DOP2006000015A - PIRAZOLO PIRIDINAS REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING PROCEDURE - Google Patents

PIRAZOLO PIRIDINAS REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING PROCEDURE

Info

Publication number
DOP2006000015A
DOP2006000015A DO2006000015A DO2006000015A DOP2006000015A DO P2006000015 A DOP2006000015 A DO P2006000015A DO 2006000015 A DO2006000015 A DO 2006000015A DO 2006000015 A DO2006000015 A DO 2006000015A DO P2006000015 A DOP2006000015 A DO P2006000015A
Authority
DO
Dominican Republic
Prior art keywords
compositions
piridinas
pirazolo
replaced
contain
Prior art date
Application number
DO2006000015A
Other languages
Spanish (es)
Inventor
Michel Tabart
Baptiste Ronan
Fabrice Viviani
Catherine Souaille
Franck Halley
Eric Bacque
Antonio Ugolini
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of DOP2006000015A publication Critical patent/DOP2006000015A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación y utilización. La presente invención se refiere especialmente a la preparación de pirazolo piridinas sustituidas, composiciones que las contienen, su procedimiento de preparación, y su utilización como medicamento, en particular como agentes anticancerígenos.Pyrazolo substituted pyridines, compositions containing them, manufacturing and use process. The present invention relates especially to the preparation of pyrazolo substituted pyridines, compositions containing them, their preparation process, and their use as a medicament, in particular as anticancer agents.

DO2006000015A 2005-01-19 2006-01-17 PIRAZOLO PIRIDINAS REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING PROCEDURE DOP2006000015A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0500555A FR2880891B1 (en) 2005-01-19 2005-01-19 SUBSTITUTED PYRAZOLO PYRIDINES, COMPOSITIONS CONTAINING SAME, METHOD OF MANUFACTURE AND USE

Publications (1)

Publication Number Publication Date
DOP2006000015A true DOP2006000015A (en) 2006-07-31

Family

ID=35124733

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2006000015A DOP2006000015A (en) 2005-01-19 2006-01-17 PIRAZOLO PIRIDINAS REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING PROCEDURE

Country Status (5)

Country Link
CN (1) CN101146534A (en)
DO (1) DOP2006000015A (en)
ES (1) ES2351160T3 (en)
FR (1) FR2880891B1 (en)
SV (1) SV2006002384A (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2464647B1 (en) 2009-08-11 2016-09-21 Bristol-Myers Squibb Company Azaindazoles as btk kinase modulators and use thereof
EP2593453B1 (en) * 2010-07-15 2014-09-17 Bristol-Myers Squibb Company Azaindazole compounds
GB201015949D0 (en) * 2010-09-22 2010-11-03 Medical Res Council Technology Compounds
JP2013542259A (en) * 2010-11-12 2013-11-21 ブリストル−マイヤーズ スクイブ カンパニー Substituted azaindazole compounds
CN103214479A (en) * 2012-01-18 2013-07-24 武汉东宇生物医药科技有限公司 Pyrazole naphthylurea tyrosine kinase inhibitor and its application
JPWO2013125543A1 (en) * 2012-02-20 2015-07-30 武田薬品工業株式会社 Heterocyclic compounds
CN103524421B (en) * 2013-09-29 2015-04-01 镇江蓝德特药业科技有限公司 Novel naphthoyl urea derivate and medical application thereof
CN104098564A (en) * 2014-07-30 2014-10-15 天津市斯芬克司药物研发有限公司 Pyrazol pyridine compound and preparation method thereof
CN108117551B (en) * 2016-11-29 2020-03-27 华东理工大学 Substituted (1H-pyrazolo [3,4-b ] pyridine) urea compound and anti-tumor application thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA03001169A (en) * 2000-08-10 2003-06-30 Pharmacia Italia Spa Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them.
JP2006514918A (en) * 2002-07-23 2006-05-18 スミスクライン ビーチャム コーポレーション Pyrazolopyrimidines as kinase inhibitors
CA2495216A1 (en) * 2002-08-12 2004-02-19 Sugen, Inc. 3-pyrrolyl-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors
AU2004215644B2 (en) * 2003-02-27 2010-09-02 Palau Pharma, S.A. Pyrazolopyridine derivates
WO2005000813A1 (en) * 2003-05-30 2005-01-06 Imclone Systems Incorporated Heteroarylamino-phenylketone derivatives and their use as kinase inhibitors

Also Published As

Publication number Publication date
FR2880891B1 (en) 2007-02-23
FR2880891A1 (en) 2006-07-21
CN101146534A (en) 2008-03-19
ES2351160T3 (en) 2011-02-01
SV2006002384A (en) 2006-08-25

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