DK122393B - Analogifremgangsmåde til fremstilling af phenylthiazolyl-α-alkylmalonsyrederivater. - Google Patents

Analogifremgangsmåde til fremstilling af phenylthiazolyl-α-alkylmalonsyrederivater.

Info

Publication number
DK122393B
DK122393B DK498970AA DK498970A DK122393B DK 122393 B DK122393 B DK 122393B DK 498970A A DK498970A A DK 498970AA DK 498970 A DK498970 A DK 498970A DK 122393 B DK122393 B DK 122393B
Authority
DK
Denmark
Prior art keywords
phenylthiazolyl
preparation
acid derivatives
analogous process
alkylmalonic acid
Prior art date
Application number
DK498970AA
Other languages
English (en)
Inventor
G Stacey
W Hepworth
Original Assignee
Ici Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Ltd filed Critical Ici Ltd
Publication of DK122393B publication Critical patent/DK122393B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/12Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/30Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F1/00Compounds containing elements of Groups 1 or 11 of the Periodic Table

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
DK498970AA 1968-03-22 1970-09-30 Analogifremgangsmåde til fremstilling af phenylthiazolyl-α-alkylmalonsyrederivater. DK122393B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB03989/68A GB1192701A (en) 1968-03-22 1968-03-22 Novel Thiazole Derivatives, the preparation thereof and Compositions containing the same

Publications (1)

Publication Number Publication Date
DK122393B true DK122393B (da) 1972-02-28

Family

ID=10033003

Family Applications (3)

Application Number Title Priority Date Filing Date
DK157569AA DK125251B (da) 1968-03-22 1969-03-21 Analogifremgangsmåde til fremstilling af thiazolylmalonsyrederivater.
DK498870AA DK125326B (da) 1968-03-22 1970-09-30 Analogifremgangsmåde til fremstilling af phenylthiazol-2-ylmalonsyrederivater.
DK498970AA DK122393B (da) 1968-03-22 1970-09-30 Analogifremgangsmåde til fremstilling af phenylthiazolyl-α-alkylmalonsyrederivater.

Family Applications Before (2)

Application Number Title Priority Date Filing Date
DK157569AA DK125251B (da) 1968-03-22 1969-03-21 Analogifremgangsmåde til fremstilling af thiazolylmalonsyrederivater.
DK498870AA DK125326B (da) 1968-03-22 1970-09-30 Analogifremgangsmåde til fremstilling af phenylthiazol-2-ylmalonsyrederivater.

Country Status (15)

Country Link
US (1) US3661920A (da)
AT (1) AT284841B (da)
BE (1) BE730284A (da)
BR (1) BR6807374D0 (da)
CA (1) CA948199A (da)
CH (2) CH513907A (da)
CS (3) CS154268B2 (da)
DE (1) DE1913472A1 (da)
DK (3) DK125251B (da)
ES (1) ES365089A1 (da)
FR (1) FR2004544A1 (da)
GB (1) GB1192701A (da)
IE (1) IE32967B1 (da)
IL (1) IL31679A (da)
NL (1) NL6903963A (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2703542C2 (de) * 1977-01-26 1985-09-26 Schering AG, 1000 Berlin und 4709 Bergkamen Thiazolylzimtsäurenitrile, Insektenbekämpfungsmittel enthaltend diese Verbindungen sowie Verfahren zu ihrer Herstellung
US4197306A (en) * 1977-06-30 1980-04-08 Uniroyal, Inc. Aryl-substituted thiazoles
US4153703A (en) * 1977-06-30 1979-05-08 Uniroyal, Inc. Method of controlling insects and acarids with certain aryl-substituted thiazoles
DE2801794A1 (de) 1978-01-17 1979-07-19 Basf Ag Verfahren zur herstellung von thiazolderivaten und neue thiazole
DE2920183A1 (de) * 1979-05-17 1981-04-30 Schering Ag Berlin Und Bergkamen, 1000 Berlin Thiazolyliden-oxo-propionitrile, insektizide mittel enthaltend diese verbindungen sowie verfahren zu ihrer herstellung
US4346094A (en) * 1980-09-22 1982-08-24 Eli Lilly And Company 3-Aryl-5-isothiazolecarboxylic acids and related compounds used to lower uric acid levels
US5077305A (en) * 1990-02-13 1991-12-31 Bristol-Myers Squibb Co. Thiazole carboxylic acids and esters
EP0442448A3 (en) 1990-02-13 1992-08-12 Bristol-Myers Squibb Company Heterocyclic carboxylic acids and esters
DE10331675A1 (de) * 2003-07-14 2005-02-10 Bayer Cropscience Ag Hetarylsubstituierte Pyrazolidindion-Derivate
EP2200649A4 (en) * 2007-10-19 2012-09-26 Univ California COMPOSITIONS AND METHODS FOR TREATING CNS INFUSION, PSYCHOSIS, DELIRE, PTSD OR PTSS

Also Published As

Publication number Publication date
GB1192701A (en) 1970-05-20
CA948199A (en) 1974-05-28
US3661920A (en) 1972-05-09
NL6903963A (da) 1969-09-24
CS154268B2 (da) 1974-03-29
CH513907A (de) 1971-10-15
IL31679A (en) 1972-08-30
AT284841B (de) 1970-09-25
FR2004544A1 (da) 1969-11-28
CH553209A (de) 1974-08-30
CS154266B2 (da) 1974-03-29
ES365089A1 (es) 1971-01-01
DE1913472A1 (de) 1969-11-06
CS154267B2 (da) 1974-03-29
BE730284A (da) 1969-09-22
DK125251B (da) 1973-01-22
IE32967L (en) 1969-09-22
DK125326B (da) 1973-02-05
BR6807374D0 (pt) 1973-02-08
IE32967B1 (en) 1974-02-06

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