EP1663231A4 - Oral itraconazole composition which is not affected by ingested food and process for preparing same - Google Patents

Oral itraconazole composition which is not affected by ingested food and process for preparing same

Info

Publication number: EP1663231A4
Authority: EP; European Patent Office
Prior art keywords: affected; preparing same; ingested food; oral itraconazole; itraconazole composition
Prior art date: 2003-09-09
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Withdrawn

Application number

EP04774524A

Other languages

German (de)

French (fr)

Other versions

EP1663231A1 (en

Inventor

Jong Soo Woo

Hong Gi Yi

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Hanmi Pharmaceutical Co Ltd

Hanmi Pharmaceutical Industries Co Ltd

Original Assignee

Hanmi Pharmaceutical Co Ltd

Hanmi Pharmaceutical Industries Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-09-09

Filing date

2004-09-07

Publication date

2009-04-29

2004-09-07 Application filed by Hanmi Pharmaceutical Co Ltd, Hanmi Pharmaceutical Industries Co Ltd filed Critical Hanmi Pharmaceutical Co Ltd

2004-09-07 Priority claimed from PCT/KR2004/002264 external-priority patent/WO2005023262A1/en

2006-06-07 Publication of EP1663231A1 publication Critical patent/EP1663231A1/en

2009-04-29 Publication of EP1663231A4 publication Critical patent/EP1663231A4/en

Status Withdrawn legal-status Critical Current

Links

VHVPQPYKVGDNFY-DFMJLFEVSA-N 2-[(2r)-butan-2-yl]-4-[4-[4-[4-[[(2r,4s)-2-(2,4-dichlorophenyl)-2-(1,2,4-triazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]piperazin-1-yl]phenyl]-1,2,4-triazol-3-one Chemical compound O=C1N([C@H](C)CC)N=CN1C1=CC=C(N2CCN(CC2)C=2C=CC(OC[C@@H]3O[C@](CN4N=CN=C4)(OC3)C=3C(=CC(Cl)=CC=3)Cl)=CC=2)C=C1 VHVPQPYKVGDNFY-DFMJLFEVSA-N 0.000 title 1
229960004130 itraconazole Drugs 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/485—Inorganic compounds

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Epidemiology (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Inorganic Chemistry (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Dispersion Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Plural Heterocyclic Compounds (AREA)

EP04774524A 2003-09-09 2004-09-07 Oral itraconazole composition which is not affected by ingested food and process for preparing same Withdrawn EP1663231A4 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
KR10-2003-0063147A KR100529766B1 (en)	2003-09-09	2003-09-09	Oral itraconazole composition which is not affected by ingested food and preparation thereof
PCT/KR2004/002264 WO2005023262A1 (en)	2003-09-09	2004-09-07	Oral itraconazole composition which is not affected by ingested food and process for preparing same

Publications (2)

Publication Number	Publication Date
EP1663231A1 EP1663231A1 (en)	2006-06-07
EP1663231A4 true EP1663231A4 (en)	2009-04-29

Family

ID=36096818

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EP04774524A Withdrawn EP1663231A4 (en)	2003-09-09	2004-09-07	Oral itraconazole composition which is not affected by ingested food and process for preparing same

Country Status (10)

Country	Link
EP (1)	EP1663231A4 (en)
JP (1)	JP2007505103A (en)
KR (1)	KR100529766B1 (en)
CN (1)	CN100475211C (en)
AU (1)	AU2004270069B2 (en)
BR (1)	BRPI0414192A (en)
CA (1)	CA2538019C (en)
IL (1)	IL173743A (en)
MX (1)	MXPA06002239A (en)
RU (1)	RU2006111477A (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN104507480A (en)	2012-06-21	2015-04-08	梅恩医药国际有限公司	Itraconazole compositions and dosage forms, and methods of using the same
CN104688536B (en) *	2015-02-03	2016-06-08	常州制药厂有限公司	A kind of preparation method of itraconazole preparation

Citations (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2000000179A1 (en) *	1998-06-27	2000-01-06	Won Jin Biopharma Co., Ltd.	Solid dispersed preparation of poorly water-soluble drug containing oil, fatty acid or mixtures thereof
WO2000059475A1 (en) *	1999-04-06	2000-10-12	Lipocine, Inc.	Compositions and methods for improved delivery of ionizable hydrophobic therapeutic agents
KR20020054573A (en) *	2000-12-28	2002-07-08	민경윤	Composition for oral administration of poorly soluble antifungal agent and process for the preparation thereof
KR20030000799A (en) *	2001-06-27	2003-01-06	한미약품공업 주식회사	Composition for oral administration of poorly soluble antifungal agent and process for the preparation thereof

2003
- 2003-09-09 KR KR10-2003-0063147A patent/KR100529766B1/en not_active IP Right Cessation
2004
- 2004-09-07 CN CNB2004800258516A patent/CN100475211C/en not_active Expired - Fee Related
- 2004-09-07 RU RU2006111477/15A patent/RU2006111477A/en not_active Application Discontinuation
- 2004-09-07 EP EP04774524A patent/EP1663231A4/en not_active Withdrawn
- 2004-09-07 JP JP2006526025A patent/JP2007505103A/en active Pending
- 2004-09-07 MX MXPA06002239A patent/MXPA06002239A/en not_active Application Discontinuation
- 2004-09-07 AU AU2004270069A patent/AU2004270069B2/en not_active Ceased
- 2004-09-07 BR BRPI0414192-0A patent/BRPI0414192A/en not_active IP Right Cessation
- 2004-09-07 CA CA002538019A patent/CA2538019C/en not_active Expired - Fee Related
2006
- 2006-02-15 IL IL173743A patent/IL173743A/en not_active IP Right Cessation

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2000000179A1 (en) *	1998-06-27	2000-01-06	Won Jin Biopharma Co., Ltd.	Solid dispersed preparation of poorly water-soluble drug containing oil, fatty acid or mixtures thereof
WO2000059475A1 (en) *	1999-04-06	2000-10-12	Lipocine, Inc.	Compositions and methods for improved delivery of ionizable hydrophobic therapeutic agents
KR20020054573A (en) *	2000-12-28	2002-07-08	민경윤	Composition for oral administration of poorly soluble antifungal agent and process for the preparation thereof
KR20030000799A (en) *	2001-06-27	2003-01-06	한미약품공업 주식회사	Composition for oral administration of poorly soluble antifungal agent and process for the preparation thereof

Also Published As

Publication number	Publication date
KR100529766B1 (en)	2005-11-17
JP2007505103A (en)	2007-03-08
BRPI0414192A (en)	2006-10-31
CA2538019A1 (en)	2005-03-17
CN100475211C (en)	2009-04-08
RU2006111477A (en)	2006-08-27
KR20050026169A (en)	2005-03-15
CA2538019C (en)	2009-09-01
IL173743A0 (en)	2006-07-05
CN1849123A (en)	2006-10-18
IL173743A (en)	2012-08-30
AU2004270069B2 (en)	2008-03-13
MXPA06002239A (en)	2006-06-20
EP1663231A1 (en)	2006-06-07
AU2004270069A1 (en)	2005-03-17

Legal Events

Date	Code	Title	Description
2006-05-05	PUAI	Public reference made under article 153(3) epc to a published international application that has entered the european phase	Free format text: ORIGINAL CODE: 0009012
2006-06-07	17P	Request for examination filed	Effective date: 20060216
2006-06-07	AK	Designated contracting states	Kind code of ref document: A1 Designated state(s): AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
2006-12-13	DAX	Request for extension of the european patent (deleted)
2009-04-29	A4	Supplementary search report drawn up and despatched	Effective date: 20090331
2009-08-19	17Q	First examination report despatched	Effective date: 20090715
2011-03-11	STAA	Information on the status of an ep patent application or granted ep patent	Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN
2011-04-13	18D	Application deemed to be withdrawn	Effective date: 20101026

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