DK123718B - Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller salte deraf. - Google Patents

Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller salte deraf.

Info

Publication number
DK123718B
DK123718B DK384669AA DK384669A DK123718B DK 123718 B DK123718 B DK 123718B DK 384669A A DK384669A A DK 384669AA DK 384669 A DK384669 A DK 384669A DK 123718 B DK123718 B DK 123718B
Authority
DK
Denmark
Prior art keywords
salts
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
DK384669AA
Other languages
English (en)
Inventor
Y Usui
Y Hara
T Masuda
T Komatsu
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of DK123718B publication Critical patent/DK123718B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/30Preparation including building-up the benzodiazepine skeleton from compounds already containing hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DK384669AA 1968-07-17 1969-07-16 Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller salte deraf. DK123718B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP5030668 1968-07-17

Publications (1)

Publication Number Publication Date
DK123718B true DK123718B (da) 1972-07-24

Family

ID=12855196

Family Applications (1)

Application Number Title Priority Date Filing Date
DK384669AA DK123718B (da) 1968-07-17 1969-07-16 Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller salte deraf.

Country Status (10)

Country Link
US (1) US3644339A (da)
CH (1) CH517104A (da)
DE (1) DE1931870C3 (da)
DK (1) DK123718B (da)
ES (1) ES369319A1 (da)
FR (1) FR2013094A1 (da)
GB (1) GB1284122A (da)
NL (1) NL144933B (da)
NO (1) NO124033B (da)
SE (1) SE348200B (da)

Also Published As

Publication number Publication date
NL6910938A (da) 1970-01-20
ES369319A1 (es) 1971-06-01
FR2013094A1 (da) 1970-03-27
CH517104A (de) 1971-12-31
US3644339A (en) 1972-02-22
DE1931870B2 (de) 1980-01-10
DE1931870A1 (de) 1970-01-22
GB1284122A (en) 1972-08-02
DE1931870C3 (de) 1980-09-18
NL144933B (nl) 1975-02-17
SE348200B (da) 1972-08-28
NO124033B (da) 1972-02-21

Similar Documents

Publication Publication Date Title
DK134113B (da) Analogifremgangsmåde til fremstilling af 1,2,3,4-tetrahydro-7-halogen-eller 7-trifluormethyl-6-sulfamyl-4-quinazolinoner eller salte heraf.
DK132172B (da) Analogifremgangsmåde til fremstilling af 6,7-benzomorphaner eller salte deraf.
DK128078B (da) Analogifremgangsmåde til fremstilling af 1,2,3,4-tetrahydroisoquinolinderivater eller salte deraf.
DK135534B (da) Fremgangsmåde til fremstilling af pyrasol-(3,4-d)-pyrimidiner eller salte heraf.
DK120548B (da) Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller 4-oxider eller syreadditionssalte deraf.
DK138797B (da) Analogifremgangsmåde til fremstilling af 1,4-benzodiazepin-derivater eller N-oxider eller salte deraf.
DK125025B (da) Analogifremgangsmåde til fremstilling af 2,1,3-benzothiadiazol-forbindelser eller salte deraf.
DK131374B (da) Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller salte deraf.
DK137754B (da) Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater.
DK118509B (da) Fremgangsmåde til fremstilling af 1,1-diphenyl-1-metoxy-3-benzylaminopropan eller salte heraf.
DK126201B (da) Analogifremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller salte deraf.
DK124035B (da) Fremgangsmåde til fremstilling af α-carboxybenzylpencillin eller salte deraf.
DK120796B (da) Analogifremgangsmåde til fremstilling af 1,2-oxazinderivater eller salte deraf.
DK137237B (da) Analogifremgangsmåde til fremstilling af 1,4-benzodiazepinforbindelser eller 4-N-oxider eller salte heraf.
DK122725B (da) Analogifremgangsmåde til fremstilling af 10,11-dihydro-5H-dibenz(b,f)azepineddikesyrederivater eller salte deraf.
DK124885B (da) Analogifremgangsmåde til fremstilling af 4-alkenyl-substituerede 1,2-difenyl-3,5-dioxopyrazolidiner eller salte heraf.
DK124545B (da) Analogifremgangsmåde til fremstilling af bisimidazolyl-bisphenylmethaner eller salte deraf.
DK123718B (da) Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller salte deraf.
DK127473B (da) Fremgangsmåde til fremstilling af 2,5- eller 3,4-dihydroxyarylsulfoniumsalte.
DK127115B (da) Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater.
DK108974C (da) Fremgangsmåde til fremstilling af azepinderivater eller salte deraf.
DK124030B (da) Analogifremgangsmåde til fremstilling af 2,4-dialkanoylamino-6-amino-quinazoliner eller salte deraf.
DK136364B (da) Analogifremgangsmåde til fremstilling af 4(5)-trifluormethylimidazolderivater eller salte deraf.
DK125646B (da) Fremgangsmåde til fremstilling af 1,1'-disubstitueret-4,4'-bipyridyliumsalte eller 1,1'-disubstitueret-2,2'-bipyridyliumsalte.
DK123599B (da) Fremgangsmåde til fremstilling af (-)-norscopolamin eller salte deraf.