DK0605474T3 - Carbamatanaloger af thiaphysovenin, farmaceutiske præparater og fremgangsmåder til inhibering af cholinesteraser - Google Patents
Carbamatanaloger af thiaphysovenin, farmaceutiske præparater og fremgangsmåder til inhibering af cholinesteraserInfo
- Publication number
- DK0605474T3 DK0605474T3 DK92919058T DK92919058T DK0605474T3 DK 0605474 T3 DK0605474 T3 DK 0605474T3 DK 92919058 T DK92919058 T DK 92919058T DK 92919058 T DK92919058 T DK 92919058T DK 0605474 T3 DK0605474 T3 DK 0605474T3
- Authority
- DK
- Denmark
- Prior art keywords
- thiaphysovenin
- methods
- pharmaceutical preparations
- compounds
- cholinesterases
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Ophthalmology & Optometry (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Enzymes And Modification Thereof (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US76576691A | 1991-09-26 | 1991-09-26 | |
US84508192A | 1992-03-03 | 1992-03-03 | |
PCT/US1992/007085 WO1993005779A1 (en) | 1991-09-26 | 1992-08-26 | Carbamate analogs of thiaphysovenine, pharmaceutical compositions, and method for inhibiting cholinesterases |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0605474T3 true DK0605474T3 (da) | 2004-02-23 |
Family
ID=27117648
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK92919058T DK0605474T3 (da) | 1991-09-26 | 1992-08-26 | Carbamatanaloger af thiaphysovenin, farmaceutiske præparater og fremgangsmåder til inhibering af cholinesteraser |
Country Status (10)
Country | Link |
---|---|
US (1) | US5378723A (da) |
EP (2) | EP0605474B1 (da) |
JP (1) | JP3193717B2 (da) |
AT (1) | ATE254916T1 (da) |
AU (1) | AU667318B2 (da) |
CA (1) | CA2119782C (da) |
DE (1) | DE69233255T2 (da) |
DK (1) | DK0605474T3 (da) |
ES (1) | ES2206449T3 (da) |
WO (1) | WO1993005779A1 (da) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE311876T1 (de) * | 1997-07-09 | 2005-12-15 | Axonyx | Hochselektive butyrylcholinesterase inhibitoren zur behandlung und zur diagnose von demenz und alzheimers krankheit |
US6534541B1 (en) | 1999-10-19 | 2003-03-18 | Novartis Ag | Treatment of ocular disorders |
US7153882B2 (en) * | 2000-11-02 | 2006-12-26 | The United States Of America As Represented By The Department Of Health And Human Services | Agents useful for reducing amyloid precursor protein and treating demantia and methods of use thereof |
EP1554572B1 (en) | 2001-07-25 | 2009-10-14 | Raptor Pharmaceutical Inc. | Compositions and methods for modulating blood-brain barrier transport |
EP1718294A4 (en) * | 2004-01-30 | 2007-10-03 | Axonyx Inc | METHODS OF TREATING COMPLICATIONS OF DIABETES |
AU2006239221C1 (en) | 2005-04-28 | 2012-08-16 | Otsuka Pharmaceutical Co., Ltd. | Pharma-informatics system |
WO2008036682A2 (en) | 2006-09-18 | 2008-03-27 | Raptor Pharmaceutical Inc. | Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates |
ES2728225T3 (es) | 2009-02-20 | 2019-10-23 | 2 Bbb Medicines B V | Sistema de administración de fármacos a base de glutatión |
KR101741629B1 (ko) | 2009-05-06 | 2017-05-31 | 라보라토리 스킨 케어, 인크. | 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법 |
US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
KR101667215B1 (ko) | 2014-10-21 | 2016-10-18 | 한밭대학교 산학협력단 | 신규한 트립타민 컨쥬게이트 화합물 및 그의 용도 |
KR102233120B1 (ko) | 2018-12-18 | 2021-03-29 | 한밭대학교 산학협력단 | 신규한 파에오놀-트립타민 화합물 및 그의 용도 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3133930A (en) * | 1961-08-15 | 1964-05-19 | Ciba Geigy Corp | Ester and amide derivatives of thieno-[3, 2-b] indole 3-carboxylic acids |
US4900748A (en) * | 1988-03-04 | 1990-02-13 | The United States Of America As Represented By The Department Of Health And Human Services | Carbamates related to (-)-physostigmine as cholinergic agents |
-
1992
- 1992-08-26 DE DE69233255T patent/DE69233255T2/de not_active Expired - Fee Related
- 1992-08-26 AT AT92919058T patent/ATE254916T1/de not_active IP Right Cessation
- 1992-08-26 DK DK92919058T patent/DK0605474T3/da active
- 1992-08-26 WO PCT/US1992/007085 patent/WO1993005779A1/en active IP Right Grant
- 1992-08-26 EP EP92919058A patent/EP0605474B1/en not_active Expired - Lifetime
- 1992-08-26 CA CA002119782A patent/CA2119782C/en not_active Expired - Fee Related
- 1992-08-26 JP JP50604593A patent/JP3193717B2/ja not_active Expired - Fee Related
- 1992-08-26 ES ES92919058T patent/ES2206449T3/es not_active Expired - Lifetime
- 1992-08-26 AU AU25042/92A patent/AU667318B2/en not_active Ceased
- 1992-08-28 EP EP02013799A patent/EP1251131A3/en not_active Withdrawn
-
1994
- 1994-01-18 US US08/182,301 patent/US5378723A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
CA2119782A1 (en) | 1993-04-01 |
DE69233255D1 (de) | 2004-01-08 |
EP1251131A3 (en) | 2002-10-30 |
ES2206449T3 (es) | 2004-05-16 |
EP0605474A4 (da) | 1994-08-03 |
EP1251131A2 (en) | 2002-10-23 |
JP3193717B2 (ja) | 2001-07-30 |
AU2504292A (en) | 1993-04-27 |
WO1993005779A1 (en) | 1993-04-01 |
DE69233255T2 (de) | 2004-05-27 |
ATE254916T1 (de) | 2003-12-15 |
CA2119782C (en) | 2005-08-23 |
EP0605474A1 (en) | 1994-07-13 |
EP0605474B1 (en) | 2003-11-26 |
AU667318B2 (en) | 1996-03-21 |
JPH07505120A (ja) | 1995-06-08 |
US5378723A (en) | 1995-01-03 |
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