DK152505C - Analogifremgangsmaade til fremstilling af et somatostatin-analogt cyclisk hexapeptid - Google Patents

Analogifremgangsmaade til fremstilling af et somatostatin-analogt cyclisk hexapeptid

Info

Publication number: DK152505C
Authority: DK; Denmark
Prior art keywords: preparing; somatostatin analogue; cyclic hexapeptide; analogy procedure; analogue cyclic
Prior art date: 1979-10-31

Application number

DK460580A

Other languages

English (en)

Other versions

DK460580A (da

DK152505B (da

Inventor

Daniel F Veber

Roger M Freidinger

Original Assignee

Merck & Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-10-31

Filing date

1980-10-30

Publication date

1988-07-25

1979-10-31 Priority claimed from US06/089,827 external-priority patent/US4235886A/en

1980-10-30 Application filed by Merck & Co Inc filed Critical Merck & Co Inc

1981-05-01 Publication of DK460580A publication Critical patent/DK460580A/da

1988-03-07 Publication of DK152505B publication Critical patent/DK152505B/da

1988-07-25 Application granted granted Critical

1988-07-25 Publication of DK152505C publication Critical patent/DK152505C/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biochemistry (AREA)
Biophysics (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Medicinal Chemistry (AREA)
Analytical Chemistry (AREA)
Gastroenterology & Hepatology (AREA)
Zoology (AREA)
Toxicology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Endocrinology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)

DK460580A 1979-10-31 1980-10-30 Analogifremgangsmaade til fremstilling af et somatostatin-analogt cyclisk hexapeptid DK152505C (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US8982879A	1979-10-31	1979-10-31
US8982779		1979-10-31
US06/089,827 US4235886A (en)	1979-10-31	1979-10-31	Cyclic hexapeptide somatostatin analogs
US8982879		1979-10-31

Publications (3)

Publication Number	Publication Date
DK460580A DK460580A (da)	1981-05-01
DK152505B DK152505B (da)	1988-03-07
DK152505C true DK152505C (da)	1988-07-25

Family

ID=26780979

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK460580A DK152505C (da)	1979-10-31	1980-10-30	Analogifremgangsmaade til fremstilling af et somatostatin-analogt cyclisk hexapeptid

Country Status (17)

Country	Link
EP (1)	EP0029310B1 (da)
KR (1)	KR860001961B1 (da)
AU (1)	AU540140B2 (da)
CA (1)	CA1216844A (da)
DD (1)	DD153684A5 (da)
DE (1)	DE3064499D1 (da)
DK (1)	DK152505C (da)
ES (1)	ES496424A0 (da)
FI (1)	FI74711C (da)
GR (1)	GR70725B (da)
IE (1)	IE50364B1 (da)
NO (1)	NO150958C (da)
NZ (1)	NZ195303A (da)
PL (1)	PL128347B1 (da)
PT (1)	PT71966B (da)
RO (1)	RO81523A (da)
YU (1)	YU278780A (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4360516A (en) *	1981-04-13	1982-11-23	Merck & Co., Inc.	Modified D-retro cyclic hexapeptide somatostatin analogs
US4374060A (en) *	1981-07-15	1983-02-15	Merck & Co., Inc.	Process for the preparation of cyclic hexapeptide
US4427661A (en) *	1982-07-30	1984-01-24	Merck & Co., Inc.	Fluorinated cyclic hexapeptide somatostatin analogs
EP0113029B1 (en) *	1982-12-06	1989-04-19	Merck & Co. Inc.	Dicyclic hexapeptides, processes for their preparation and pharmaceutical compositions containing them
DE3303345A1 (de) *	1983-02-02	1984-08-02	Hoechst Ag, 6230 Frankfurt	Cyclische peptide mit somatostatin-wirkung
US4505897A (en) *	1983-04-18	1985-03-19	The Administrators Of The Tulane Educational Fund	Cyclic pentapeptides displaying somatostatin antagonism and method of treatment of mammals therewith
US5620675A (en)	1992-06-23	1997-04-15	Diatech, Inc.	Radioactive peptides
EP1092726B1 (en) *	1993-06-23	2006-08-23	Diatide, Inc.	Radioactively-labeled somatostatin derived peptides for imaging and therapeutics uses
US5932189A (en) *	1994-07-29	1999-08-03	Diatech, Inc.	Cyclic peptide somatostatin analogs
US6051206A (en) *	1994-06-03	2000-04-18	Diatide, Inc	Radiolabeled somatostatin-derived peptides for imaging and therapeutic uses
MY147327A (en)	1995-06-29	2012-11-30	Novartis Ag	Somatostatin peptides
GB0018891D0 (en)	2000-08-01	2000-09-20	Novartis Ag	Organic compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SE7708136L (sv) *	1976-08-02	1978-02-03	Merck & Co Inc	Cykliska hexapeptider
IT1105131B (it) *	1977-06-08	1985-10-28	Merck & Co Inc	Peptidi analoghi della somatostatina dotati di piu' lunga e maggiore attivita' biologica e relativo procedimento di protezione
LU78191A1 (de) *	1977-09-28	1979-05-25	Ciba Geigy Ag	Verfahren zur herstellung von neuen cyclopeptiden

1980
- 1980-10-20 NZ NZ195303A patent/NZ195303A/en unknown
- 1980-10-21 FI FI803306A patent/FI74711C/fi not_active IP Right Cessation
- 1980-10-22 AU AU63581/80A patent/AU540140B2/en not_active Ceased
- 1980-10-24 PT PT71966A patent/PT71966B/pt unknown
- 1980-10-25 GR GR63223A patent/GR70725B/el unknown
- 1980-10-27 RO RO80102446A patent/RO81523A/ro unknown
- 1980-10-28 DE DE8080303826T patent/DE3064499D1/de not_active Expired
- 1980-10-28 EP EP80303826A patent/EP0029310B1/en not_active Expired
- 1980-10-28 DD DD80224779A patent/DD153684A5/de unknown
- 1980-10-28 CA CA000363416A patent/CA1216844A/en not_active Expired
- 1980-10-28 IE IE2224/80A patent/IE50364B1/en not_active IP Right Cessation
- 1980-10-29 KR KR1019800004142A patent/KR860001961B1/ko active
- 1980-10-30 NO NO803245A patent/NO150958C/no unknown
- 1980-10-30 ES ES496424A patent/ES496424A0/es active Granted
- 1980-10-30 PL PL1980227577A patent/PL128347B1/pl unknown
- 1980-10-30 YU YU02787/80A patent/YU278780A/xx unknown
- 1980-10-30 DK DK460580A patent/DK152505C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
FI74711C (fi)	1988-03-10
PL227577A1 (da)	1981-10-02
PL128347B1 (en)	1984-01-31
DK460580A (da)	1981-05-01
ES8202787A1 (es)	1982-02-16
DK152505B (da)	1988-03-07
GR70725B (da)	1983-01-18
RO81523A (ro)	1983-08-03
IE802224L (en)	1981-04-30
NO803245L (no)	1981-05-04
EP0029310A1 (en)	1981-05-27
KR860001961B1 (ko)	1986-11-05
DE3064499D1 (en)	1983-09-08
YU278780A (en)	1983-01-21
IE50364B1 (en)	1986-04-02
FI74711B (fi)	1987-11-30
NO150958C (no)	1985-01-16
CA1216844A (en)	1987-01-20
ES496424A0 (es)	1982-02-16
AU6358180A (en)	1981-05-07
PT71966B (en)	1982-03-31
EP0029310B1 (en)	1983-08-03
KR830004223A (ko)	1983-07-09
NO150958B (no)	1984-10-08
FI803306L (fi)	1981-05-01
AU540140B2 (en)	1984-11-01
RO81523B (ro)	1983-07-30
NZ195303A (en)	1984-10-19
PT71966A (en)	1980-11-01
DD153684A5 (de)	1982-01-27

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Legal Events

Date	Code	Title	Description
1994-06-20	PBP	Patent lapsed