DOP2003000786A - BICYCLE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELLULAR GROWTH. - Google Patents

BICYCLE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELLULAR GROWTH.

Info

Publication number
DOP2003000786A
DOP2003000786A DO2003000786A DO2003000786A DOP2003000786A DO P2003000786 A DOP2003000786 A DO P2003000786A DO 2003000786 A DO2003000786 A DO 2003000786A DO 2003000786 A DO2003000786 A DO 2003000786A DO P2003000786 A DOP2003000786 A DO P2003000786A
Authority
DO
Dominican Republic
Prior art keywords
compounds
formula
treatment
cellular growth
abnormal cellular
Prior art date
Application number
DO2003000786A
Other languages
Spanish (es)
Inventor
Zheng Liu
John Charles Kath
Maria Steflik Brown
Steven Mark Winter
Susan Jane Truesdell
Ruby Anthea Szewc
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Priority to DO2003000786A priority Critical patent/DOP2003000786A/en
Publication of DOP2003000786A publication Critical patent/DOP2003000786A/en

Links

Abstract

La invención se refiere a compuestos de formula 1 Y a sales, Pro fármacos y solvatos farmaceuticamente aceptables de los mismos, en la que R1, R2, R3 y R4 son como se definen en la presente memoria, y en la que el compuesto de formula 1 comprende opcionalmente además un sustituyente hidroxi o un acido O-glucuronico. La invención se refiere también a procedimientos de tratamiento del crecimiento celular anormal en mamíferos mediante la administración de los compuestos de formula 1 y a composiciones farmacéuticas para tratar dichos trastornos que contienen los compuestos de formula 1. la invención se refiere también a procedimientos de preparación de los compuestos de formula 1.The invention relates to compounds of formula 1 and pharmaceutically acceptable salts, Pro drugs and solvates thereof, wherein R1, R2, R3 and R4 are as defined herein, and in which the compound of formula 1 optionally further comprises a hydroxy substituent or an O-glucuronic acid. The invention also relates to methods of treating abnormal cell growth in mammals by administering the compounds of formula 1 and pharmaceutical compositions for treating such disorders containing the compounds of formula 1. The invention also relates to methods of preparing the compounds. compounds of formula 1.

DO2003000786A 2003-12-10 2003-12-10 BICYCLE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELLULAR GROWTH. DOP2003000786A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DO2003000786A DOP2003000786A (en) 2003-12-10 2003-12-10 BICYCLE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELLULAR GROWTH.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DO2003000786A DOP2003000786A (en) 2003-12-10 2003-12-10 BICYCLE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELLULAR GROWTH.

Publications (1)

Publication Number Publication Date
DOP2003000786A true DOP2003000786A (en) 2004-06-30

Family

ID=44261271

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2003000786A DOP2003000786A (en) 2003-12-10 2003-12-10 BICYCLE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELLULAR GROWTH.

Country Status (1)

Country Link
DO (1) DOP2003000786A (en)

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