DE69232406T2 - Verfahren zur Herstellung von Fluoro-Chinolin-3-Carbonsäurederivate - Google Patents

Verfahren zur Herstellung von Fluoro-Chinolin-3-Carbonsäurederivate

Info

Publication number: DE69232406T2
Authority: DE; Germany
Prior art keywords: preparation; acid derivatives; fluoro; quinoline; carboxylic acid
Prior art date: 1991-10-10
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Fee Related

Application number

DE69232406T

Other languages

English (en)

Other versions

DE69232406D1 (de

Inventor

Christophe Daubie

Jean-Jacques Legrand

Clive Pemberton

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Aventis Pharma SA

Original Assignee

Aventis Pharma SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-10-10

Filing date

1992-10-08

Publication date

2002-08-22

1992-10-08 Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA

2002-03-21 Publication of DE69232406D1 publication Critical patent/DE69232406D1/de

2002-08-22 Application granted granted Critical

2002-08-22 Publication of DE69232406T2 publication Critical patent/DE69232406T2/de

2012-10-09 Anticipated expiration legal-status Critical

Status Expired - Fee Related legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/44—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by —CHO groups
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Quinoline Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DE69232406T 1991-10-10 1992-10-08 Verfahren zur Herstellung von Fluoro-Chinolin-3-Carbonsäurederivate Expired - Fee Related DE69232406T2 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9112480A FR2682378B1 (fr)	1991-10-10	1991-10-10	Nouveaux derives de l'acide fluoroquinoleine carboxylique-3 et leur preparation.

Publications (2)

Publication Number	Publication Date
DE69232406D1 DE69232406D1 (de)	2002-03-21
DE69232406T2 true DE69232406T2 (de)	2002-08-22

Family

ID=9417775

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DE69232406T Expired - Fee Related DE69232406T2 (de)	1991-10-10	1992-10-08	Verfahren zur Herstellung von Fluoro-Chinolin-3-Carbonsäurederivate

Country Status (25)

Country	Link
US (1)	US5442070A (de)
EP (2)	EP0538100B1 (de)
JP (1)	JP3252852B2 (de)
KR (1)	KR100249637B1 (de)
AT (1)	ATE212982T1 (de)
AU (1)	AU672370B2 (de)
CA (1)	CA2119757C (de)
CZ (1)	CZ284595B6 (de)
DE (1)	DE69232406T2 (de)
DK (1)	DK0538100T3 (de)
ES (1)	ES2176185T3 (de)
FI (1)	FI105400B (de)
FR (1)	FR2682378B1 (de)
HU (1)	HU214955B (de)
IL (1)	IL103403A (de)
MX (1)	MX9205773A (de)
NO (1)	NO301640B1 (de)
NZ (1)	NZ244646A (de)
PT (1)	PT538100E (de)
RU (1)	RU2109014C1 (de)
SK (1)	SK280886B6 (de)
TW (1)	TW224093B (de)
WO (1)	WO1993007127A1 (de)
YU (1)	YU48443B (de)
ZA (1)	ZA927744B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2703681B1 (fr) *	1993-04-08	1995-05-12	Bellon Labor Sa Roger	Procede de preparation de fluoro-6-halogeno-2 quinoleine
WO2005026166A1 (fr) *	2003-09-16	2005-03-24	'chemical Diversity Research Institute', Ltd.	Composition physiologiquement active, composition pharmaceutique, 1,2-dihydro[2,7]naphtyridine, procedes de fabrication et application
MD2909C2 (ro) *	2005-01-14	2006-06-30	Николае ТАРАН	Procedeu de fabricare a vinurilor naturale cu zahăr rezidual

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1458205A (en) *	1973-04-13	1976-12-08	Pfizer	Fused pyrimidin-4- 3h-ones as antiallergy agents
FR2593961B1 (fr) *	1986-02-04	1988-04-15	Orega Electro Mecanique	Transformateur haute tension en technologie fractionnee, en particulier pour tube cathodique trichrome
DK111387A (da) *	1986-03-05	1987-09-06	Otsuka Pharma Co Ltd	Carbostyrilderivater og salte deraf, laegemiddel indeholdende saadanne derivater samt fremgangsmaade til fremstilling af derivaterne
US4909829A (en) *	1987-12-29	1990-03-20	Fmc Corporation	Substituted quinolinonyl and dihydroquinolinonyl tetrazolinone herbicides
US4894084A (en) *	1987-12-29	1990-01-16	Fmc Corporation	Substituted quinolinonyl and dihydroquinolinonyl triazolinone herbicides
NZ232090A (en) *	1989-01-16	1990-12-21	Bellon Labor Sa Roger	Halogen-containing 1-substituted-4-oxo-1,4-dihydro-benzo(b)(1,8)naphthyridine-3-carboxylic acid derivatives, preparation and pharmaceutical compositions thereof
NZ232092A (en) *	1989-01-16	1992-05-26	Bellon Labor Sa Roger	8-halo-7-fluoro-4-oxo-1,4-dihydro-benzo(b)(1,8) naphthyridine-3-carboxylic acid esters and preparation thereof
AU623474B2 (en) *	1989-01-16	1992-05-14	Laboratoire Roger Bellon	New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them
US5385913A (en) *	1989-10-06	1995-01-31	Pfizer Inc.	1,4-dihydro-4-oxo-3-quinoline derivatives as selectively toxic mammalian antibacterial agents

1991
- 1991-10-10 FR FR9112480A patent/FR2682378B1/fr not_active Expired - Fee Related
1992
- 1992-10-07 NZ NZ244646A patent/NZ244646A/en not_active IP Right Cessation
- 1992-10-08 PT PT92402742T patent/PT538100E/pt unknown
- 1992-10-08 AT AT92402742T patent/ATE212982T1/de not_active IP Right Cessation
- 1992-10-08 DE DE69232406T patent/DE69232406T2/de not_active Expired - Fee Related
- 1992-10-08 JP JP50667593A patent/JP3252852B2/ja not_active Expired - Fee Related
- 1992-10-08 CZ CS94833A patent/CZ284595B6/cs not_active IP Right Cessation
- 1992-10-08 AU AU28744/92A patent/AU672370B2/en not_active Ceased
- 1992-10-08 SK SK403-94A patent/SK280886B6/sk unknown
- 1992-10-08 RU RU94022265/04A patent/RU2109014C1/ru not_active IP Right Cessation
- 1992-10-08 CA CA002119757A patent/CA2119757C/fr not_active Expired - Fee Related
- 1992-10-08 ES ES92402742T patent/ES2176185T3/es not_active Expired - Lifetime
- 1992-10-08 TW TW081107996A patent/TW224093B/zh active
- 1992-10-08 KR KR1019940701166A patent/KR100249637B1/ko not_active IP Right Cessation
- 1992-10-08 HU HU9401004A patent/HU214955B/hu not_active IP Right Cessation
- 1992-10-08 EP EP92402742A patent/EP0538100B1/de not_active Expired - Lifetime
- 1992-10-08 ZA ZA927744A patent/ZA927744B/xx unknown
- 1992-10-08 US US08/211,325 patent/US5442070A/en not_active Expired - Lifetime
- 1992-10-08 WO PCT/FR1992/000936 patent/WO1993007127A1/fr active IP Right Grant
- 1992-10-08 EP EP92922225A patent/EP0607329A1/de active Pending
- 1992-10-08 MX MX9205773A patent/MX9205773A/es not_active IP Right Cessation
- 1992-10-08 DK DK92402742T patent/DK0538100T3/da active
- 1992-10-09 YU YU91192A patent/YU48443B/sh unknown
- 1992-10-09 IL IL10340392A patent/IL103403A/en not_active IP Right Cessation
1994
- 1994-04-06 NO NO941244A patent/NO301640B1/no unknown
- 1994-04-08 FI FI941650A patent/FI105400B/fi active

Also Published As

Publication number	Publication date
CZ83394A3 (en)	1995-02-15
IL103403A0 (en)	1993-03-15
RU2109014C1 (ru)	1998-04-20
NZ244646A (en)	1994-04-27
DE69232406D1 (de)	2002-03-21
FI105400B (fi)	2000-08-15
FR2682378B1 (fr)	1995-04-07
HUT67486A (en)	1995-04-28
DK0538100T3 (da)	2002-04-29
EP0607329A1 (de)	1994-07-27
YU48443B (sh)	1998-07-10
YU91192A (sh)	1995-03-27
WO1993007127A1 (fr)	1993-04-15
EP0538100B1 (de)	2002-02-06
CA2119757A1 (fr)	1993-04-15
FR2682378A1 (fr)	1993-04-16
SK40394A3 (en)	1995-02-08
JPH07500101A (ja)	1995-01-05
KR940702846A (ko)	1994-09-17
CZ284595B6 (cs)	1999-01-13
AU2874492A (en)	1993-05-03
AU672370B2 (en)	1996-10-03
NO301640B1 (no)	1997-11-24
FI941650A0 (fi)	1994-04-08
HU9401004D0 (en)	1994-08-29
IL103403A (en)	1996-10-16
NO941244D0 (no)	1994-04-06
TW224093B (de)	1994-05-21
CA2119757C (fr)	2005-09-20
MX9205773A (es)	1993-04-01
KR100249637B1 (ko)	2000-04-01
ATE212982T1 (de)	2002-02-15
JP3252852B2 (ja)	2002-02-04
HU214955B (hu)	1998-08-28
ZA927744B (en)	1993-04-19
FI941650A (fi)	1994-04-08
US5442070A (en)	1995-08-15
PT538100E (pt)	2002-07-31
ES2176185T3 (es)	2002-12-01
SK280886B6 (sk)	2000-09-12
NO941244L (no)	1994-05-24
EP0538100A1 (de)	1993-04-21

Legal Events

Date	Code	Title	Description
2003-03-06	8364	No opposition during term of opposition
2006-10-26	8328	Change in the person/name/address of the agent	Representative=s name: PFENNING MEINIG & PARTNER GBR, 80339 MUENCHEN
2009-07-30	8328	Change in the person/name/address of the agent	Representative=s name: MAIWALD PATENTANWALTSGESELLSCHAFT MBH, 80335 MUENC
2009-08-20	8339	Ceased/non-payment of the annual fee

Publication	Publication Date	Title
DE69013607D1 (de)	1994-12-01	Pyrazol-Derivate, Verfahren zu deren Herstellung und Anwendung.
DE69207194T2 (de)	1996-09-05	Verfahren zur Herstellung von Bacchatin III und von Desacetyl-10-Bacchatin III Derivate
ATE166357T1 (de)	1998-06-15	Galakturonsäurederivate, verfahren zur ihrer herstellung und ihre verwendung
DE69232406D1 (de)	2002-03-21	Verfahren zur Herstellung von Fluoro-Chinolin-3-Carbonsäurederivate
ATE115567T1 (de)	1994-12-15	Verfahren zur herstellung von halogensulfonyl- substituierten pyridinen.
ATE150453T1 (de)	1997-04-15	Verfahren zur herstellung von trans-piperidin-2,5-dicarboxylaten
DE69119714D1 (de)	1996-06-27	Verfahren zur Herstellung von Benzylphthalazinonderivaten und von deren Salzen
ATE23993T1 (de)	1986-12-15	Verfahren zur herstellung von o,o'dithiobenzamiden.
ATE82747T1 (de)	1992-12-15	Verfahren zur herstellung von hydroxyalkylierungsmitteln, die erhaltenen mittel und deren verwendung.
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DE68910931D1 (de)	1994-01-05	Verfahren zur Herstellung von Propionsäurederivaten.
ATE29253T1 (de)	1987-09-15	Verfahren zur herstellung von 4-chinolinonen.
DE59202229D1 (de)	1995-06-22	Verfahren zur Herstellung substituierter Indole.
ATE24899T1 (de)	1987-01-15	Verfahren zur herstellung von 4-quinolinonen.
ATE144255T1 (de)	1996-11-15	Verfahren zur herstellung von pyridazinonderivaten
DE59900666D1 (de)	2002-02-21	Verfahren zur Herstellung von Malonsäuredinitril
DE3853110D1 (de)	1995-04-06	Verfahren zur Herstellung von 4-Alkoxyalkyl-beta-carbolinen.
FI953246A (fi)	1995-06-30	Välituotteet kinoliini-3-karboksyylihappojohdannaisten valmistamiseksi