DK138536B - Analogifremgangsmåde til fremstilling af 1-naphthalen- eller 4-quinolincarboxamider eller farmaceutisk acceptable syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af 1-naphthalen- eller 4-quinolincarboxamider eller farmaceutisk acceptable syreadditionssalte deraf.

Info

Publication number
DK138536B
DK138536B DK589075AA DK589075A DK138536B DK 138536 B DK138536 B DK 138536B DK 589075A A DK589075A A DK 589075AA DK 589075 A DK589075 A DK 589075A DK 138536 B DK138536 B DK 138536B
Authority
DK
Denmark
Prior art keywords
naphthalene
preparation
pharmaceutically acceptable
acid addition
addition salts
Prior art date
Application number
DK589075AA
Other languages
English (en)
Other versions
DK138536C (da
DK589075A (da
Inventor
Albert Duncan Cale Jr
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of DK589075A publication Critical patent/DK589075A/da
Publication of DK138536B publication Critical patent/DK138536B/da
Application granted granted Critical
Publication of DK138536C publication Critical patent/DK138536C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14—Nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Otolaryngology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
DK589075AA 1974-12-26 1975-12-23 Analogifremgangsmåde til fremstilling af 1-naphthalen- eller 4-quinolincarboxamider eller farmaceutisk acceptable syreadditionssalte deraf. DK138536B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/536,514 US4002757A (en) 1974-12-26 1974-12-26 N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides

Publications (3)

Publication Number Publication Date
DK589075A DK589075A (da) 1976-06-27
DK138536B true DK138536B (da) 1978-09-25
DK138536C DK138536C (da) 1979-03-05

Family

ID=24138812

Family Applications (1)

Application Number Title Priority Date Filing Date
DK589075AA DK138536B (da) 1974-12-26 1975-12-23 Analogifremgangsmåde til fremstilling af 1-naphthalen- eller 4-quinolincarboxamider eller farmaceutisk acceptable syreadditionssalte deraf.

Country Status (18)

Country Link
US (3) US4002757A (da)
JP (2) JPS5191254A (da)
AU (1) AU499075B2 (da)
BE (1) BE836975A (da)
CA (1) CA1071636A (da)
CH (1) CH611603A5 (da)
DE (1) DE2558348A1 (da)
DK (1) DK138536B (da)
ES (1) ES443845A1 (da)
FI (1) FI61480C (da)
FR (1) FR2295744A1 (da)
GB (1) GB1537848A (da)
IE (1) IE43819B1 (da)
NL (1) NL7515084A (da)
NO (1) NO144670C (da)
PH (1) PH13883A (da)
SE (1) SE408417B (da)
ZA (1) ZA757972B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4279822A (en) * 1972-04-03 1981-07-21 A. H. Robins Company, Inc. N-(1-Substituted-3-pyrrolidinyl)benzamides
US4002757A (en) * 1974-12-26 1977-01-11 A. H. Robins Company, Incorporated N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides
US4143150A (en) * 1977-08-19 1979-03-06 A. H. Robins Company, Inc. Derivatives of oxanilic acid
DE3473442D1 (de) * 1983-01-21 1988-09-22 Alkaloida Vegyeszeti Gyar New alkyl diamine derivatives
US5210329A (en) * 1992-02-18 1993-05-11 General Electric Company Process for preparing bisphenol-A
EP1430027B1 (en) 2001-09-14 2010-09-01 High Point Pharmaceuticals, LLC Novel aminoazetidine, -pyrrolidine and -piperidine derivatives
US6673829B2 (en) 2001-09-14 2004-01-06 Novo Nordisk A/S Aminoazetidine,-pyrrolidine and -piperidine derivatives
ES2305776T3 (es) * 2003-06-17 2008-11-01 Pfizer Inc. Derivados de n-pirrolidin-3-il-amida como inhibidores de la re-captacion de serotonina y noradrenalina.
US7348434B2 (en) * 2003-08-08 2008-03-25 Antony Bigot 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
CA2590226A1 (en) * 2004-12-14 2006-06-22 Pfizer Limited N-pyrrolidin-3yl-amide derivatives as serotonin and noradrenalin re-uptake inhibitors
US20090239928A1 (en) * 2004-12-14 2009-09-24 Paul Vincent Fish N-Pyrrolidin-3YL-Amide Derivatives As Serotonin and Noradrenalin Re-Uptake Inhibitors
EP1828122A2 (en) * 2004-12-16 2007-09-05 Pfizer Limited N-pyrrolidin-3-yl-amide derivatives as serotonin and noradrenalin re-uptake inhibitors
KR20090130347A (ko) * 2007-05-09 2009-12-22 화이자 인코포레이티드 치환된 헤테로사이클릭 유도체 및 조성물 및 항균제로서의 이의 약학적 용도

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1825623A (en) * 1931-09-29 Oonhohachzn
DE67123C (de) * L. THOMAS in Montegnee-les-Siege, Belgien Handdrehbohrmaschine für Gruben und Steinbrüche
US3133061A (en) * 1962-11-13 1964-05-12 Sterling Drug Inc Piperidine carboxamides and derivatives thereof
US3342826A (en) * 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
US3577440A (en) * 1968-12-23 1971-05-04 Robins Co Inc A H 1-substituted-3-amido-pyrrolidines
GB1364231A (en) * 1968-12-23 1974-08-21 Robins Co Inc A H N-/1-substituted-3-pyrrolidinyl/benzamides and thiobenzamides
US3829434A (en) * 1972-11-10 1974-08-13 Pfizer Piperidinesulfonylurea derivatives
US4002757A (en) * 1974-12-26 1977-01-11 A. H. Robins Company, Incorporated N-(1-substituted-3-pyrrolidinyl)-4-quinolinecarboxamides

Also Published As

Publication number Publication date
CA1071636A (en) 1980-02-12
ES443845A1 (es) 1977-04-16
NO754376L (da) 1976-06-29
US4087428A (en) 1978-05-02
PH13883A (en) 1980-10-27
IE43819L (en) 1976-06-26
AU499075B2 (en) 1979-04-05
NL7515084A (nl) 1976-06-29
JPS5191254A (en) 1976-08-10
DK138536C (da) 1979-03-05
FR2295744A1 (fr) 1976-07-23
US4073796A (en) 1978-02-14
DK589075A (da) 1976-06-27
IE43819B1 (en) 1981-06-03
AU8755075A (en) 1977-06-23
SE408417B (sv) 1979-06-11
JPS611426B2 (da) 1986-01-17
SE7514374L (sv) 1976-06-28
FI61480C (fi) 1982-08-10
US4002757A (en) 1977-01-11
JPS619314B2 (da) 1986-03-22
JPS60248684A (ja) 1985-12-09
DE2558348A1 (de) 1976-07-08
FI753606A (da) 1976-06-27
FI61480B (fi) 1982-04-30
GB1537848A (en) 1979-01-04
NO144670C (no) 1981-10-14
CH611603A5 (da) 1979-06-15
ZA757972B (en) 1976-12-29
FR2295744B1 (da) 1978-07-28
BE836975A (fr) 1976-04-16
NO144670B (no) 1981-07-06

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