DE69725153D1 - Kaliumkanal-blocker - Google Patents

Kaliumkanal-blocker

Info

Publication number
DE69725153D1
DE69725153D1 DE69725153T DE69725153T DE69725153D1 DE 69725153 D1 DE69725153 D1 DE 69725153D1 DE 69725153 T DE69725153 T DE 69725153T DE 69725153 T DE69725153 T DE 69725153T DE 69725153 D1 DE69725153 D1 DE 69725153D1
Authority
DE
Germany
Prior art keywords
potassium channel
channel blocker
treatment
cell proliferative
proliferative disorders
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69725153T
Other languages
English (en)
Other versions
DE69725153T2 (de
Inventor
Alexander Castle
Patrick Hollinshead
Floyd Hughes
Serafin Mendoza
Wendell Wilson
George Amato
Serge Beaudoin
Michael Gross
Grant Mcnaughton-Smith
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Icagen Inc
Original Assignee
Eli Lilly and Co
Icagen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co, Icagen Inc filed Critical Eli Lilly and Co
Publication of DE69725153D1 publication Critical patent/DE69725153D1/de
Application granted granted Critical
Publication of DE69725153T2 publication Critical patent/DE69725153T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/20—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Magnetic Heads (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Optical Communication System (AREA)
  • Separation By Low-Temperature Treatments (AREA)
  • Amplifiers (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE69725153T 1996-07-26 1997-07-23 Kaliumkanal-blocker Expired - Fee Related DE69725153T2 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US2254796P 1996-07-26 1996-07-26
US22547 1996-07-26
US08/893,160 US6083986A (en) 1996-07-26 1997-07-15 Potassium channel inhibitors
PCT/US1997/012559 WO1998004521A1 (en) 1996-07-26 1997-07-23 Potassium channel inhibitors
US893160 2001-06-27

Publications (2)

Publication Number Publication Date
DE69725153D1 true DE69725153D1 (de) 2003-10-30
DE69725153T2 DE69725153T2 (de) 2004-06-09

Family

ID=26696048

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69725153T Expired - Fee Related DE69725153T2 (de) 1996-07-26 1997-07-23 Kaliumkanal-blocker

Country Status (13)

Country Link
US (1) US6083986A (de)
EP (1) EP0923543B1 (de)
JP (1) JP2002513385A (de)
KR (1) KR20000029605A (de)
AT (1) ATE250571T1 (de)
AU (1) AU734711B2 (de)
BR (1) BR9710587A (de)
CA (1) CA2261814A1 (de)
DE (1) DE69725153T2 (de)
HK (1) HK1020334A1 (de)
HU (1) HUP0003250A3 (de)
IL (1) IL128205A (de)
WO (1) WO1998004521A1 (de)

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US6458794B2 (en) 1999-12-21 2002-10-01 Icagen, Inc. Potassium channel inhibitors
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DE10128331A1 (de) 2001-06-12 2002-12-19 Aventis Pharma Gmbh Anthranilsäureamide mit Heteroarylsulfonyl-Seitenkette, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltende pharmazeutische Zubereitungen
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NO3175985T3 (de) 2011-07-01 2018-04-28
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Also Published As

Publication number Publication date
EP0923543A1 (de) 1999-06-23
WO1998004521A1 (en) 1998-02-05
HUP0003250A1 (hu) 2002-01-28
JP2002513385A (ja) 2002-05-08
DE69725153T2 (de) 2004-06-09
IL128205A0 (en) 1999-11-30
BR9710587A (pt) 2000-10-31
EP0923543B1 (de) 2003-09-24
HUP0003250A3 (en) 2002-02-28
AU734711B2 (en) 2001-06-21
IL128205A (en) 2003-09-17
KR20000029605A (ko) 2000-05-25
ATE250571T1 (de) 2003-10-15
US6083986A (en) 2000-07-04
CA2261814A1 (en) 1998-02-05
AU3803597A (en) 1998-02-20
HK1020334A1 (en) 2000-04-14

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee