DK120600B - Fremgangsmåde til fremstilling af 5-aryl-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf. - Google Patents

Fremgangsmåde til fremstilling af 5-aryl-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf.

Info

Publication number
DK120600B
DK120600B DK346164AA DK346164A DK120600B DK 120600 B DK120600 B DK 120600B DK 346164A A DK346164A A DK 346164AA DK 346164 A DK346164 A DK 346164A DK 120600 B DK120600 B DK 120600B
Authority
DK
Denmark
Prior art keywords
benzodiazepin
aryl
ones
preparation
acid addition
Prior art date
Application number
DK346164AA
Other languages
Danish (da)
English (en)
Inventor
R Fryer
L Sternbach
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK120600B publication Critical patent/DK120600B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK346164AA 1963-07-10 1964-07-10 Fremgangsmåde til fremstilling af 5-aryl-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf. DK120600B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US294142A US3247187A (en) 1963-07-10 1963-07-10 Oxidation of 1, 4-benzodiazepines to 1, 4-benzodiazepin-2-ones

Publications (1)

Publication Number Publication Date
DK120600B true DK120600B (da) 1971-06-21

Family

ID=23132071

Family Applications (1)

Application Number Title Priority Date Filing Date
DK346164AA DK120600B (da) 1963-07-10 1964-07-10 Fremgangsmåde til fremstilling af 5-aryl-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf.

Country Status (11)

Country Link
US (1) US3247187A (pt)
BE (1) BE650261A (pt)
BR (1) BR6460685D0 (pt)
CH (1) CH458371A (pt)
DE (1) DE1445901A1 (pt)
DK (1) DK120600B (pt)
ES (1) ES301865A1 (pt)
GB (1) GB1036577A (pt)
NL (1) NL6407796A (pt)
NO (1) NO117639B (pt)
OA (1) OA00949A (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3361742A (en) * 1964-12-07 1968-01-02 Hoffmann La Roche 5-oxo-1h-pyrrolo-[2, 1-c][1, 4]-benzodiazepin-2-crylamides
US3405123A (en) * 1965-02-08 1968-10-08 Hoffmann La Roche Process for preparing 1, 4-benzodiazepin-2-ones

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3176009A (en) * 1965-03-30 Hydrolysis of l-acylated-j-acyloxy benzodiazepines
US3121076A (en) * 1964-02-11 Benzodiazepinones and processes

Also Published As

Publication number Publication date
NL6407796A (pt) 1965-01-11
US3247187A (en) 1966-04-19
CH458371A (de) 1968-06-30
GB1036577A (en) 1966-07-20
BE650261A (pt) 1965-01-08
ES301865A1 (es) 1965-02-01
NO117639B (pt) 1969-09-08
OA00949A (fr) 1968-03-22
BR6460685D0 (pt) 1973-07-19
DE1445901A1 (de) 1969-02-06

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