DK322088A - Imidazoquicxalinforbindelser, deres fremstilling og anvendelse - Google Patents

Imidazoquicxalinforbindelser, deres fremstilling og anvendelse

Info

Publication number
DK322088A
DK322088A DK322088A DK322088A DK322088A DK 322088 A DK322088 A DK 322088A DK 322088 A DK322088 A DK 322088A DK 322088 A DK322088 A DK 322088A DK 322088 A DK322088 A DK 322088A
Authority
DK
Denmark
Prior art keywords
imidazoquicxal
rines
preparation
chem
alkyl
Prior art date
Application number
DK322088A
Other languages
English (en)
Other versions
DK322088D0 (da
DK161148B (da
DK161148C (da
Inventor
Holger Claus Hansen
Frank Waetjen
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrosan As filed Critical Ferrosan As
Publication of DK322088D0 publication Critical patent/DK322088D0/da
Priority to DK322088A priority Critical patent/DK161148C/da
Priority to IL90543A priority patent/IL90543A0/xx
Priority to DE68918003T priority patent/DE68918003T2/de
Priority to ES89305728T priority patent/ES2060769T3/es
Priority to AT89305728T priority patent/ATE111100T1/de
Priority to EP89305728A priority patent/EP0347094B1/en
Priority to PH38760A priority patent/PH26337A/en
Priority to US07/363,585 priority patent/US5034530A/en
Priority to ZA894430A priority patent/ZA894430B/xx
Priority to NZ229499A priority patent/NZ229499A/xx
Priority to CA000602682A priority patent/CA1327798C/en
Priority to NO892456A priority patent/NO170806C/no
Priority to JP1148537A priority patent/JPH0236184A/ja
Priority to AU36244/89A priority patent/AU618366B2/en
Priority to IE189289A priority patent/IE69963B1/en
Priority to FI892908A priority patent/FI92204C/fi
Priority to PT90865A priority patent/PT90865B/pt
Priority to KR1019890008164A priority patent/KR910000665A/ko
Publication of DK322088A publication Critical patent/DK322088A/da
Publication of DK161148B publication Critical patent/DK161148B/da
Application granted granted Critical
Publication of DK161148C publication Critical patent/DK161148C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
DK322088A 1988-06-14 1988-06-14 Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne DK161148C (da)

Priority Applications (18)

Application Number Priority Date Filing Date Title
DK322088A DK161148C (da) 1988-06-14 1988-06-14 Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne
IL90543A IL90543A0 (en) 1988-06-14 1989-06-06 Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them
DE68918003T DE68918003T2 (de) 1988-06-14 1989-06-07 Imidazochinoxalinverbindungen und ihre Herstellung und Verwendung.
ES89305728T ES2060769T3 (es) 1988-06-14 1989-06-07 Compuestos de imidazoquinoxalina y su preparacion y uso.
AT89305728T ATE111100T1 (de) 1988-06-14 1989-06-07 Imidazochinoxalinverbindungen und ihre herstellung und verwendung.
EP89305728A EP0347094B1 (en) 1988-06-14 1989-06-07 Imidazoquinoxaline compounds and their preparation and use
PH38760A PH26337A (en) 1988-06-14 1989-06-08 Imidazoquinoxaline compounds pharmaceuticals compositions containing the same and method of use thereof
US07/363,585 US5034530A (en) 1988-06-14 1989-06-08 Imidazoquinoxaline compounds and their preparation and use
ZA894430A ZA894430B (en) 1988-06-14 1989-06-12 Imidazoquinoxaline compounds and their preparation and use
NZ229499A NZ229499A (en) 1988-06-14 1989-06-12 Imidazo(1,5-a)quinoxaline derivatives and pharmaceutical compositions
CA000602682A CA1327798C (en) 1988-06-14 1989-06-13 Imidazoquinoxaline compounds and their preparation and use
NO892456A NO170806C (no) 1988-06-14 1989-06-13 Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxalinforbindelser
JP1148537A JPH0236184A (ja) 1988-06-14 1989-06-13 イミダゾキノキサリン化合物、その製造方法並びにその使用
AU36244/89A AU618366B2 (en) 1988-06-14 1989-06-13 Imidazoquinoxaline compounds and their preparation and use
IE189289A IE69963B1 (en) 1988-06-14 1989-06-13 Imidazoquinoxaline compounds and their preparation and use
FI892908A FI92204C (fi) 1988-06-14 1989-06-14 Menetelmä uusien terapeuttisesti käyttökelpoisten imidatso/1,5-a/kinoksaliinijohdannaisten valmistamiseksi
PT90865A PT90865B (pt) 1988-06-14 1989-06-14 Processo para a preparacao de compostos de imidazoquinoxalina e de composicoes farmaceuticas que os contem
KR1019890008164A KR910000665A (ko) 1988-06-14 1989-06-14 이미다조퀴녹살린 화합물, 이의 제조방법 및 이의 용도

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK322088A DK161148C (da) 1988-06-14 1988-06-14 Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne
DK322088 1988-06-14

Publications (4)

Publication Number Publication Date
DK322088D0 DK322088D0 (da) 1988-06-14
DK322088A true DK322088A (da) 1990-03-27
DK161148B DK161148B (da) 1991-06-03
DK161148C DK161148C (da) 1991-11-18

Family

ID=8120424

Family Applications (1)

Application Number Title Priority Date Filing Date
DK322088A DK161148C (da) 1988-06-14 1988-06-14 Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne

Country Status (18)

Country Link
US (1) US5034530A (da)
EP (1) EP0347094B1 (da)
JP (1) JPH0236184A (da)
KR (1) KR910000665A (da)
AT (1) ATE111100T1 (da)
AU (1) AU618366B2 (da)
CA (1) CA1327798C (da)
DE (1) DE68918003T2 (da)
DK (1) DK161148C (da)
ES (1) ES2060769T3 (da)
FI (1) FI92204C (da)
IE (1) IE69963B1 (da)
IL (1) IL90543A0 (da)
NO (1) NO170806C (da)
NZ (1) NZ229499A (da)
PH (1) PH26337A (da)
PT (1) PT90865B (da)
ZA (1) ZA894430B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK160876C (da) * 1987-12-08 1991-10-14 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar
US5276028A (en) * 1990-06-22 1994-01-04 Nordisk A/S Imidazoquinoxaline compounds
US5371080A (en) * 1990-06-22 1994-12-06 Novo Nordisk A/S Imidazoquinazoline compounds and their use
DK151890D0 (da) * 1990-06-22 1990-06-22 Ferrosan As Heterocykliske forbindelser deres fremstilling og brug
US5153196A (en) * 1991-06-05 1992-10-06 Eli Lilly And Company Excitatory amino acid receptor antagonists and methods for the use thereof
JP3147902B2 (ja) * 1991-06-14 2001-03-19 ファルマシア・アンド・アップジョン・カンパニー イミダゾ〔１，５−ａ〕キノキサリン
US6635626B1 (en) 1997-08-25 2003-10-21 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
US6235740B1 (en) 1997-08-25 2001-05-22 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
JP2002505330A (ja) * 1998-03-04 2002-02-19 ブリストル−マイヤーズ スクイブ カンパニー ヘテロシクロ−置換イミダゾピラジン・たんぱくチロシンキナーゼ抑制剤
US20040180898A1 (en) * 2003-03-03 2004-09-16 Bang-Chi Chen Processes for preparing imidazoquinoxalinones, heterocyclic-substituted imidazopyrazinones, imidazoquinoxalines and heterocyclic-substituted imidazopyrazines
US20090143391A1 (en) * 2007-11-30 2009-06-04 Norbert Hofgen Aryl and heteroaryl fused imidazo [1,5-a] pyrazines as inhibitors of phosphodiesterase 10
WO2009070584A1 (en) 2007-11-30 2009-06-04 Wyeth Aryl and heteroaryl fused imidazo[1,5-a]pyrazines as inhibitors of phosphodiesterase 10
TW201111383A (en) * 2009-05-29 2011-04-01 Wyeth Llc Substituted imidazo[1,5-a]quinoxalines as inhibitors of phosphodiesterase 10

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
EP0221699B1 (en) * 1985-10-19 1990-01-10 Beecham Group Plc Composition for the treatment of infections
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse

Also Published As

Publication number Publication date
KR910000665A (ko) 1991-01-30
JPH0236184A (ja) 1990-02-06
DE68918003D1 (de) 1994-10-13
NO892456L (no) 1989-12-15
ES2060769T3 (es) 1994-12-01
NZ229499A (en) 1991-04-26
AU3624489A (en) 1989-12-21
NO170806C (no) 1992-12-09
EP0347094B1 (en) 1994-09-07
CA1327798C (en) 1994-03-15
DK322088D0 (da) 1988-06-14
FI92204B (fi) 1994-06-30
NO892456D0 (no) 1989-06-13
IE69963B1 (en) 1996-10-16
EP0347094A1 (en) 1989-12-20
NO170806B (no) 1992-08-31
DK161148B (da) 1991-06-03
IE891892L (en) 1989-12-14
DK161148C (da) 1991-11-18
PT90865A (pt) 1989-12-29
FI892908A (fi) 1989-12-15
ATE111100T1 (de) 1994-09-15
FI892908A0 (fi) 1989-06-14
PT90865B (pt) 1994-11-30
AU618366B2 (en) 1991-12-19
FI92204C (fi) 1994-10-10
US5034530A (en) 1991-07-23
IL90543A0 (en) 1990-01-18
DE68918003T2 (de) 1995-01-05
PH26337A (en) 1992-04-29
ZA894430B (en) 1990-02-28

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