DK265780A - Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling - Google Patents

Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling

Info

Publication number
DK265780A
DK265780A DK265780A DK265780A DK265780A DK 265780 A DK265780 A DK 265780A DK 265780 A DK265780 A DK 265780A DK 265780 A DK265780 A DK 265780A DK 265780 A DK265780 A DK 265780A
Authority
DK
Denmark
Prior art keywords
preparation
encaphalin
analgetics
antipsychotics
intermediates
Prior art date
Application number
DK265780A
Other languages
Danish (da)
English (en)
Inventor
A A Carr
R A Farr
J M Kane
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of DK265780A publication Critical patent/DK265780A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK265780A 1979-06-21 1980-06-20 Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling DK265780A (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5095079A 1979-06-21 1979-06-21
US06/130,431 US4341698A (en) 1979-06-21 1980-03-14 Enkaphalin derivatives
AU91877/82A AU559278B2 (en) 1979-06-21 1982-12-24 Piperazines

Publications (1)

Publication Number Publication Date
DK265780A true DK265780A (da) 1980-12-22

Family

ID=36764304

Family Applications (1)

Application Number Title Priority Date Filing Date
DK265780A DK265780A (da) 1979-06-21 1980-06-20 Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling

Country Status (17)

Country Link
US (1) US4341698A (de)
AU (1) AU559278B2 (de)
CA (1) CA1161838A (de)
CH (2) CH645363A5 (de)
DE (1) DE3022401A1 (de)
DK (1) DK265780A (de)
ES (1) ES8105720A1 (de)
FR (2) FR2459236A1 (de)
GB (3) GB2051821B (de)
IE (1) IE49834B1 (de)
IL (1) IL60245A (de)
IT (1) IT1148277B (de)
NL (1) NL8003580A (de)
NO (1) NO801855L (de)
NZ (1) NZ193934A (de)
PH (1) PH19222A (de)
SE (3) SE447250B (de)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6194435B1 (en) 1996-10-11 2001-02-27 Cor Therapeutics, Inc. Lactams as selective factor Xa inhibitors
US6369080B2 (en) 1996-10-11 2002-04-09 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6063794A (en) 1996-10-11 2000-05-16 Cor Therapeutics Inc. Selective factor Xa inhibitors
US6262047B1 (en) 1996-10-11 2001-07-17 Cor Therapeutics, Inc. Selective factor Xa inhibitors
WO1998046628A1 (en) * 1997-04-14 1998-10-22 Cor Therapeutics, Inc. SELECTIVE FACTOR Xa INHIBITORS
EP0977773A1 (de) 1997-04-14 2000-02-09 Cor Therapeutics, Inc. Selektive faktor xa-inhibitoren
WO1998046626A1 (en) 1997-04-14 1998-10-22 Cor Therapeutics, Inc. SELECTIVE FACTOR Xa INHIBITORS
US6333321B1 (en) 1997-08-11 2001-12-25 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6228854B1 (en) 1997-08-11 2001-05-08 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6218382B1 (en) 1997-08-11 2001-04-17 Cor Therapeutics, Inc Selective factor Xa inhibitors
CA2601709C (en) 2005-03-22 2017-02-14 Azevan Pharmaceuticals, Inc. Beta-lactamylalkanoic acids
CN101268068B (zh) 2005-07-19 2015-12-02 阿泽范药品公司 β-内酰胺基苯丙氨酸、半胱氨酸和丝氨酸血管加压素拮抗剂
US8114844B2 (en) * 2006-03-30 2012-02-14 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptidomimetics
US7964181B2 (en) * 2006-03-30 2011-06-21 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
US7795221B2 (en) * 2006-03-30 2010-09-14 Palatin Technologies, Inc. Linear natriuretic peptide constructs
US8580746B2 (en) 2006-03-30 2013-11-12 Palatin Technologies, Inc. Amide linkage cyclic natriuretic peptide constructs
DK2001518T3 (da) * 2006-03-30 2013-10-07 Palatin Technologies Inc Cykliske natriuretiske peptidfremstillinger
WO2007115164A2 (en) * 2006-03-30 2007-10-11 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
CN101563319B (zh) * 2006-12-19 2012-09-05 弗·哈夫曼-拉罗切有限公司 杂芳基吡咯烷基和哌啶基甲酮衍生物
KR20110010783A (ko) * 2008-06-18 2011-02-07 에프. 호프만-라 로슈 아게 Ｍｒｉ로서의 아릴 케톤
ES2858499T3 (es) 2010-07-01 2021-09-30 Azevan Pharmaceuticals Inc Compuestos para su uso en el tratamiento de trastorno explosivo intermitente
KR20160130853A (ko) 2014-03-28 2016-11-14 아제반 파마슈티칼스, 인코퍼레이티드 신경변성 질환을 치료하기 조성물 및 방법
TW201919625A (zh) 2017-09-15 2019-06-01 美商愛治凡製藥公司 用於治療腦損傷之組合物及方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2604845A1 (de) * 1976-02-07 1977-08-18 Knoll Ag Neue piperazinderivate
US4254107A (en) * 1979-11-27 1981-03-03 Merck & Co., Inc. Long-lasting agonists of enkephalin

Also Published As

Publication number Publication date
GB2106515B (en) 1983-11-23
CH648835A5 (de) 1985-04-15
GB2132605B (en) 1985-01-03
FR2473042B1 (de) 1983-07-01
GB2132605A (en) 1984-07-11
IT1148277B (it) 1986-11-26
SE8500877L (sv) 1985-02-22
FR2459236A1 (fr) 1981-01-09
AU559278B2 (en) 1987-03-05
NL8003580A (nl) 1980-12-23
GB2106515A (en) 1983-04-13
SE460541B (sv) 1989-10-23
US4341698A (en) 1982-07-27
DE3022401A1 (de) 1981-01-08
SE447250B (sv) 1986-11-03
SE460540B (sv) 1989-10-23
GB2051821A (en) 1981-01-21
IT8049032A0 (it) 1980-06-20
PH19222A (en) 1986-02-12
IE49834B1 (en) 1985-12-25
GB2051821B (en) 1983-04-27
SE8004254L (sv) 1980-12-22
SE8500877D0 (sv) 1985-02-22
ES492566A0 (es) 1981-06-16
NZ193934A (en) 1983-02-15
ES8105720A1 (es) 1981-06-16
IL60245A (en) 1985-08-30
NO801855L (no) 1980-12-22
SE8500878D0 (sv) 1985-02-22
AU9187782A (en) 1983-04-21
CH645363A5 (de) 1984-09-28
FR2459236B1 (de) 1984-01-06
IE801152L (en) 1980-12-21
FR2473042A1 (fr) 1981-07-10
CA1161838A (en) 1984-02-07

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Legal Events

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AHS Application shelved for other reasons than non-payment