EE200200362A - Diasepiinkarboksamiidi derivaadid, nende valmistamine ja kasutamine ravimitena ning neid sisaldavadfarmatseutilised kompositsioonid - Google Patents
Diasepiinkarboksamiidi derivaadid, nende valmistamine ja kasutamine ravimitena ning neid sisaldavadfarmatseutilised kompositsioonidInfo
- Publication number
- EE200200362A EE200200362A EEP200200362A EEP200200362A EE200200362A EE 200200362 A EE200200362 A EE 200200362A EE P200200362 A EEP200200362 A EE P200200362A EE P200200362 A EEP200200362 A EE P200200362A EE 200200362 A EE200200362 A EE 200200362A
- Authority
- EE
- Estonia
- Prior art keywords
- pharmaceuticals
- preparation
- pharmaceutical compositions
- compositions containing
- carboxamide derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Communicable Diseases (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Oncology (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9916567A FR2802927B1 (fr) | 1999-12-28 | 1999-12-28 | Nouveaux derives de diazepine carboxamide, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et leur nouvelle utilisation |
PCT/FR2000/003622 WO2001047930A1 (fr) | 1999-12-28 | 2000-12-21 | Derives de diazepine carboxamide, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et leur utilisation |
Publications (1)
Publication Number | Publication Date |
---|---|
EE200200362A true EE200200362A (et) | 2003-08-15 |
Family
ID=9553901
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EEP200200362A EE200200362A (et) | 1999-12-28 | 2000-12-21 | Diasepiinkarboksamiidi derivaadid, nende valmistamine ja kasutamine ravimitena ning neid sisaldavadfarmatseutilised kompositsioonid |
Country Status (26)
Country | Link |
---|---|
EP (1) | EP1246824B1 (et) |
JP (1) | JP2003519152A (et) |
KR (1) | KR20020062772A (et) |
AT (1) | ATE268775T1 (et) |
AU (1) | AU780522B2 (et) |
BR (1) | BR0016845A (et) |
CA (1) | CA2395275A1 (et) |
DE (1) | DE60011473T2 (et) |
DK (1) | DK1246824T3 (et) |
EA (1) | EA005288B1 (et) |
EE (1) | EE200200362A (et) |
ES (1) | ES2218275T3 (et) |
FR (1) | FR2802927B1 (et) |
HR (1) | HRP20020558A2 (et) |
HU (1) | HUP0203921A3 (et) |
IL (1) | IL150419A0 (et) |
MX (1) | MXPA02006413A (et) |
NO (1) | NO20023107L (et) |
NZ (1) | NZ519884A (et) |
PL (1) | PL355950A1 (et) |
PT (1) | PT1246824E (et) |
SI (1) | SI1246824T1 (et) |
SK (1) | SK9092002A3 (et) |
WO (1) | WO2001047930A1 (et) |
YU (1) | YU47502A (et) |
ZA (1) | ZA200205221B (et) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20220115062A (ko) | 2021-02-09 | 2022-08-17 | (주)오스티오뉴로젠 | 크로몬 구조의 화합물을 포함하는 골다공증의 예방 및 치료용 약학적 조성물 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6204261B1 (en) * | 1995-12-20 | 2001-03-20 | Vertex Pharmaceuticals Incorporated | Inhibitors of interleukin-1β Converting enzyme inhibitors |
US5552400A (en) * | 1994-06-08 | 1996-09-03 | Sterling Winthrop Inc. | Fused-bicyclic lactams as interleukin-1β converting enzyme inhibitors |
US5847135A (en) * | 1994-06-17 | 1998-12-08 | Vertex Pharmaceuticals, Incorporated | Inhibitors of interleukin-1β converting enzyme |
-
1999
- 1999-12-28 FR FR9916567A patent/FR2802927B1/fr not_active Expired - Fee Related
-
2000
- 2000-12-21 ES ES00990087T patent/ES2218275T3/es not_active Expired - Lifetime
- 2000-12-21 EE EEP200200362A patent/EE200200362A/et unknown
- 2000-12-21 JP JP2001549400A patent/JP2003519152A/ja not_active Abandoned
- 2000-12-21 EP EP00990087A patent/EP1246824B1/fr not_active Expired - Lifetime
- 2000-12-21 DE DE60011473T patent/DE60011473T2/de not_active Expired - Fee Related
- 2000-12-21 HU HU0203921A patent/HUP0203921A3/hu unknown
- 2000-12-21 KR KR1020027008366A patent/KR20020062772A/ko not_active Application Discontinuation
- 2000-12-21 CA CA002395275A patent/CA2395275A1/fr not_active Abandoned
- 2000-12-21 PT PT00990087T patent/PT1246824E/pt unknown
- 2000-12-21 AU AU26888/01A patent/AU780522B2/en not_active Ceased
- 2000-12-21 WO PCT/FR2000/003622 patent/WO2001047930A1/fr not_active Application Discontinuation
- 2000-12-21 EA EA200200721A patent/EA005288B1/ru not_active IP Right Cessation
- 2000-12-21 SK SK909-2002A patent/SK9092002A3/sk unknown
- 2000-12-21 YU YU47502A patent/YU47502A/sh unknown
- 2000-12-21 BR BR0016845-9A patent/BR0016845A/pt not_active IP Right Cessation
- 2000-12-21 MX MXPA02006413A patent/MXPA02006413A/es active IP Right Grant
- 2000-12-21 SI SI200030455T patent/SI1246824T1/xx unknown
- 2000-12-21 IL IL15041900A patent/IL150419A0/xx unknown
- 2000-12-21 AT AT00990087T patent/ATE268775T1/de not_active IP Right Cessation
- 2000-12-21 DK DK00990087T patent/DK1246824T3/da active
- 2000-12-21 PL PL00355950A patent/PL355950A1/xx not_active Application Discontinuation
- 2000-12-21 NZ NZ519884A patent/NZ519884A/en unknown
-
2002
- 2002-06-27 HR HR20020558A patent/HRP20020558A2/hr not_active Application Discontinuation
- 2002-06-27 NO NO20023107A patent/NO20023107L/no not_active Application Discontinuation
- 2002-06-28 ZA ZA200205221A patent/ZA200205221B/en unknown
Also Published As
Publication number | Publication date |
---|---|
HUP0203921A3 (en) | 2005-01-28 |
HUP0203921A2 (hu) | 2003-03-28 |
EA005288B1 (ru) | 2004-12-30 |
IL150419A0 (en) | 2002-12-01 |
EP1246824B1 (fr) | 2004-06-09 |
BR0016845A (pt) | 2002-10-15 |
PT1246824E (pt) | 2004-10-29 |
PL355950A1 (en) | 2004-05-31 |
MXPA02006413A (es) | 2002-11-29 |
DE60011473T2 (de) | 2005-06-30 |
NO20023107D0 (no) | 2002-06-27 |
AU2688801A (en) | 2001-07-09 |
SK9092002A3 (en) | 2003-04-01 |
NO20023107L (no) | 2002-08-27 |
HRP20020558A2 (en) | 2004-02-29 |
CA2395275A1 (fr) | 2001-07-05 |
KR20020062772A (ko) | 2002-07-29 |
ZA200205221B (en) | 2003-09-04 |
NZ519884A (en) | 2005-03-24 |
EA200200721A1 (ru) | 2002-12-26 |
SI1246824T1 (en) | 2004-10-31 |
DK1246824T3 (da) | 2004-10-18 |
AU780522B2 (en) | 2005-03-24 |
YU47502A (sh) | 2005-03-15 |
EP1246824A1 (fr) | 2002-10-09 |
ATE268775T1 (de) | 2004-06-15 |
FR2802927A1 (fr) | 2001-06-29 |
JP2003519152A (ja) | 2003-06-17 |
WO2001047930A1 (fr) | 2001-07-05 |
FR2802927B1 (fr) | 2002-03-01 |
DE60011473D1 (de) | 2004-07-15 |
ES2218275T3 (es) | 2004-11-16 |
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