DK104677A - Fremgangsmade til fremstilling af hidtil ukendte 2,3-dihydro-imidazo (2,1-b)-thiazolderivater - Google Patents

Fremgangsmade til fremstilling af hidtil ukendte 2,3-dihydro-imidazo (2,1-b)-thiazolderivater

Info

Publication number: DK104677A
Authority: DK; Denmark
Prior art keywords: imidazo; dihydro; procedure; preparation; thiazole derivatives
Prior art date: 1976-03-10

Application number

DK104677A

Other languages

English (en)

Other versions

DK144702C (da

DK144702B (da

Inventor

J L E Baetz

Original Assignee

Metabio

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-03-10

Filing date

1977-03-09

Publication date

1977-09-11

1977-03-09 Application filed by Metabio filed Critical Metabio

1977-09-11 Publication of DK104677A publication Critical patent/DK104677A/da

1982-05-17 Publication of DK144702B publication Critical patent/DK144702B/da

1982-10-11 Application granted granted Critical

1982-10-11 Publication of DK144702C publication Critical patent/DK144702C/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pain & Pain Management (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK104677A 1976-03-10 1977-03-09 Analogifremgangsmaade til fremstilling af 2,3-dihydro-imidazo(2,1-b)-thiazolderivater DK144702C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB951776		1976-03-10
GB9517/76A GB1541321A (en)	1976-03-10	1976-03-10	2,3-dihydroimidazo(2,1-b)thiazole derivatives and process for their preparation

Publications (3)

Publication Number	Publication Date
DK104677A true DK104677A (da)	1977-09-11
DK144702B DK144702B (da)	1982-05-17
DK144702C DK144702C (da)	1982-10-11

Family

ID=9873507

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK104677A DK144702C (da)	1976-03-10	1977-03-09	Analogifremgangsmaade til fremstilling af 2,3-dihydro-imidazo(2,1-b)-thiazolderivater

Country Status (28)

Country	Link
US (1)	US4110460A (da)
JP (1)	JPS5927357B2 (da)
AT (1)	AT352716B (da)
AU (1)	AU503912B2 (da)
BE (1)	BE852259A (da)
BG (1)	BG28262A3 (da)
CA (1)	CA1074324A (da)
CH (1)	CH598267A5 (da)
CS (1)	CS190341B2 (da)
DE (1)	DE2709639A1 (da)
DK (1)	DK144702C (da)
ES (1)	ES456575A1 (da)
FI (1)	FI62313C (da)
FR (1)	FR2343748A1 (da)
GB (1)	GB1541321A (da)
HU (1)	HU172685B (da)
IE (1)	IE44280B1 (da)
IL (1)	IL51581A (da)
LU (1)	LU76879A1 (da)
NL (1)	NL7702446A (da)
NO (1)	NO150884C (da)
PL (1)	PL102603B1 (da)
PT (1)	PT66278B (da)
RO (1)	RO71301A (da)
SE (1)	SE431653B (da)
SU (1)	SU629882A3 (da)
YU (1)	YU61977A (da)
ZA (1)	ZA771303B (da)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4204067A (en) *	1976-09-24	1980-05-20	Adhikary Parimal K	Derivatives of imidazo[2,1-b] thiazole
US4263311A (en) *	1976-09-27	1981-04-21	Smithkline Corporation	5,6-Phenyl-2,3-dihydroimidazo [2,1-b] thiazoles
LU77703A1 (de) *	1977-07-07	1979-03-26	Ciba Geigy Ag	Verfahren zur herstellung von bicyclischen thia-diaza-verbindungen
US4153706A (en)	1978-02-13	1979-05-08	Smithkline Corporation	6-Hydroxy-5,6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazoles
US4175127A (en) *	1978-09-27	1979-11-20	Smithkline Corporation	Pyridyl substituted 2,3-dihydroimidazo[2,1-b]thiazoles
PL221188A1 (da) *	1979-01-05	1980-12-01	Ciba Geigy Ag
US4364942A (en) *	1979-06-21	1982-12-21	Janssen Pharmaceutica N.V.	2,3-Dihydro-imidazo (2,1-b)benzothiazoles compositions useful as anti-parkinsonism agents
FR2463774A1 (fr) *	1979-08-21	1981-02-27	Yamanouchi Pharma Co Ltd	Derives du 2-phenylimidazo(2,1-b)benzothiazole
FR2479831A1 (fr) *	1980-04-08	1981-10-09	Synthelabo	Derives de thiazole, leur preparation et leur application en therapeutique
US4327221A (en) *	1980-10-15	1982-04-27	American Home Products Corporation	2-Substituted-3-hydroxythiazolo(2,3-8)-thiazolium salts and mesoionic didehydro derivatives thereof
US5134150A (en) *	1985-12-12	1992-07-28	Smithkline Beecham Corporation	Inhibition of the 5-lipoxygenase pathway
US5002941A (en) *	1985-12-12	1991-03-26	Smithkline Beecham Corporation	Pyrrolo(1,2-a)imidazole and imidazo(1,2-a)pyridine derivatives and their use as 5-lipoxygenase pathway inhibitors
US4719218A (en) *	1985-12-12	1988-01-12	Smithkline Beckman Corporation	Pyrrolo[1,2-a]imidazole and pyrrolo[1,2-a]pyridine derivatives and their use as 5-lipoxygenase pathway inhibitor
US4751310A (en) *	1985-12-12	1988-06-14	Smithkline Beckman Corporation	Inhibition of the 5-lipoxygenase pathway
ZW24186A1 (en) *	1985-12-12	1987-07-08	Smithkline Beckman Corp	Inhibition of the 5-lipoxygenase pathway
US5145858A (en) *	1985-12-12	1992-09-08	Smithkline Beecham Corp.	Pyrrolo [1,2-a] imidazole and imidazo [1,2a] pyridine derivatives and their use as 5-lipoxygenase pathway inhibitors
US4794114A (en) *	1986-08-19	1988-12-27	Smithkline Beckman Corporation	Inhibition of interleukin-1 production by monocytes and/or macrophages
US5630014A (en) *	1993-10-27	1997-05-13	Nec Corporation	Gain controller with automatic adjustment using integration energy values
US6127387A (en) *	1996-12-10	2000-10-03	Thomas Jefferson University	Use of CD4-binding small molecules to inhibit immune responses
WO2007034282A2 (en) *	2005-09-19	2007-03-29	Pfizer Products Inc.	Diaryl-imidazole compounds condensed with a heterocycle as c3a receptor antagonists

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL131034C (da) *	1964-05-11
US3455924A (en) *	1967-02-08	1969-07-15	Upjohn Co	Dianisylimidazoles
NL164285C (nl) *	1968-01-09	1980-12-15	Rhone Poulenc Sa	Werkwijze ter bereiding van een farmaceutisch preparaat, dat een imidazoÿ2.1-bÿthiazoolderivaat bevat, de gevormde farmaceutische preparaten, alsmede werkwijze voor het bereiden van dit imidazoÿ2.1-bÿthiazoolderivaat.

1976
- 1976-03-10 GB GB9517/76A patent/GB1541321A/en not_active Expired
1977
- 1977-03-02 IL IL51581A patent/IL51581A/xx unknown
- 1977-03-02 CH CH259777A patent/CH598267A5/xx not_active IP Right Cessation
- 1977-03-02 LU LU76879A patent/LU76879A1/xx unknown
- 1977-03-03 IE IE467/77A patent/IE44280B1/en unknown
- 1977-03-04 US US05/774,497 patent/US4110460A/en not_active Expired - Lifetime
- 1977-03-04 CA CA273,239A patent/CA1074324A/en not_active Expired
- 1977-03-04 FR FR7706434A patent/FR2343748A1/fr active Granted
- 1977-03-04 ZA ZA00771303A patent/ZA771303B/xx unknown
- 1977-03-05 DE DE19772709639 patent/DE2709639A1/de not_active Withdrawn
- 1977-03-07 ES ES456575A patent/ES456575A1/es not_active Expired
- 1977-03-07 NL NL7702446A patent/NL7702446A/xx not_active Application Discontinuation
- 1977-03-07 SE SE7702503A patent/SE431653B/xx unknown
- 1977-03-08 BG BG7735610A patent/BG28262A3/xx unknown
- 1977-03-08 YU YU00619/77A patent/YU61977A/xx unknown
- 1977-03-08 PT PT66278A patent/PT66278B/pt unknown
- 1977-03-09 RO RO7789635A patent/RO71301A/ro unknown
- 1977-03-09 HU HU77ME00002049A patent/HU172685B/hu unknown
- 1977-03-09 NO NO770841A patent/NO150884C/no unknown
- 1977-03-09 CS CS771589A patent/CS190341B2/cs unknown
- 1977-03-09 DK DK104677A patent/DK144702C/da not_active IP Right Cessation
- 1977-03-09 BE BE175621A patent/BE852259A/xx not_active IP Right Cessation
- 1977-03-09 PL PL1977196539A patent/PL102603B1/pl unknown
- 1977-03-09 FI FI770759A patent/FI62313C/fi not_active IP Right Cessation
- 1977-03-10 AU AU23156/77A patent/AU503912B2/en not_active Expired
- 1977-03-10 JP JP52026581A patent/JPS5927357B2/ja not_active Expired
- 1977-03-10 SU SU772459651A patent/SU629882A3/ru active
- 1977-03-10 AT AT164477A patent/AT352716B/de not_active IP Right Cessation

Also Published As

Publication number	Publication date
SE431653B (sv)	1984-02-20
ES456575A1 (es)	1978-02-16
PL102603B1 (pl)	1979-04-30
BE852259A (fr)	1977-09-09
FR2343748A1 (fr)	1977-10-07
NO770841L (no)	1977-09-13
JPS5927357B2 (ja)	1984-07-05
DE2709639A1 (de)	1977-09-15
NO150884B (no)	1984-09-24
PT66278B (fr)	1978-08-08
ATA164477A (de)	1979-03-15
SU629882A3 (ru)	1978-10-25
IL51581A0 (en)	1977-05-31
AU503912B2 (en)	1979-09-27
FI770759A (da)	1977-09-11
AU2315677A (en)	1978-09-14
LU76879A1 (da)	1977-07-12
FI62313B (fi)	1982-08-31
FI62313C (fi)	1982-12-10
CA1074324A (en)	1980-03-25
HU172685B (hu)	1978-11-28
GB1541321A (en)	1979-02-28
CH598267A5 (da)	1978-04-28
BG28262A3 (en)	1980-03-25
NO150884C (no)	1985-01-09
YU61977A (en)	1982-06-30
US4110460A (en)	1978-08-29
ZA771303B (en)	1978-01-25
FR2343748B1 (da)	1980-07-18
CS190341B2 (en)	1979-05-31
DK144702C (da)	1982-10-11
IL51581A (en)	1980-02-29
NL7702446A (nl)	1977-09-13
IE44280B1 (en)	1981-09-23
SE7702503L (sv)	1977-09-11
IE44280L (en)	1977-09-10
AT352716B (de)	1979-10-10
RO71301A (ro)	1981-11-24
JPS52136195A (en)	1977-11-14
DK144702B (da)	1982-05-17
PT66278A (fr)	1977-04-01

Legal Events

Date	Code	Title	Description
1985-11-11	PBP	Patent lapsed

Publication	Publication Date	Title
DK142372C (da)	1981-03-23	Fremgangsmaade til fremstilling af androstan-17-on-derivater
DK104677A (da)	1977-09-11	Fremgangsmade til fremstilling af hidtil ukendte 2,3-dihydro-imidazo (2,1-b)-thiazolderivater
DK177679A (da)	1979-12-03	Fremgangsmaade til fremstilling af hidtil ukendte aminothiazoler
DK258078A (da)	1979-01-23	Fremgangsmaade til fremstilling af 7alfa-methoxy-7beta-(1,3-dithiethan-2-carboxamido) cephalosporansyre-derivater
DK118277A (da)	1977-09-30	Fremgangsmade til fremstilling af n-5-tetrazololyl)-4-oxo-4h-pyrimido (2,1-b)benzothiazol-3-carboxamider
DK387177A (da)	1978-03-02	Fremgangsmaade til fremstilling af derivater af perhydro-aza-heterocycler
NO151365C (no)	1985-03-27	Fremgangsmaate for fremstilling av 4-halogen-dihydropyran-derivater.
DK271977A (da)	1977-12-22	Fremgangsmade til fremstilling af dispeptidderivater
DK273776A (da)	1976-12-22	Fremgangsmade til fremstilling af 2,4-dioxo-1,2,3,4-tetrahydro-s-triazino-(1,2-a)-benzimidazoler
DK118177A (da)	1977-09-18	Fremgangsmade til fremstilling af isobutyramidderivater
DK46577A (da)	1977-08-13	Fremgangsmade til fremstilling af tetrahydroechinocandinderivater
DK165677A (da)	1977-10-16	Fremgangsmade til fremstilling af thiourinstofderivater
DK154970C (da)	1989-06-12	Analogifremgangsmaade til fremstilling af carbostyrilderivater
DK364677A (da)	1978-02-17	Fremgangsmaade til fremstilling af antibiotiske midler
DK528777A (da)	1978-05-31	Fremgangsmaade til fremstilling af cephalosporinderivater
DK127976A (da)	1976-09-25	Fremgangsmade til fremstilling af thiazolinonderivater
DK538777A (da)	1978-06-04	Fremgangsmaade til fremstilling af isoxazolderivater
DK211277A (da)	1977-11-15	Fremgangsmade til fremstilling af isothiourinstofderivater
DK264377A (da)	1978-01-02	Fremgangsmade til fremstilling af 1alfa-hydroxycholesterol-derivater
DK579876A (da)	1977-07-13	Fremgangsmade til fremstilling af 2-methyl-4-hydroxy-1,2-benzothiazin-3-carboxamid-1,1-dioxid
DK129277A (da)	1977-09-25	Fremgangsmade til fremstilling af dibenzothiophenderivater
DK88277A (da)	1977-09-03	Fremgangsmade til fremstilling af halogenderivater af 16alfamethylpregnanrekken
DK351377A (da)	1978-02-07	Fremgangsmade til fremstilling af triazolbenzazepinderivater
DK337977A (da)	1978-02-05	Fremgangsmade til fremstilling af furanderivater
AR215629A1 (es)	1979-10-31	Procedimiento para la preparacion de derivados 6-halonicotinoilicos de 6-(m-aminofenil)-2,3,5,6-tetrahidroimidazo(2,1-b)tiazol(m-aminotetramisol)