DK131567B - Analogifremgangsmåde til fremstilling af 3H-1,4-benzodiazepiner eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af 3H-1,4-benzodiazepiner eller syreadditionssalte deraf.

Info

Publication number
DK131567B
DK131567B DK100670AA DK100670A DK131567B DK 131567 B DK131567 B DK 131567B DK 100670A A DK100670A A DK 100670AA DK 100670 A DK100670 A DK 100670A DK 131567 B DK131567 B DK 131567B
Authority
DK
Denmark
Prior art keywords
benzodiazepines
preparation
acid addition
addition salts
analogous process
Prior art date
Application number
DK100670AA
Other languages
English (en)
Other versions
DK131567C (da
Inventor
J B Hester Jr
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of DK131567B publication Critical patent/DK131567B/da
Application granted granted Critical
Publication of DK131567C publication Critical patent/DK131567C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Fodder In General (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
DK100670A 1969-02-28 1970-02-27 Analogifremgangsmade til fremstilling af 3h-1,4-benzodiazepiner eller syreadditionssalte deraf DK131567C (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US80345069A 1969-02-28 1969-02-28

Publications (2)

Publication Number Publication Date
DK131567B true DK131567B (da) 1975-08-04
DK131567C DK131567C (da) 1976-03-01

Family

ID=25186534

Family Applications (1)

Application Number Title Priority Date Filing Date
DK100670A DK131567C (da) 1969-02-28 1970-02-27 Analogifremgangsmade til fremstilling af 3h-1,4-benzodiazepiner eller syreadditionssalte deraf

Country Status (12)

Country Link
JP (1) JPS4810799B1 (da)
BE (1) BE746664A (da)
BR (1) BR6915069D0 (da)
CH (1) CH535773A (da)
DE (1) DE2005176A1 (da)
DK (1) DK131567C (da)
ES (1) ES376688A1 (da)
FR (1) FR2034577B1 (da)
GB (1) GB1243953A (da)
IL (1) IL33735A (da)
NL (1) NL7002712A (da)
SE (1) SE367631B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3649617A (en) * 1970-07-20 1972-03-14 Upjohn Co 2-substituted amino-5-phenyl-3h-1 4-benzodiazepines
US7160880B1 (en) 1999-05-14 2007-01-09 Cenes Limited Short-acting benzodiazepines
GB9911152D0 (en) * 1999-05-14 1999-07-14 Glaxo Group Ltd Short-acting benzodiazepines
KR20150081370A (ko) 2006-07-10 2015-07-13 파이온 유케이 리미티드 속효형 벤조디아제핀 염 및 이의 중합체 형태
EP2450039A1 (en) 2010-11-08 2012-05-09 PAION UK Ltd. Dosing regimen for sedation with CNS 7056 (Remimazolam)
AR094963A1 (es) 2013-03-04 2015-09-09 Ono Pharmaceutical Co Reacción de oxidación excelente en el índice de conversión

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB956592A (en) * 1960-04-20 1964-04-29 Smith Kline French Lab Improvements in or relating to trifluoromethyl-1,4-benzodiazepine derivatives

Also Published As

Publication number Publication date
FR2034577A1 (da) 1970-12-11
BR6915069D0 (pt) 1973-08-16
DE2005176A1 (de) 1970-09-10
BE746664A (fr) 1970-08-27
FR2034577B1 (da) 1973-07-13
GB1243953A (en) 1971-08-25
JPS4810799B1 (da) 1973-04-07
DK131567C (da) 1976-03-01
IL33735A (en) 1972-12-29
SE367631B (da) 1974-06-04
ES376688A1 (es) 1972-05-01
IL33735A0 (en) 1970-03-22
CH535773A (de) 1973-04-15
NL7002712A (da) 1970-09-01

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