DK23088A - Piperazinylpyrimidinforbindelse og farmaceutisk praeparat indeholdende en saadan forbindelse - Google Patents

Piperazinylpyrimidinforbindelse og farmaceutisk praeparat indeholdende en saadan forbindelse

Info

Publication number
DK23088A
DK23088A DK23088A DK23088A DK23088A DK 23088 A DK23088 A DK 23088A DK 23088 A DK23088 A DK 23088A DK 23088 A DK23088 A DK 23088A DK 23088 A DK23088 A DK 23088A
Authority
DK
Denmark
Prior art keywords
connection
piperazinylpyrimide
pharmaceutical preparation
preparation containing
pharmaceutical
Prior art date
Application number
DK23088A
Other languages
English (en)
Other versions
DK23088D0 (da
Inventor
John J Baldwin
Richard L Tolman
Mu T Wu
Arthur F Wagner
Adolph Pietruszkiewicz
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/005,720 external-priority patent/US4871739A/en
Priority claimed from US07/091,471 external-priority patent/US4889856A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK23088D0 publication Critical patent/DK23088D0/da
Publication of DK23088A publication Critical patent/DK23088A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK23088A 1987-01-21 1988-01-20 Piperazinylpyrimidinforbindelse og farmaceutisk praeparat indeholdende en saadan forbindelse DK23088A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/005,720 US4871739A (en) 1987-01-21 1987-01-21 Substituted 6H-7,8-dihydrothiapyrano(3,2-D)-pyrimidines as hyopglycemic agents
US07/091,471 US4889856A (en) 1987-08-31 1987-08-31 7,8-dihydro-4-(1-pierazinyl)-6H-thiopyrano-[3,2-d] pyrimidines as β-blockers

Publications (2)

Publication Number Publication Date
DK23088D0 DK23088D0 (da) 1988-01-20
DK23088A true DK23088A (da) 1988-07-22

Family

ID=26674696

Family Applications (1)

Application Number Title Priority Date Filing Date
DK23088A DK23088A (da) 1987-01-21 1988-01-20 Piperazinylpyrimidinforbindelse og farmaceutisk praeparat indeholdende en saadan forbindelse

Country Status (4)

Country Link
EP (1) EP0276057B1 (da)
CA (1) CA1308410C (da)
DE (1) DE3888215T2 (da)
DK (1) DK23088A (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8912335D0 (en) * 1989-05-30 1989-07-12 Smithkline Beckman Intercredit Compounds
US6608053B2 (en) * 2000-04-27 2003-08-19 Yamanouchi Pharmaceutical Co., Ltd. Fused heteroaryl derivatives
US7968545B2 (en) * 2003-08-05 2011-06-28 Vertex Pharmaceuticals Inc. Compositions useful as inhibitors of voltage-gated ion channels
JP4862654B2 (ja) 2004-10-08 2012-01-25 アステラス製薬株式会社 芳香環縮合ピリミジン誘導体
TW200621257A (en) * 2004-10-20 2006-07-01 Astellas Pharma Inc Pyrimidine derivative fused with nonaromatic ring
CA3008171A1 (en) 2015-12-22 2017-06-29 SHY Therapeutics LLC Compounds for the treatment of cancer and inflammatory disease
BR112019027640A2 (pt) 2017-06-21 2020-07-07 SHY Therapeutics LLC composto, método para testar a capacidade de um ou mais compostos, método para inibir a função de ras, método para inibir a função de rho, método para inibir a função de rac, composição farmacêutica

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1470336A1 (de) * 1962-07-04 1969-03-20 Thomae Gmbh Dr K Neue Dihydrothieno-[3,4-d]-pyrimidine und Verfahren zu ihrer Herstellung
NL124131C (da) * 1963-06-17
DE1251765B (de) * 1963-07-23 1967-10-12 Dr Karl Thomae Gesellschaft mit beschrankter Haftung Biberach/Riß Verfahren zur Herstellung von neuen 5H - Dihydrothiopyrano [4 3 d] pynmidinen
DE1470354A1 (de) * 1963-12-16 1969-10-09 Thomae Gmbh Dr K Neue 4H-m-Dithiino[5,4-d]-pyrimidine und Verfahren zu ihrer Herstellung
DE1470356A1 (de) * 1964-01-15 1970-04-30 Thomae Gmbh Dr K Neue Thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
DE3888215T2 (de) 1994-09-08
CA1308410C (en) 1992-10-06
EP0276057A3 (en) 1989-09-06
DE3888215D1 (de) 1994-04-14
EP0276057B1 (en) 1994-03-09
EP0276057A2 (en) 1988-07-27
DK23088D0 (da) 1988-01-20

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment