EA200601842A1 - D-гомо-17-хлор-16(17)-ен-стероиды - Google Patents

D-гомо-17-хлор-16(17)-ен-стероиды

Info

Publication number
EA200601842A1
EA200601842A1 EA200601842A EA200601842A EA200601842A1 EA 200601842 A1 EA200601842 A1 EA 200601842A1 EA 200601842 A EA200601842 A EA 200601842A EA 200601842 A EA200601842 A EA 200601842A EA 200601842 A1 EA200601842 A1 EA 200601842A1
Authority
EA
Eurasian Patent Office
Prior art keywords
хоч
стероиды
гоо
eno
steroids
Prior art date
Application number
EA200601842A
Other languages
English (en)
Inventor
Свен Ринг
Ральф Вырва
Гюнтер Кауфманн
Original Assignee
Шеринг Акциенгезельшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Шеринг Акциенгезельшафт filed Critical Шеринг Акциенгезельшафт
Publication of EA200601842A1 publication Critical patent/EA200601842A1/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Изобретение относится к D-гомо-17-хлор-16(17)-ен-стероидам формулы I с андрогенным действиемспособу их получения, фармацевтическим композициям, которые содержат эти соединения, а также их применению для получения лекарственных средств.
EA200601842A 2004-04-08 2005-04-07 D-гомо-17-хлор-16(17)-ен-стероиды EA200601842A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004018441A DE102004018441B4 (de) 2004-04-08 2004-04-08 D-Homo-17-chlor-16(17)en Steroide
PCT/EP2005/003792 WO2005097819A1 (de) 2004-04-08 2005-04-07 D-homo-17-chlor-16(17)en steroide

Publications (1)

Publication Number Publication Date
EA200601842A1 true EA200601842A1 (ru) 2007-04-27

Family

ID=34966688

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200601842A EA200601842A1 (ru) 2004-04-08 2005-04-07 D-гомо-17-хлор-16(17)-ен-стероиды

Country Status (18)

Country Link
EP (1) EP1735331A1 (ru)
KR (1) KR20070007910A (ru)
CN (1) CN1997659A (ru)
AR (1) AR048536A1 (ru)
AU (1) AU2005231970A1 (ru)
CA (1) CA2563541A1 (ru)
CR (1) CR8736A (ru)
DE (1) DE102004018441B4 (ru)
EA (1) EA200601842A1 (ru)
EC (1) ECSP066973A (ru)
GT (1) GT200500084A (ru)
MX (1) MXPA06012849A (ru)
NO (1) NO20065126L (ru)
PA (1) PA8629401A1 (ru)
SV (1) SV2005002076A (ru)
TW (1) TW200603812A (ru)
WO (1) WO2005097819A1 (ru)
ZA (1) ZA200609275B (ru)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4788218A (en) * 1984-05-21 1988-11-29 Sri International 17 a β-hydroxy-7 α-methyl-d-homo-19-norandrost-4,16-diene-3-one and the 17-esters thereof: methods of preparation and uses
DE4042005A1 (de) * 1990-12-22 1992-06-25 Schering Ag D-homo-(16-en)-11(beta)-aryl-4-estrene
DE69301149T3 (de) * 1993-08-21 2000-01-05 Nestle Sa Herstellung eines Gewürzes
DE10151365A1 (de) * 2001-10-17 2003-04-30 Schering Ag 17-Chlor-D-Homosteroide als selektive Estrogenrezeptorantagonisten

Also Published As

Publication number Publication date
DE102004018441A1 (de) 2005-11-03
SV2005002076A (es) 2005-12-06
EP1735331A1 (de) 2006-12-27
NO20065126L (no) 2007-01-04
AU2005231970A1 (en) 2005-10-20
PA8629401A1 (es) 2006-07-03
CR8736A (es) 2007-08-28
ZA200609275B (en) 2009-08-26
DE102004018441B4 (de) 2007-12-20
AR048536A1 (es) 2006-05-03
WO2005097819A1 (de) 2005-10-20
ECSP066973A (es) 2006-12-29
CA2563541A1 (en) 2005-10-20
TW200603812A (en) 2006-02-01
CN1997659A (zh) 2007-07-11
MXPA06012849A (es) 2007-01-26
GT200500084A (es) 2006-03-24
KR20070007910A (ko) 2007-01-16

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