DOP2022000171A - Compuestos tetracíclicos para el tratamiento de infecciones por vih - Google Patents

Compuestos tetracíclicos para el tratamiento de infecciones por vih

Info

Publication number
DOP2022000171A
DOP2022000171A DO2022000171A DO2022000171A DOP2022000171A DO P2022000171 A DOP2022000171 A DO P2022000171A DO 2022000171 A DO2022000171 A DO 2022000171A DO 2022000171 A DO2022000171 A DO 2022000171A DO P2022000171 A DOP2022000171 A DO P2022000171A
Authority
DO
Dominican Republic
Prior art keywords
compounds
treatment
hiv infections
tetracyclic compounds
pharmaceutical compositions
Prior art date
Application number
DO2022000171A
Other languages
English (en)
Inventor
L Mitchell Michael
Jiang Lan
w lin David
Roberts Ezra
M Schwarzwalder Gregg
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of DOP2022000171A publication Critical patent/DOP2022000171A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/22—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed systems contains four or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • AIDS & HIV (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente divulgación se refiere en general a ciertos compuestos tetracíclicos, composiciones farmacéuticas que comprenden dichos compuestos y métodos para preparar dichos compuestos y composiciones farmacéuticas. Los compuestos de la divulgación son útiles para tratar o prevenir la infección por el virus de la inmunodeficiencia humana (VIH).
DO2022000171A 2020-02-24 2022-08-23 Compuestos tetracíclicos para el tratamiento de infecciones por vih DOP2022000171A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US202062980857P 2020-02-24 2020-02-24
US202063036268P 2020-06-08 2020-06-08
US202063128670P 2020-12-21 2020-12-21
PCT/US2021/019179 WO2021173522A1 (en) 2020-02-24 2021-02-23 Tetracyclic compounds for treating hiv infection

Publications (1)

Publication Number Publication Date
DOP2022000171A true DOP2022000171A (es) 2022-10-16

Family

ID=74885056

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2022000171A DOP2022000171A (es) 2020-02-24 2022-08-23 Compuestos tetracíclicos para el tratamiento de infecciones por vih

Country Status (15)

Country Link
US (2) US11697652B2 (es)
EP (1) EP4110783A1 (es)
JP (2) JP7453399B2 (es)
CN (1) CN115151545A (es)
AU (2) AU2021225809B2 (es)
BR (1) BR112022015771A2 (es)
CA (1) CA3166480A1 (es)
CO (1) CO2022011947A2 (es)
CR (1) CR20220418A (es)
DO (1) DOP2022000171A (es)
IL (1) IL295677A (es)
MX (1) MX2022009871A (es)
PE (1) PE20221569A1 (es)
TW (2) TWI777425B (es)
WO (1) WO2021173522A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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Also Published As

Publication number Publication date
EP4110783A1 (en) 2023-01-04
TW202140481A (zh) 2021-11-01
WO2021173522A1 (en) 2021-09-02
CR20220418A (es) 2022-10-10
PE20221569A1 (es) 2022-10-06
JP7453399B2 (ja) 2024-03-19
US20240010650A1 (en) 2024-01-11
CO2022011947A2 (es) 2022-08-30
AU2023266279A1 (en) 2023-12-07
CN115151545A (zh) 2022-10-04
BR112022015771A2 (pt) 2022-10-11
AU2021225809B2 (en) 2023-08-24
AU2021225809A1 (en) 2022-10-13
TWI777425B (zh) 2022-09-11
MX2022009871A (es) 2022-08-19
TW202248199A (zh) 2022-12-16
US11697652B2 (en) 2023-07-11
CA3166480A1 (en) 2021-09-02
IL295677A (en) 2022-10-01
JP2023514635A (ja) 2023-04-06
US20210284642A1 (en) 2021-09-16
JP2023184696A (ja) 2023-12-28

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