DE69418656D1 - 2-acyloxycephemderivate als elastaseinhibitoren - Google Patents

2-acyloxycephemderivate als elastaseinhibitoren

Info

Publication number
DE69418656D1
DE69418656D1 DE69418656T DE69418656T DE69418656D1 DE 69418656 D1 DE69418656 D1 DE 69418656D1 DE 69418656 T DE69418656 T DE 69418656T DE 69418656 T DE69418656 T DE 69418656T DE 69418656 D1 DE69418656 D1 DE 69418656D1
Authority
DE
Germany
Prior art keywords
elastas
acyloxycephemic
inhibitors
derivatives
elastas inhibitors
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69418656T
Other languages
English (en)
Other versions
DE69418656T2 (de
Inventor
Marco Alpegiani
Pierluigi Bissolino
Ettore Perrone
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Pharmacia and Upjohn SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn SpA filed Critical Pharmacia and Upjohn SpA
Application granted granted Critical
Publication of DE69418656D1 publication Critical patent/DE69418656D1/de
Publication of DE69418656T2 publication Critical patent/DE69418656T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DE69418656T 1993-03-04 1994-02-24 2-acyloxycephemderivate als elastaseinhibitoren Expired - Fee Related DE69418656T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB939304440A GB9304440D0 (en) 1993-03-04 1993-03-04 2-acyloxycephem derivatives
PCT/EP1994/000529 WO1994020504A1 (en) 1993-03-04 1994-02-24 2-acyloxycephem derivatives as elastase inhibitors

Publications (2)

Publication Number Publication Date
DE69418656D1 true DE69418656D1 (de) 1999-07-01
DE69418656T2 DE69418656T2 (de) 1999-12-30

Family

ID=10731476

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69418656T Expired - Fee Related DE69418656T2 (de) 1993-03-04 1994-02-24 2-acyloxycephemderivate als elastaseinhibitoren

Country Status (9)

Country Link
US (1) US5587373A (de)
EP (1) EP0639195B1 (de)
JP (1) JPH07506841A (de)
AU (1) AU671202B2 (de)
CA (1) CA2118422A1 (de)
DE (1) DE69418656T2 (de)
ES (1) ES2134345T3 (de)
GB (1) GB9304440D0 (de)
WO (1) WO1994020504A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9513818D0 (en) * 1995-07-06 1995-09-06 Pharmacia Spa 7,7-Disubstituted cephem-4-ketones
GB9525697D0 (en) * 1995-12-15 1996-02-14 Pharmacia Spa Cephem derivatives

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3578660A (en) * 1968-10-07 1971-05-11 Lilly Co Eli 2-acyloxycephalosporin compounds
US3852282A (en) * 1969-04-01 1974-12-03 Squibb & Sons Inc Certain 2-substituted cephalosporins
JPS5834184A (ja) * 1981-08-25 1983-02-28 Otsuka Chem Co Ltd 2−オキシセフアロスポリン誘導体の製造方法
GB8808701D0 (en) * 1988-04-13 1988-05-18 Erba Carlo Spa Beta-lactam derivatives
GB8928373D0 (en) * 1989-12-15 1990-02-21 Erba Carlo Spa Beta-lactam derivatives
GB9207715D0 (en) * 1992-04-08 1992-05-27 Erba Carlo Spa 2,2-disubstituted cephem sulphones

Also Published As

Publication number Publication date
AU6205594A (en) 1994-09-26
CA2118422A1 (en) 1994-09-15
GB9304440D0 (en) 1993-04-21
EP0639195A1 (de) 1995-02-22
AU671202B2 (en) 1996-08-15
DE69418656T2 (de) 1999-12-30
EP0639195B1 (de) 1999-05-26
ES2134345T3 (es) 1999-10-01
US5587373A (en) 1996-12-24
JPH07506841A (ja) 1995-07-27
WO1994020504A1 (en) 1994-09-15

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee