EA199900821A1 - Способ получения производных пиразола - Google Patents

Способ получения производных пиразола

Info

Publication number
EA199900821A1
EA199900821A1 EA199900821A EA199900821A EA199900821A1 EA 199900821 A1 EA199900821 A1 EA 199900821A1 EA 199900821 A EA199900821 A EA 199900821A EA 199900821 A EA199900821 A EA 199900821A EA 199900821 A1 EA199900821 A1 EA 199900821A1
Authority
EA
Eurasian Patent Office
Prior art keywords
formula
pyrazole derivatives
producing pyrazole
compound
producing
Prior art date
Application number
EA199900821A
Other languages
English (en)
Other versions
EA002086B1 (ru
Inventor
Питер Вайэтт Ньюсам
Original Assignee
Рон-Пуленк Агро
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Рон-Пуленк Агро filed Critical Рон-Пуленк Агро
Publication of EA199900821A1 publication Critical patent/EA199900821A1/ru
Publication of EA002086B1 publication Critical patent/EA002086B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/63—Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C255/65—Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton with the nitrogen atoms further bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C317/30—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of rings other than six-membered aromatic rings of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C07C317/48—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Изобретение относится к способу получения соединений, имеющих формулу (IV), где R, R, Rи Ar имеют значения, определенные в описании, с помощью реакции соединения формулы (I) с соединением формулы (II) согласно схеме реакций. Соединения формулы (IV) полезны в качестве пестицидов.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA199900821A 1997-03-12 1998-03-05 Способ получения 3,4,5-тризамещённых 1-арилпиразолов EA002086B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/815,848 US5907041A (en) 1997-03-12 1997-03-12 Process for preparing pyrazole derivatives
PCT/EP1998/001226 WO1998040358A1 (en) 1997-03-12 1998-03-05 Process for preparing pyrazole derivatives

Publications (2)

Publication Number Publication Date
EA199900821A1 true EA199900821A1 (ru) 2000-04-24
EA002086B1 EA002086B1 (ru) 2001-12-24

Family

ID=25219006

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199900821A EA002086B1 (ru) 1997-03-12 1998-03-05 Способ получения 3,4,5-тризамещённых 1-арилпиразолов

Country Status (25)

Country Link
US (2) US5907041A (ru)
EP (1) EP0966444B1 (ru)
JP (1) JP4429389B2 (ru)
KR (1) KR100536795B1 (ru)
CN (2) CN1107672C (ru)
AR (1) AR015108A1 (ru)
AT (1) ATE223382T1 (ru)
AU (1) AU750836B2 (ru)
BG (1) BG64648B1 (ru)
BR (1) BR9808854B1 (ru)
CA (1) CA2283507C (ru)
CZ (1) CZ296302B6 (ru)
DE (1) DE69807660T2 (ru)
DK (1) DK0966444T3 (ru)
EA (1) EA002086B1 (ru)
ES (1) ES2179476T3 (ru)
HU (1) HU229879B1 (ru)
ID (1) ID23447A (ru)
IL (1) IL131856A0 (ru)
NZ (1) NZ337766A (ru)
PL (1) PL196442B1 (ru)
SK (1) SK284800B6 (ru)
TR (1) TR199902213T2 (ru)
WO (1) WO1998040358A1 (ru)
ZA (1) ZA981875B (ru)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2772381C1 (ru) * 2021-07-01 2022-05-19 Федеральное государственное бюджетное учреждение науки Институт органического синтеза им. И.Я. Постовского Уральского отделения Российской академии наук 4-(4-Метоксифенилдиазенил)-3,5-диметил-1-(4-нитрофенил)-1H-пиразол с антимикотической активностью в отношении штаммов патогенных грибов - дерматофитов

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GB9907458D0 (en) * 1999-03-31 1999-05-26 Rhone Poulenc Agrochimie Processes for preparing pesticidal intermediates
EP1264823A1 (en) * 2001-06-08 2002-12-11 Novartis AG Process for the preparation of 2,3-dicyanopropionates
WO2005023773A1 (en) * 2003-09-04 2005-03-17 Pfizer Limited Process for the preparation of substituted aryl pyrazoles
KR101389246B1 (ko) 2004-07-15 2014-04-24 브리스톨-마이어스스퀴브컴파니 아릴- 및 헤테로아릴-치환된 테트라히드로이소퀴놀린, 및 이것의 노르에피네프린, 도파민 및 세로토닌의 재흡수를 차단하기 위한 용도
KR101594898B1 (ko) 2005-07-15 2016-02-18 알바니 몰레큘라 리써치, 인크. 아릴- 및 헤테로아릴-치환된 테트라히드로벤자제핀, 및 노르에피네프린, 도파민 및 세로토닌의 재흡수를 차단하기 위한 용도
US9156812B2 (en) 2008-06-04 2015-10-13 Bristol-Myers Squibb Company Crystalline form of 6-[(4S)-2-methyl-4-(2-naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine
JP5739415B2 (ja) 2009-05-12 2015-06-24 ブリストル−マイヤーズ スクウィブ カンパニー （Ｓ）−７−（［１，２，４］トリアゾロ［１，５−ａ］ピリジン−６−イル）−４−（３，４−ジクロロフェニル）−１，２，３，４−テトラヒドロイソキノリンの結晶形態およびその使用
WO2010132437A1 (en) 2009-05-12 2010-11-18 Albany Molecular Research, Inc. Aryl, heteroaryl, and heterocycle substituted tetrahydroisoquinolines and use thereof
CN103270119B (zh) * 2010-12-30 2016-04-20 巴斯夫欧洲公司 表面改性的颜料制剂
CN111825653A (zh) 2019-04-19 2020-10-27 安道麦马克西姆有限公司 取代吡唑类化合物的制备及其作为邻氨基苯甲酰胺前体的用途
CN110483480A (zh) * 2019-09-11 2019-11-22 江苏优普生物化学科技股份有限公司 2-(3-氯吡啶-2-基)-5-羟基-3-吡唑烷甲酸乙酯的合成方法
CN110981806A (zh) * 2019-12-06 2020-04-10 江苏优普生物化学科技股份有限公司 合成芳基吡唑腈副产碳酸二酯的方法
CN111592510A (zh) * 2020-04-26 2020-08-28 衡水均凯化工有限公司 一种4,4-(六氟亚异丙烯基)二邻二甲酸酐的合成方法
CN111592511A (zh) * 2020-04-26 2020-08-28 衡水均凯化工有限公司 一种4,4-(六氟亚异丙烯基)二邻二甲酸酐的制备工艺

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2772381C1 (ru) * 2021-07-01 2022-05-19 Федеральное государственное бюджетное учреждение науки Институт органического синтеза им. И.Я. Постовского Уральского отделения Российской академии наук 4-(4-Метоксифенилдиазенил)-3,5-диметил-1-(4-нитрофенил)-1H-пиразол с антимикотической активностью в отношении штаммов патогенных грибов - дерматофитов

Also Published As

Publication number Publication date
KR20000076109A (ko) 2000-12-26
CA2283507C (en) 2008-10-28
AU6827098A (en) 1998-09-29
HU229879B1 (en) 2014-11-28
PL335610A1 (en) 2000-05-08
NZ337766A (en) 2001-03-30
DE69807660D1 (de) 2002-10-10
CN1184206C (zh) 2005-01-12
JP4429389B2 (ja) 2010-03-10
TR199902213T2 (xx) 1999-12-21
EA002086B1 (ru) 2001-12-24
ZA981875B (en) 1998-09-09
HUP0002931A2 (hu) 2000-12-28
CN1250440A (zh) 2000-04-12
CZ319799A3 (cs) 2000-01-12
ATE223382T1 (de) 2002-09-15
AR015108A1 (es) 2001-04-18
DK0966444T3 (da) 2002-10-07
CA2283507A1 (en) 1998-09-17
SK123199A3 (en) 2000-05-16
KR100536795B1 (ko) 2005-12-14
US5907041A (en) 1999-05-25
CZ296302B6 (cs) 2006-02-15
BG64648B1 (bg) 2005-10-31
DE69807660T2 (de) 2003-05-08
EP0966444A1 (en) 1999-12-29
BR9808854A (pt) 2000-07-25
SK284800B6 (sk) 2005-11-03
BG103778A (en) 2001-05-31
ID23447A (id) 2000-04-20
JP2001514642A (ja) 2001-09-11
HUP0002931A3 (en) 2001-02-28
PL196442B1 (pl) 2008-01-31
CN1107672C (zh) 2003-05-07
US6090927A (en) 2000-07-18
CN1432569A (zh) 2003-07-30
EP0966444B1 (en) 2002-09-04
ES2179476T3 (es) 2003-01-16
BR9808854B1 (pt) 2011-06-28
AU750836B2 (en) 2002-08-01
IL131856A0 (en) 2001-03-19
WO1998040358A1 (en) 1998-09-17

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Legal Events

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ KG TJ TM

MK4A Patent expired

Designated state(s): BY KZ MD RU