DE69307712D1 - Pyridopyrimidinone als wirkstoffe gegen angina - Google Patents

Pyridopyrimidinone als wirkstoffe gegen angina

Info

Publication number
DE69307712D1
DE69307712D1 DE69307712T DE69307712T DE69307712D1 DE 69307712 D1 DE69307712 D1 DE 69307712D1 DE 69307712 T DE69307712 T DE 69307712T DE 69307712 T DE69307712 T DE 69307712T DE 69307712 D1 DE69307712 D1 DE 69307712D1
Authority
DE
Germany
Prior art keywords
alkyl
pct
co2r9
onyl
morpholino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69307712T
Other languages
English (en)
Other versions
DE69307712T2 (de
Inventor
Andrew Simon Bell
Nicholas Kenneth Terrett
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Research and Development Co NV SA
Original Assignee
Pfizer Research and Development Co NV SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Research and Development Co NV SA filed Critical Pfizer Research and Development Co NV SA
Publication of DE69307712D1 publication Critical patent/DE69307712D1/de
Application granted granted Critical
Publication of DE69307712T2 publication Critical patent/DE69307712T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Liquid Crystal Substances (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Road Signs Or Road Markings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE69307712T 1992-08-28 1993-08-04 Pyridopyrimidinone als wirkstoffe gegen angina Expired - Fee Related DE69307712T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929218322A GB9218322D0 (en) 1992-08-28 1992-08-28 Therapeutic agents
PCT/EP1993/002097 WO1994005661A1 (en) 1992-08-28 1993-08-04 Pyridopyrimidinone antianginal agents

Publications (2)

Publication Number Publication Date
DE69307712D1 true DE69307712D1 (de) 1997-03-06
DE69307712T2 DE69307712T2 (de) 1997-05-15

Family

ID=10721102

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69307712T Expired - Fee Related DE69307712T2 (de) 1992-08-28 1993-08-04 Pyridopyrimidinone als wirkstoffe gegen angina

Country Status (12)

Country Link
US (1) US5591742A (de)
EP (1) EP0656898B1 (de)
JP (1) JP2660103B2 (de)
AT (1) ATE148118T1 (de)
CA (1) CA2138298C (de)
DE (1) DE69307712T2 (de)
DK (1) DK0656898T3 (de)
ES (1) ES2096936T3 (de)
FI (1) FI112484B (de)
GB (1) GB9218322D0 (de)
GR (1) GR3022852T3 (de)
WO (1) WO1994005661A1 (de)

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Also Published As

Publication number Publication date
ES2096936T3 (es) 1997-03-16
EP0656898A1 (de) 1995-06-14
FI950889A (fi) 1995-02-27
CA2138298A1 (en) 1994-03-17
DE69307712T2 (de) 1997-05-15
JP2660103B2 (ja) 1997-10-08
GR3022852T3 (en) 1997-06-30
EP0656898B1 (de) 1997-01-22
DK0656898T3 (da) 1997-08-18
US5591742A (en) 1997-01-07
ATE148118T1 (de) 1997-02-15
FI950889A0 (fi) 1995-02-27
JPH07506838A (ja) 1995-07-27
WO1994005661A1 (en) 1994-03-17
FI112484B (fi) 2003-12-15
CA2138298C (en) 1998-04-14
GB9218322D0 (en) 1992-10-14

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