EA200802417A1 - SUBSTITUTED PHENYLACETIC ACIDS AS DP-2 ANTAGONISTS - Google Patents

SUBSTITUTED PHENYLACETIC ACIDS AS DP-2 ANTAGONISTS

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Publication number
EA200802417A1
EA200802417A1 EA200802417A EA200802417A EA200802417A1 EA 200802417 A1 EA200802417 A1 EA 200802417A1 EA 200802417 A EA200802417 A EA 200802417A EA 200802417 A EA200802417 A EA 200802417A EA 200802417 A1 EA200802417 A1 EA 200802417A1
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EA
Eurasian Patent Office
Prior art keywords
antagonists
substituted phenylacetic
phenylacetic acids
methods
conditions
Prior art date
Application number
EA200802417A
Other languages
Russian (ru)
Inventor
Томас Дадлер
Франсьен Фаруз
Керри Фаулер
Натали Хоторн
Данвен Хуанг
Цзинь Бохан
Мусон Ким
Эндрю Лавер
Джошуа Одинго
Эми Оливер
Марк Рид
Фуцян Руан
Юджин Торсет
Original Assignee
Икос Корпорейшн
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Publication date
Application filed by Икос Корпорейшн filed Critical Икос Корпорейшн
Publication of EA200802417A1 publication Critical patent/EA200802417A1/en

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Abstract

Предложены замещенные производные фенилуксусной кислоты формулы (I), фармацевтические композиции, способы их получения и способы, которые являются полезными в лечении и предупреждении нарушений или состояний, чувствительных к модуляции DP-2-рецептора, в частности воспалительных и связанных с иммунитетом нарушений и состояний, таких как астма, аллергический ринит и атопический дерматит.Proposed substituted phenylacetic acid derivatives of formula (I), pharmaceutical compositions, methods for their preparation and methods that are useful in the treatment and prevention of disorders or conditions sensitive to modulation of the DP-2 receptor, in particular inflammatory and immune-related disorders and conditions, such as asthma, allergic rhinitis and atopic dermatitis.

EA200802417A 2006-06-09 2007-06-08 SUBSTITUTED PHENYLACETIC ACIDS AS DP-2 ANTAGONISTS EA200802417A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81239906P 2006-06-09 2006-06-09
PCT/US2007/070805 WO2007146838A2 (en) 2006-06-09 2007-06-08 Substituted phenyl acetic acids as dp-2 antagonists

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EA200802417A1 true EA200802417A1 (en) 2009-06-30

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EA201200423A EA201200423A1 (en) 2006-06-09 2007-06-08 SUBSTITUTED PHENYLACETIC ACIDS AS DP-2 ANTAGONISTS

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EP (1) EP2044017A2 (en)
JP (1) JP2009539881A (en)
CN (1) CN101490001A (en)
AU (1) AU2007257841A1 (en)
BR (1) BRPI0712332A2 (en)
CA (1) CA2654927A1 (en)
EA (2) EA200802417A1 (en)
MX (1) MX2008015638A (en)
NO (1) NO20090139L (en)
WO (1) WO2007146838A2 (en)

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