ECSP993019A - PYROLEUM COMPOUNDS [2,3-d] PIRIMIDINE - Google Patents
PYROLEUM COMPOUNDS [2,3-d] PIRIMIDINEInfo
- Publication number
- ECSP993019A ECSP993019A ECSP993019A ECSP993019A EC SP993019 A ECSP993019 A EC SP993019A EC SP993019 A ECSP993019 A EC SP993019A EC SP993019 A ECSP993019 A EC SP993019A
- Authority
- EC
- Ecuador
- Prior art keywords
- diabetes
- pyroleum
- pirimidine
- compounds
- crohn
- Prior art date
Links
Abstract
La presente invención proporciona un compuesto de fórmula: (gráfico), en la que R1, R2 y R3 son como se han definido antes, que son inhibidores de las enzimas proteína tirosina quinasas, como Janus Quinasa 3 y, como tales, son una terapia útil como agentes inmunosupresores para el transplante de órganos, lupus, esclerosis múltiple, artritis reumatoide, psoriasis, diabetes Tipo I y complicaciones de la diabetes, cáncer, asma, dermatitis atópica, trastornos autoinmunes del tiroides, colitis ulcerosa, enfermedad de Crohn, enfermedad de Alzheimer, leucemia y otras enfermedades autoinmunes.The present invention provides a compound of the formula: (graph), wherein R1, R2 and R3 are as defined above, that they are inhibitors of protein tyrosine kinase enzymes, such as Janus kinase 3 and, as such, are a therapy Useful as immunosuppressive agents for organ transplantation, lupus, multiple sclerosis, rheumatoid arthritis, psoriasis, Type I diabetes and complications of diabetes, cancer, asthma, atopic dermatitis, autoimmune thyroid disorders, ulcerative colitis, Crohn's disease, Alzheimer, leukemia and other autoimmune diseases.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP993019 ECSP993019A (en) | 1999-06-16 | 1999-06-16 | PYROLEUM COMPOUNDS [2,3-d] PIRIMIDINE |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP993019 ECSP993019A (en) | 1999-06-16 | 1999-06-16 | PYROLEUM COMPOUNDS [2,3-d] PIRIMIDINE |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP993019A true ECSP993019A (en) | 1999-08-12 |
Family
ID=42044008
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSP993019 ECSP993019A (en) | 1999-06-16 | 1999-06-16 | PYROLEUM COMPOUNDS [2,3-d] PIRIMIDINE |
Country Status (1)
Country | Link |
---|---|
EC (1) | ECSP993019A (en) |
-
1999
- 1999-06-16 EC ECSP993019 patent/ECSP993019A/en unknown
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