ALI20090930BHEP Ipc: C07D 513/04 20060101AFI20090930BHEP Ipc: A61K 31/496 20060101ALI20090930BHEP Ipc: A61P 35/00 20060101ALI20090930BHEP Ipc: A61K 31/437 20060101ALI20090930BHEP |
|
A4 | Supplementary search report drawn up and despatched |
Effective date: 20091008 |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
18D | Application deemed to be withdrawn |
Effective date: 20100108 |