DK561487A - 4-phenylsulfonyl-3,4-dihydro-2(1h)-quinoxalinon-1-alkansyre-forbindelser og farmaceutiske praeparater indeholdende disse - Google Patents

4-phenylsulfonyl-3,4-dihydro-2(1h)-quinoxalinon-1-alkansyre-forbindelser og farmaceutiske praeparater indeholdende disse

Info

Publication number: DK561487A
Authority: DK; Denmark
Prior art keywords: quinoxalinon; phenylsulphonyl; dihydro; pharmaceutical preparations; acid compounds
Prior art date: 1986-10-30

Application number

DK561487A

Other languages

English (en)

Other versions

DK561487D0 (da

Inventor

Reinhard Sarges

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-10-30

Filing date

1987-10-27

Publication date

1988-08-08

1987-10-27 Application filed by Pfizer filed Critical Pfizer

1987-10-27 Publication of DK561487D0 publication Critical patent/DK561487D0/da

1988-08-08 Publication of DK561487A publication Critical patent/DK561487A/da

Links

239000002253 acid Substances 0.000 title abstract 2
150000001875 compounds Chemical class 0.000 title 1
239000000825 pharmaceutical preparation Substances 0.000 title 1
FFRYUAVNPBUEIC-UHFFFAOYSA-N quinoxalin-2-ol Chemical compound C1=CC=CC2=NC(O)=CN=C21 FFRYUAVNPBUEIC-UHFFFAOYSA-N 0.000 abstract 2
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
125000005036 alkoxyphenyl group Chemical group 0.000 abstract 1
125000005037 alkyl phenyl group Chemical group 0.000 abstract 1
125000004799 bromophenyl group Chemical group 0.000 abstract 1
150000001768 cations Chemical class 0.000 abstract 1
125000000068 chlorophenyl group Chemical group 0.000 abstract 1
230000001684 chronic effect Effects 0.000 abstract 1
206010012601 diabetes mellitus Diseases 0.000 abstract 1
125000004188 dichlorophenyl group Chemical group 0.000 abstract 1
125000001207 fluorophenyl group Chemical group 0.000 abstract 1
125000004464 hydroxyphenyl group Chemical group 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/50—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to ring nitrogen atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Diabetes (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Obesity (AREA)
Hematology (AREA)
Emergency Medicine (AREA)
Endocrinology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Ophthalmology & Optometry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)
Cosmetics (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK561487A 1986-10-30 1987-10-27 4-phenylsulfonyl-3,4-dihydro-2(1h)-quinoxalinon-1-alkansyre-forbindelser og farmaceutiske praeparater indeholdende disse DK561487A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/US1986/002335 WO1992005160A1 (en)	1986-10-30	1986-10-30	4-arylsulfonyl-3,4-dihydro-2(1h)-quinoxalinone-1-alkanoic acids, esters, and salts

Publications (2)

Publication Number	Publication Date
DK561487D0 DK561487D0 (da)	1987-10-27
DK561487A true DK561487A (da)	1988-08-08

Family

ID=22195697

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK561487A DK561487A (da)	1986-10-30	1987-10-27	4-phenylsulfonyl-3,4-dihydro-2(1h)-quinoxalinon-1-alkansyre-forbindelser og farmaceutiske praeparater indeholdende disse

Country Status (11)

Country	Link
US (1)	US4940708A (da)
EP (1)	EP0266102B1 (da)
JP (1)	JPS63295566A (da)
AT (1)	ATE86985T1 (da)
DE (1)	DE3784835T2 (da)
DK (1)	DK561487A (da)
ES (1)	ES2046206T3 (da)
GR (1)	GR3007402T3 (da)
IE (1)	IE68851B1 (da)
PT (1)	PT85998B (da)
WO (1)	WO1992005160A1 (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4940708A (en) *	1986-10-30	1990-07-10	Pfizer Inc.	4-arylsulfonyl-3,4-dihydro-2(1H)-quinoxalinone-1-alkanoic acids, esters, and salts
DK0509398T3 (da) *	1991-04-15	2002-01-14	Aventis Pharma Gmbh	Quinoxaliner, fremgangsmåder til deres fremstilling samt deres anvendelse
US6369057B1 (en)	1991-04-15	2002-04-09	Aventis Pharma Deutschland Gmbh	Quinoxalines, processes for their preparation and their use
US7351709B2 (en)	2004-06-09	2008-04-01	Wyeth	Estrogen receptor ligands
EP1940805A4 (en) *	2005-08-26	2009-11-11	Methylgene Inc	BENZODIAZEPIN AND BENZOPIPERAZINANALOGA AS INHIBITORS OF HISTONDEACETYLASE
SI2276795T1 (sl)	2008-04-30	2015-09-30	Xyleco, Inc.	Obdelava biomase
US8236535B2 (en)	2008-04-30	2012-08-07	Xyleco, Inc.	Processing biomass
US7867358B2 (en)	2008-04-30	2011-01-11	Xyleco, Inc.	Paper products and methods and systems for manufacturing such products
US8212087B2 (en)	2008-04-30	2012-07-03	Xyleco, Inc.	Processing biomass
KR101689797B1 (ko)	2008-10-28	2016-12-26	질레코 인코포레이티드	재료의 처리방법

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3821383A (en) *	1972-07-10	1974-06-28	Ayerst Mckenna & Harrison	Compositions for and a method of treating diabetic complications
JPS5559314A (en) *	1978-10-27	1980-05-02	Sony Corp	Magnetic scale signal detector
US4209527A (en) *	1979-05-16	1980-06-24	Pfizer Inc.	Benzimidazolone derivatives
US4940708A (en) *	1986-10-30	1990-07-10	Pfizer Inc.	4-arylsulfonyl-3,4-dihydro-2(1H)-quinoxalinone-1-alkanoic acids, esters, and salts

1986
- 1986-10-30 US US07/424,298 patent/US4940708A/en not_active Expired - Fee Related
- 1986-10-30 WO PCT/US1986/002335 patent/WO1992005160A1/en unknown
1987
- 1987-01-27 IE IE287787A patent/IE68851B1/en not_active IP Right Cessation
- 1987-10-16 DE DE8787309160T patent/DE3784835T2/de not_active Expired - Fee Related
- 1987-10-16 ES ES198787309160T patent/ES2046206T3/es not_active Expired - Lifetime
- 1987-10-16 AT AT87309160T patent/ATE86985T1/de active
- 1987-10-16 EP EP87309160A patent/EP0266102B1/en not_active Expired - Lifetime
- 1987-10-22 JP JP62267597A patent/JPS63295566A/ja active Granted
- 1987-10-27 PT PT85998A patent/PT85998B/pt not_active IP Right Cessation
- 1987-10-27 DK DK561487A patent/DK561487A/da not_active Application Discontinuation
1993
- 1993-03-18 GR GR930400553T patent/GR3007402T3/el unknown

Also Published As

Publication number	Publication date
EP0266102A2 (en)	1988-05-04
DE3784835D1 (de)	1993-04-22
DK561487D0 (da)	1987-10-27
EP0266102B1 (en)	1993-03-17
ATE86985T1 (de)	1993-04-15
ES2046206T3 (es)	1994-02-01
WO1992005160A1 (en)	1992-04-02
DE3784835T2 (de)	1993-06-24
EP0266102A3 (en)	1989-11-23
IE68851B1 (en)	1996-07-24
PT85998B (pt)	1990-08-31
JPS63295566A (ja)	1988-12-01
JPH0536436B2 (da)	1993-05-31
US4940708A (en)	1990-07-10
IE872877L (en)	1988-04-28
PT85998A (en)	1987-11-01
GR3007402T3 (da)	1993-07-30

Legal Events

Date	Code	Title	Description
1987-10-27	A0	Application filed
1997-06-16	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
NO905572D0 (no)	1990-12-21	Fremgangsmaate for fremstilling av peptidforbindelser.
DK57388A (da)	1988-08-05	Thiazolidinonderivater, fremgangsmaade til deres fremstilling samt anvendelsen heraf
FI904602A0 (fi)	1990-09-19	Pyrazoloderivat, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska blandningar.
DK0379979T3 (da)	1997-04-07
ATE68180T1 (de)	1991-10-15	Morpholinoethylester von mycophenolsaeure und ihre derivate, ihre herstellung und verwendung in pharmazeutische zusammensetzungen.
DK0622361T3 (da)	2001-12-03	Heterocykliske forbindelser som bradykininantagonister
DK355287D0 (da)	1987-07-09	2-oxoindolin-1-alkansyre-forbindelser og farmaceutiske praeparater indeholdende disse
DK0412404T3 (da)	1996-02-26	Thiazolderivater, fremgangsmåder til fremstilling deraf og farmaceutiske præparater omfattende derivaterne
ATE104971T1 (de)	1994-05-15	2-aminopyrimidinon-derivate.
DK0516941T3 (da)	1997-01-06	Pyrazolopyridinforbindelser og fremgangsmåder til fremstilling deraf
DK561487A (da)	1988-08-08	4-phenylsulfonyl-3,4-dihydro-2(1h)-quinoxalinon-1-alkansyre-forbindelser og farmaceutiske praeparater indeholdende disse
ES2063452T3 (es)	1995-01-01	Preparacion y uso de esteres y derivados de n-yodopropargil oxicarbonil aminoacido como agentes antimicrobianos.
DE3866012D1 (de)	1991-12-12	Antiarrhythmische heilmittel.
DK148288A (da)	1988-12-30	N-phenethylaminoalkyl-benzamid-forbindelser, deres anvendelse til fremstilling af antiarrhythmia-laegemidler og farmaceutiske praeparater indeholdende forbindelserne
DE68923231D1 (de)	1995-08-03	Antihypertensive 3-Piperidinylindazol-Derivate.
DK655088D0 (da)	1988-11-24	N-(biphenyl-2-ylmethyl)-3-hydroxyglutaramidsyre-forbindelser, farmaceutiske praeparater indeholdende disse og deres anvendelse til fremstilling af hypocholesterolaemiske laegemidler
NO903084D0 (no)	1990-07-11	Farmasoeytisk anvendbare thiazol-derivater og fremgangsmaate for deres fremstilling.
DK210387A (da)	1987-10-29	Heterocykliske forbindelser og fremgangsmaade til deres fremstilling samt farmaceutiske midler indeholdende disse
DE69011174D1 (de)	1994-09-08	Catecholaminester.