ECSP12012357A - Análogos del glucagón - Google Patents

Análogos del glucagón

Info

Publication number
ECSP12012357A
ECSP12012357A ECSP12012357A ECSP12012357A EC SP12012357 A ECSP12012357 A EC SP12012357A EC SP12012357 A ECSP12012357 A EC SP12012357A EC SP12012357 A ECSP12012357 A EC SP12012357A
Authority
EC
Ecuador
Prior art keywords
glucagon
glucagon analogs
compounds
glp
diabetes
Prior art date
Application number
Other languages
English (en)
Inventor
Ditte Riber
Eddi Meier
Original Assignee
Zealand Pharma As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44630046&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP12012357(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Zealand Pharma As filed Critical Zealand Pharma As
Publication of ECSP12012357A publication Critical patent/ECSP12012357A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/605Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/26Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Epidemiology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención proporciona materiales y procedimientos para promover la pérdida de peso o evitar el aumento de peso y para el tratamiento de la diabetes y de los trastornos metabólicos asociados. En particular, la invención proporciona novedosos compuestos peptídicos análogos al glucagón efectivos en tales procedimientos. El efecto de los compuestos puede estar mediado, por ejemplo, aumentando la selectividad por el receptor de GLP-1 en comparación con el glucagón humano.
ECSP12012357 2010-06-24 2012-12-26 Análogos del glucagón ECSP12012357A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA201000558 2010-06-24
US35861410P 2010-06-25 2010-06-25

Publications (1)

Publication Number Publication Date
ECSP12012357A true ECSP12012357A (es) 2013-01-31

Family

ID=44630046

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP12012357 ECSP12012357A (es) 2010-06-24 2012-12-26 Análogos del glucagón

Country Status (20)

Country Link
US (2) US9169310B2 (es)
EP (1) EP2585482B1 (es)
JP (1) JP6023048B2 (es)
KR (1) KR20130086343A (es)
CN (1) CN103068841A (es)
AP (1) AP2013006671A0 (es)
AU (1) AU2011269430A1 (es)
BR (1) BR112012033225A2 (es)
CA (1) CA2802897A1 (es)
CL (1) CL2012003641A1 (es)
CO (1) CO6660483A2 (es)
EA (1) EA201291234A1 (es)
EC (1) ECSP12012357A (es)
MA (1) MA34383B1 (es)
MX (1) MX2012014961A (es)
NZ (1) NZ604208A (es)
PE (1) PE20130338A1 (es)
SG (1) SG186764A1 (es)
TN (1) TN2012000560A1 (es)
WO (1) WO2011160633A1 (es)

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Also Published As

Publication number Publication date
WO2011160633A1 (en) 2011-12-29
CA2802897A1 (en) 2011-12-29
JP2013530969A (ja) 2013-08-01
AP2013006671A0 (en) 2013-01-31
US20150376257A1 (en) 2015-12-31
CL2012003641A1 (es) 2013-09-06
KR20130086343A (ko) 2013-08-01
SG186764A1 (en) 2013-02-28
CN103068841A (zh) 2013-04-24
MX2012014961A (es) 2013-02-26
MA34383B1 (fr) 2013-07-03
EP2585482A1 (en) 2013-05-01
BR112012033225A2 (pt) 2017-06-20
US20130157929A1 (en) 2013-06-20
PE20130338A1 (es) 2013-03-16
JP6023048B2 (ja) 2016-11-09
NZ604208A (en) 2014-10-31
CO6660483A2 (es) 2013-04-30
TN2012000560A1 (en) 2014-04-01
EP2585482B1 (en) 2019-03-27
EA201291234A1 (ru) 2013-07-30
US9169310B2 (en) 2015-10-27
AU2011269430A1 (en) 2013-01-10

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