DK140498C - - Google Patents

Info

Publication number
DK140498C
DK140498C DK145373A DK145373A DK140498C DK 140498 C DK140498 C DK 140498C DK 145373 A DK145373 A DK 145373A DK 145373 A DK145373 A DK 145373A DK 140498 C DK140498 C DK 140498C
Authority
DK
Denmark
Application number
DK145373A
Other versions
DK140498B (da
Inventor
H Nishimura
M Shimizu
H Uno
T Hirooka
Y Masuda
M Kurokawa
Original Assignee
Dainippon Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2786672A external-priority patent/JPS5616154B2/ja
Priority claimed from JP2786572A external-priority patent/JPS5545545B2/ja
Application filed by Dainippon Pharmaceutical Co Ltd filed Critical Dainippon Pharmaceutical Co Ltd
Publication of DK140498B publication Critical patent/DK140498B/da
Application granted granted Critical
Publication of DK140498C publication Critical patent/DK140498C/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK145373AA 1972-03-17 1973-03-16 Analogifremgangsmåde til fremstilling af 3-substituerede 1,2-benzisoxazolderivater. DK140498B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2786672A JPS5616154B2 (da) 1972-03-17 1972-03-17
JP2786572A JPS5545545B2 (da) 1972-03-17 1972-03-17

Publications (2)

Publication Number Publication Date
DK140498B DK140498B (da) 1979-09-17
DK140498C true DK140498C (da) 1980-03-17

Family

ID=26365855

Family Applications (1)

Application Number Title Priority Date Filing Date
DK145373AA DK140498B (da) 1972-03-17 1973-03-16 Analogifremgangsmåde til fremstilling af 3-substituerede 1,2-benzisoxazolderivater.

Country Status (10)

Country Link
US (1) US3948928A (da)
AU (1) AU466970B2 (da)
CA (1) CA1025857A (da)
CH (1) CH577984A5 (da)
DK (1) DK140498B (da)
ES (1) ES412813A1 (da)
FR (1) FR2181831B1 (da)
GB (1) GB1416071A (da)
NL (1) NL168833C (da)
SE (1) SE381047B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
JPS58201770A (ja) * 1982-05-18 1983-11-24 Dainippon Pharmaceut Co Ltd α−置換−1,2−ベンズイソキサゾ−ル−3−酢酸エステル類並びにその酸付加塩類及び第4級アンモニウム塩類
EP1846401B1 (en) * 2005-02-04 2008-06-18 CTG Pharma S.r.l. New 4-aminoquinoline derivatives as antimalarials
DK2559690T3 (da) 2005-05-10 2016-04-25 Incyte Holdings Corp Modulatorer af indolamin-2,3-dioxygenase og fremgangsmåder til anvendelse deraf
CA2634198C (en) 2005-12-20 2014-06-03 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
WO2007081335A1 (en) * 2006-01-12 2007-07-19 Merck & Co., Inc. Therapeutic compounds for treating dyslipidemic conditions
CA2663057C (en) * 2006-09-19 2015-12-08 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
CL2007002650A1 (es) 2006-09-19 2008-02-08 Incyte Corp Compuestos derivados de heterociclo n-hidroxiamino; composicion farmaceutica, util para tratar cancer, infecciones virales y desordenes neurodegenerativos entre otras.
WO2008036652A2 (en) * 2006-09-19 2008-03-27 Incyte Corporation Amidines as modulators of indoleamine 2,3-dioxygenase
WO2008058178A1 (en) * 2006-11-08 2008-05-15 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
JP2010527965A (ja) * 2007-05-24 2010-08-19 ノイロサーチ アクティーゼルスカブ 例えば呼吸器疾患、てんかん及び痙攣の治療のためのカリウムチャネル調節剤としてのベンゾイソオキサゾール誘導体
PE20110308A1 (es) 2008-07-08 2011-06-10 Incyte Corp 1,2,5-oxadiazoles como inhibidores de indolamina 2,3-dioxigenasa
TW202309014A (zh) 2013-11-08 2023-03-01 美商英塞特控股公司 用於合成吲哚胺2,3-雙加氧酶抑制劑之方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670497C3 (de) * 1967-06-06 1973-12-20 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt, Budapest Isochinohnderivate und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
NL168833B (nl) 1981-12-16
SE381047B (sv) 1975-11-24
AU466970B2 (en) 1975-11-13
FR2181831B1 (da) 1975-10-10
DK140498B (da) 1979-09-17
FR2181831A1 (da) 1973-12-07
CA1025857A (en) 1978-02-07
AU5347973A (en) 1974-09-19
NL168833C (nl) 1982-05-17
ES412813A1 (es) 1976-07-01
US3948928A (en) 1976-04-06
NL7303682A (da) 1973-09-19
CH577984A5 (da) 1976-07-30
GB1416071A (en) 1975-12-03

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